Name: Lidocaine N-ethyl bromide
SKU: A22615
Price: 320 USD
Rating: 5 (288 reviews)

Catalog No.

Product Name

Application

Product Information

Product Citation

A12185

Nav1.7-IN-2

Nav inhibitor

Nav1.7-IN-2 is an inhibitor of voltage-gated sodium channels (Nav), in particular Nav 1.7, with IC50 of 80 nM.

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A13626

Nav1.7-IN-3

voltage-gated sodium channel Nav1.7 inhibitor

Nav1.7-IN-3 is a selective, orally bioavailable voltage-gated sodium channel Nav1.7 inhibitor with an IC50 of 8 nM. Pain relief. Limited CNS penetration.

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A19046

GNE-616

Nav1.7 inhibitor

GNE-616 is a highly potent, metabolically stable, orally bioavailable, and subtype selective Nav1.7 inhibitor (Ki of 0.79 nM and Kd of 0.38 nM for hNav1.7) for the treatment of chronic pain.

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A19138

GNE-0439

Nav1.7-selective inhibitor

GNE-0439 is a novel Nav1.7-selective inhibitor with IC50 of 0.34 uM and inhibits Nav1.5 with an IC50 of 38.3 μM.

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A21141

Nav1.7 inhibitor

Nav1.7 inhibitor

Nav1.7 inhibitor is a potent Nav1.7 inhibitor.

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A21298

Funapide

Sodium Channel Nav1.7 inhibitor

Funapide (TV 45070; XEN402) is a potent Sodium Channel Nav1.7 inhibitor.

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A22002

Ralfinamide mesylate

Na+ channel blocker

Ralfinamide mesylate (FCE-26742A mesylate) is an orally available Na+ channel blocker derived from α-aminoamide, with function of suppressing pain.

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A22615

Lidocaine N-ethyl bromide

blocker of fast Na+-dependent action potentials and voltage-dependent

Lidocaine N-ethyl bromide is a non-membrane-permeable blocker of fast Na+-dependent action potentials and voltage-dependent, non-inactivating Na+ conductance.

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Sodium Channels