Estrogen Receptors

Toremifene citrate (Z-Toremifene citrate) is a second-generation selective estrogen-receptor modulator (SERM) in development for the prevention of osteoporosis. Toremifene citrate also potent inhibits infectious EBOV Zaire and Marburg (MARV) with IC50 of 0.07 ?M and 2.6 ?M, respectively.

Ospemifene is a non-hormonal selective estrogen receptor modulator (SERM).

Bazedoxifene is a third generation selective modulator of estrogen receptor.

Toremifene is a second-generation selective estrogen-receptor modulator (SERM) in development for the prevention of osteoporosis.

Tamoxifen (ICI 47699) is a selective estrogen receptor modulator (SERM) which blocks estrogen action in breast cells and can activate estrogen activity in other cells, such as bone, liver, and uterine cells.

Lasofoxifene tartrate is a third-generation selective estrogen receptor modulator.

4-Hydroxytamoxifen is a selective estrogen receptor modulator (SERM).