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GRK

Catalog No.

Product Name

Application

Product Information

Product Citation

A19795

CMPD101

GRK2/GRK3 inhibitor

CMPD101, is a novel membrane-permeable, small-molecule inhibitor of both GRK2 and GRK3 with IC50s of 18 nM and 5.4 nM. CMPD101 also inhibits ROCK-2 and PKCα (IC50s=1.4 μM and 8.1 μM, respectively).

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A20736

GSK180736A

GRK2 inhibitor

GSK180736A is a G protein-coupled receptor kinase 2 (GRK2) inhibitor with an IC50 of 0.77 μM.

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