Glucocorticoid receptors

16 Item(s)

per page

Set Descending Direction
  1. Betamethasone dipropionate

    Catalog No. A10130
    Quick View
    Glucocorticoid Receptor Agonist
    Betamethasone dipropionate is a glucocorticoid steroid with anti-inflammatory and immunosuppressive abilities. Learn More
  2. Exicorilant

    Catalog No. A18620
    Quick View
    Glucocorticoid receptor (GR) antagonist
    Exicorilant (CORT 125281) is a selective and oral active glucocorticoid receptor (GR) antagonist, with a Ki value of 7 nM. Exicorilant (CORT 125281) has potential to overcome adiposity, glucose intolerance and dyslipidaemia. Learn More
  3. AZD9567

    Catalog No. A18850
    Quick View
    selective glucocorticoid receptor modulator
    AZD9567 is a potent, oral active, non-steroidal and selective glucocorticoid receptor modulator (SGRM), with an IC50 of 3.8 nM. Learn More
  4. Beclometasone

    Catalog No. A18177
    Quick View
    glucocorticoid receptor agonist
    Beclometasone, also known as Beclomethasone, is an anti-inflammatory, synthetic glucocorticoid. It is used topically as an anti-inflammatory agent and in aerosol form for the treatment of asthma. Learn More
  5. GW-870086

    Catalog No. A18343
    Quick View
    Glucocorticoid receptor agonist
    GW-870086 is a potent anti-inflammatory agent, acting as a glucocorticoid receptor agonist, with a pIC50 of 10.1 in A549 cells expressing NF-κB. Learn More
  6. RU43044

    Catalog No. A14340
    Glucocorticoid receptor antagonist
    The antiglucocorticoid RU43044 exerted significant agonist activity and activated MMTV-Luc transcription in osteosarcoma cells but not human breast cancer cells. Learn More
  7. Fluticasone propionate

    Catalog No. A11860
    Quick View
    Fluticasone propionate is a high affinity, selective glucocorticoid receptor agonist (Kd = 0.5 nM). Learn More
  8. Prednisone (Adasone)

    Catalog No. A10752
    Quick View
    Glucocorticoid Receptor agonist
    Prednisone reduces mucosal TNF-a production, intestinal permeability and levels of NF-kB expression. Learn More
  9. Methylprednisolone

    Catalog No. A10582
    Quick View
    Methylprednisolone is an apoptosis inducer and was also found to inhibit human small cell lung cancer cell growth in vitro. Learn More
  10. Meprednisone (Betapar)

    Catalog No. A10567
    Quick View
    Meprednisone is a glucocorticoid and a methylated derivative of prednisone Learn More
  11. Hydrocortisone(Cortisol)

    Catalog No. A10457
    Quick View
    Hydrocortisone is a steroid hormone or glucocorticoid produced by the adrenal gland. Learn More
  12. Deflazacort

    Catalog No. A10294
    Quick View
    Deflazacort is a glucocorticoid used as an anti-inflammatory and immunosuppressant. Learn More
  13. Prednisolone acetate (Omnipred)

    Catalog No. A11687
    Quick View
    Prednisolone is a synthetic glucocorticoid, a derivative of cortisol, which is used to treat a variety of inflammatory and auto-immune conditions. Learn More
  14. Budesonide

    Catalog No. A10166
    Quick View
    Budesonide is a glucocorticoid steroid for the treatment of asthma, non-infectious rhinitis. Learn More
  15. Betamethasone valerate (Betnovate, Celestone)

    Catalog No. A10131
    Quick View
    Betamethasone valerate is a potent glucocorticoid steroid with anti-inflammatory and immunosuppressive properties. Learn More
  16. OP-3633

    Catalog No. A18468
    Quick View
    Glucocorticoid Receptor Antagonist
    OP-3633 is a Potent Steroidal Glucocorticoid Receptor Antagonist with Enhanced Selectivity against the Progesterone and Androgen Receptors (IC50 = 29 nM). Learn More

16 Item(s)

per page

Set Descending Direction