Glucocorticoid receptors
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Fluorometholone
Catalog No. A17651 glucocorticoidFluorometholone is a glucocorticoid employed, usually as eye drops, in the treatment of allergic and inflammatory conditions of the eye. It has also been used topically in the treatment of various skin disorders. Learn More -
Mapracorat
Catalog No. A21953 glucocorticoid receptor agonistMapracorat is a novel non-steroidal selective glucocorticoid receptor agonist. Learn More -
(S)-Mapracorat
Catalog No. A21528 glucocorticoid receptor agonist(S)-Mapracorat is a selective and less active glucocorticoid receptor agonist. Learn More -
Dagrocorat
Catalog No. A21312 glucocorticoid receptor agonistDagrocorat (PF-00251802) is a novel and dissociated glucocorticoid receptor agonist. Learn More -
Fosdagrocorat
Catalog No. A21303 dissociated glucocorticoid receptor agonistFosdagrocorat (PF-04171327) is a dissociated glucocorticoid receptor agonist. Learn More -
Beclometasone dipropionate
Catalog No. A17254 glucocorticoid agonistBeclometasone dipropionate is a potent glucocorticoid agonist; it is a prodrug of the free form, beclometasone. Learn More -
Dexamethasone acetate
Catalog No. A16494 glucocorticoid receptor agonistDexamethasone acetate (Dexamethasone 21-acetate) is a glucocorticoid receptor agonist. Learn More -
Glucocorticoid receptor agonist
Catalog No. A11431 Glucocorticoid receptor agonistGlucocorticoid receptor agonist is a potent Glucocorticoid receptor agonist. Learn More -
Betamethasone acibutate
Catalog No. A18697 glucocorticoidBetamethasone acibutate, derives from Betamethasone, is an acetate ester. Betamethasone acibutate is a glucocorticoid. Learn More -
AZD2906
Catalog No. A18936 glucocorticoid receptor agonistAZD2906 is a selective glucocorticoid receptor (GR) agonist, increases micronucleated immature erythrocytes in the bone marrow of rats. AZD2906 shows IC50s of 2.2, 0.3, 41.6 and 7.5 nM at GR in human, rat PBMC and human, rat whole blood, respectively. Learn More -
AZD5423
Catalog No. A13249 nonsteroidal glucocorticoid receptor agonistAZD5423 is a novel nonsteroidal glucocorticoid receptor agonist. Learn More -
RU43044
Catalog No. A14340 Glucocorticoid receptor antagonistThe antiglucocorticoid RU43044 exerted significant agonist activity and activated MMTV-Luc transcription in osteosarcoma cells but not human breast cancer cells. Learn More -
GW-870086
Catalog No. A18343 Glucocorticoid receptor agonistGW-870086 is a potent anti-inflammatory agent, acting as a glucocorticoid receptor agonist, with a pIC50 of 10.1 in A549 cells expressing NF-κB. Learn More -
Betamethasone dipropionate
Catalog No. A10130 Glucocorticoid Receptor AgonistBetamethasone dipropionate is a glucocorticoid steroid with anti-inflammatory and immunosuppressive abilities. Learn More -
Beclometasone
Catalog No. A18177 glucocorticoid receptor agonistBeclometasone, also known as Beclomethasone, is an anti-inflammatory, synthetic glucocorticoid. It is used topically as an anti-inflammatory agent and in aerosol form for the treatment of asthma. Learn More -
AZD9567
Catalog No. A18850 selective glucocorticoid receptor modulatorAZD9567 is a potent, oral active, non-steroidal and selective glucocorticoid receptor modulator (SGRM), with an IC50 of 3.8 nM. Learn More -
OP-3633
Catalog No. A18468 Glucocorticoid Receptor AntagonistOP-3633 is a Potent Steroidal Glucocorticoid Receptor Antagonist with Enhanced Selectivity against the Progesterone and Androgen Receptors (IC50 = 29 nM). Learn More -
Fluticasone propionate
Catalog No. A11860 Fluticasone propionate is a high affinity, selective glucocorticoid receptor agonist (Kd = 0.5 nM). Learn More -
Prednisone (Adasone)
Catalog No. A10752 Glucocorticoid Receptor agonistPrednisone reduces mucosal TNF-a production, intestinal permeability and levels of NF-kB expression. Learn More -
Methylprednisolone
Catalog No. A10582 Methylprednisolone is an apoptosis inducer and was also found to inhibit human small cell lung cancer cell growth in vitro. Learn More -
Meprednisone (Betapar)
Catalog No. A10567 Meprednisone is a glucocorticoid and a methylated derivative of prednisone Learn More -
Hydrocortisone(Cortisol)
Catalog No. A10457 Hydrocortisone is a steroid hormone or glucocorticoid produced by the adrenal gland. Learn More -
Deflazacort
Catalog No. A10294 Deflazacort is a glucocorticoid used as an anti-inflammatory and immunosuppressant. Learn More -
Prednisolone acetate (Omnipred)
Catalog No. A11687 Prednisolone is a synthetic glucocorticoid, a derivative of cortisol, which is used to treat a variety of inflammatory and auto-immune conditions. Learn More -
Budesonide
Catalog No. A10166 Budesonide is a glucocorticoid steroid for the treatment of asthma, non-infectious rhinitis. Learn More -
Betamethasone valerate (Betnovate, Celestone)
Catalog No. A10131 Betamethasone valerate is a potent glucocorticoid steroid with anti-inflammatory and immunosuppressive properties. Learn More