Glucocorticoid receptors

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  1. Mapracorat

    Catalog No. A21953
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    glucocorticoid receptor agonist
    Mapracorat is a novel non-steroidal selective glucocorticoid receptor agonist. Learn More
  2. AZD2906

    Catalog No. A18936
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    glucocorticoid receptor agonist
    AZD2906 is a selective glucocorticoid receptor (GR) agonist, increases micronucleated immature erythrocytes in the bone marrow of rats. AZD2906 shows IC50s of 2.2, 0.3, 41.6 and 7.5 nM at GR in human, rat PBMC and human, rat whole blood, respectively. Learn More
  3. Betamethasone acibutate

    Catalog No. A18697
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    glucocorticoid
    Betamethasone acibutate, derives from Betamethasone, is an acetate ester. Betamethasone acibutate is a glucocorticoid. Learn More
  4. Glucocorticoid receptor agonist

    Catalog No. A11431
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    Glucocorticoid receptor agonist
    Glucocorticoid receptor agonist is a potent Glucocorticoid receptor agonist. Learn More
  5. Dexamethasone acetate

    Catalog No. A16494
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    glucocorticoid receptor agonist
    Dexamethasone acetate (Dexamethasone 21-acetate) is a glucocorticoid receptor agonist. Learn More
  6. Beclometasone dipropionate

    Catalog No. A17254
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    glucocorticoid agonist
    Beclometasone dipropionate is a potent glucocorticoid agonist; it is a prodrug of the free form, beclometasone. Learn More
  7. Fosdagrocorat

    Catalog No. A21303
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    dissociated glucocorticoid receptor agonist
    Fosdagrocorat (PF-04171327) is a dissociated glucocorticoid receptor agonist. Learn More
  8. Dagrocorat

    Catalog No. A21312
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    glucocorticoid receptor agonist
    Dagrocorat (PF-00251802) is a novel and dissociated glucocorticoid receptor agonist. Learn More
  9. (S)-Mapracorat

    Catalog No. A21528
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    glucocorticoid receptor agonist
    (S)-Mapracorat is a selective and less active glucocorticoid receptor agonist. Learn More
  10. Fluorometholone

    Catalog No. A17651
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    glucocorticoid
    Fluorometholone is a glucocorticoid employed, usually as eye drops, in the treatment of allergic and inflammatory conditions of the eye. It has also been used topically in the treatment of various skin disorders. Learn More
  11. AZD5423

    Catalog No. A13249
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    nonsteroidal glucocorticoid receptor agonist
    AZD5423 is a novel nonsteroidal glucocorticoid receptor agonist. Learn More
  12. RU43044

    Catalog No. A14340
    Glucocorticoid receptor antagonist
    The antiglucocorticoid RU43044 exerted significant agonist activity and activated MMTV-Luc transcription in osteosarcoma cells but not human breast cancer cells. Learn More
  13. Betamethasone valerate (Betnovate, Celestone)

    Catalog No. A10131
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    Betamethasone valerate is a potent glucocorticoid steroid with anti-inflammatory and immunosuppressive properties. Learn More
  14. Budesonide

    Catalog No. A10166
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    Budesonide is a glucocorticoid steroid for the treatment of asthma, non-infectious rhinitis. Learn More
  15. Prednisolone acetate (Omnipred)

    Catalog No. A11687
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    Prednisolone is a synthetic glucocorticoid, a derivative of cortisol, which is used to treat a variety of inflammatory and auto-immune conditions. Learn More
  16. Deflazacort

    Catalog No. A10294
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    Deflazacort is a glucocorticoid used as an anti-inflammatory and immunosuppressant. Learn More
  17. Hydrocortisone(Cortisol)

    Catalog No. A10457
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    Hydrocortisone is a steroid hormone or glucocorticoid produced by the adrenal gland. Learn More
  18. Meprednisone (Betapar)

    Catalog No. A10567
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    Meprednisone is a glucocorticoid and a methylated derivative of prednisone Learn More
  19. Methylprednisolone

    Catalog No. A10582
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    Methylprednisolone is an apoptosis inducer and was also found to inhibit human small cell lung cancer cell growth in vitro. Learn More
  20. Prednisone (Adasone)

    Catalog No. A10752
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    Glucocorticoid Receptor agonist
    Prednisone reduces mucosal TNF-a production, intestinal permeability and levels of NF-kB expression. Learn More
  21. OP-3633

    Catalog No. A18468
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    Glucocorticoid Receptor Antagonist
    OP-3633 is a Potent Steroidal Glucocorticoid Receptor Antagonist with Enhanced Selectivity against the Progesterone and Androgen Receptors (IC50 = 29 nM). Learn More
  22. Exicorilant

    Catalog No. A18620
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    Glucocorticoid receptor (GR) antagonist
    Exicorilant (CORT 125281) is a selective and oral active glucocorticoid receptor (GR) antagonist, with a Ki value of 7 nM. Exicorilant (CORT 125281) has potential to overcome adiposity, glucose intolerance and dyslipidaemia. Learn More
  23. AZD9567

    Catalog No. A18850
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    selective glucocorticoid receptor modulator
    AZD9567 is a potent, oral active, non-steroidal and selective glucocorticoid receptor modulator (SGRM), with an IC50 of 3.8 nM. Learn More
  24. Beclometasone

    Catalog No. A18177
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    glucocorticoid receptor agonist
    Beclometasone, also known as Beclomethasone, is an anti-inflammatory, synthetic glucocorticoid. It is used topically as an anti-inflammatory agent and in aerosol form for the treatment of asthma. Learn More
  25. Fluticasone propionate

    Catalog No. A11860
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    Fluticasone propionate is a high affinity, selective glucocorticoid receptor agonist (Kd = 0.5 nM). Learn More
  26. GW-870086

    Catalog No. A18343
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    Glucocorticoid receptor agonist
    GW-870086 is a potent anti-inflammatory agent, acting as a glucocorticoid receptor agonist, with a pIC50 of 10.1 in A549 cells expressing NF-κB. Learn More
  27. Betamethasone dipropionate

    Catalog No. A10130
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    Glucocorticoid Receptor Agonist
    Betamethasone dipropionate is a glucocorticoid steroid with anti-inflammatory and immunosuppressive abilities. Learn More

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