CETP

Catalog No.Inhibitor Name CETP
A11084Anacetrapib (MK-0859)
***
A11242Torcetrapib (CP-529414)
**
A11213JTT-705 (Dalcetrapib)
*
A11397Evacetrapib (LY2484595)
****

Notes:
1.Hover mouse over " * " to view the IC50 value.(A few compounds have proven potency but without published IC50 data.)
2.For more details about the compound, click on the product name of your interest.
3.The higher the number of " * " is, the more potent the inhibitor or activator is.
4."" refers to compounds which do inhibitory effects on the related isoform, but without specific value.

4 Item(s)

per page

Set Descending Direction
  1. Anacetrapib (MK-0859)

    Catalog No. A11084
    Quick View
    CETP inhibitor
    Anacetrapib (MK-0859) is a CETP inhibitor being developed to treat hypercholesterolemia (elevated cholesterol levels) and prevent cardiovascular disease. Learn More
  2. JTT-705 (Dalcetrapib)

    Catalog No. A11213
    Quick View
    CETP inhibitor
    JTT-705 (Dalcetrapib) is a CETP inhibitor.Inhibition of CETP is a target to increase HDL-cholesterol and potentially reduce atherosclerosis. Learn More
  3. Torcetrapib (CP-529414)

    Catalog No. A11242
    Quick View
    CETP inhibitor
    Torcetrapib (CP-529414) is a CETP inhibitor with IC50 of 37 nM. Learn More
  4. Evacetrapib (LY2484595)

    Catalog No. A11397
    Quick View
    CETP inhibitor
    Evacetrapib (LY2484595) is a potent and selective inhibitor of CETP with IC50 of 5.5 nM, elevates HDL cholesterol without increases in aldosterone or blood pressure. Phase 3. Learn More

4 Item(s)

per page

Set Descending Direction
Rewards