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GPR35 agonist 1
Catalog No. A12462 GPR35/CXCR8 agonistGPR35 agonist 1 (compound 50) is a potent and specific G protein-coupled receptor-35 (GPR35)/CXCR8 agonist with an EC50 of 5.8 nM, displays good druggability. Learn More -
AMG 837
Catalog No. A21160 GPR40 agonistAMG 837 is a potent GPR40 agonist(EC50=13 nM) with a superior pharmacokinetic profile and robust glucose-dependent stimulation of insulin secretion in rodents. Learn More -
MK-0354
Catalog No. A22008 GPR109a receptor agonistMK-0354 is a partial agonist of GPR109a receptor, for hGPR109a/ mGPR109a with EC50 of 1.65/1.08 μM, showed no activation of GPR109b. Learn More -
AMG 837 sodium salt
Catalog No. A21793 GPR40 agonistAMG 837 sodium salt is a potent GPR40 agonist(EC50=13 nM) with a superior pharmacokinetic profile and robust glucose-dependent stimulation of insulin secretion in rodents. Learn More -
AM-4668
Catalog No. A21778 GPR40 agonistAM-4668 is a GPR40 agonist for type 2 diabetes. EC50s of 3.6 nM and 36 nM for GPR40 in A9 cells (GPR40 IP3 assay) and CHO cells (GPR40 aequorin assay), respectively. Learn More -
(1R,2R)-2-PCCA(hydrochloride)
Catalog No. A21655 GPR88 receptor agonist(1R,2R)-2-PCCA hydrochloride is a diastereomer of 2-PCCA, and acts as a potent GPR88 receptor agonist, with an EC50 of 3 nM in cell-free assay, and 603 nM in cell assay. Learn More -
GPR40 Activator 2
Catalog No. A21642 GPR40 activatorGPR40 Activator 2 is a potent GPR40 activator from patents WO 2012147516 A1, WO 2012046869A1 and WO 2011078371 A1. Learn More -
AF64394
Catalog No. A21574 GPR3 inverse agonistAF64394 is a GPR3 inverse agonist, with a pIC50 of 7.3. Learn More -
AM-1638
Catalog No. A21505 GPR40/FFA1 full agonistAM-1638 is a potent and orally bioavailable GPR40/FFA1 full agonist with an EC50 of 0.16 μM. Learn More -
GLPG0974
Catalog No. A21466 FFA2/GPR43 antagonistGLPG0974 is a free fatty acid receptor-2 (FFA2/GPR43) antagonist with an IC50 of 9 nM. Learn More -
GPR40 Activator 1
Catalog No. A21154 GPR40 activatorGPR40 Activator 1 is a potent GPR40 activator for treatment of type 2 diabetes. Learn More -
PSN632408
Catalog No. A20902 GPR119 receptors agonistPSN632408 is an optimized agonist of GPR119 receptors that shows similar potency to OEA at both recombinant mouse and human GPR119 receptors, exhibiting EC50 values of 5.6 and 7.9 uM, respectively. Learn More -
Kynurenic acid sodium
Catalog No. A20000 GPR35/CXCR8 agonistKynurenic acid sodium, an endogenous tryptophan metabolite, is a broad-spectrum antagonist targeting NMDA, glutamate, α7 nicotinic acetylcholine receptor. Kynurenic acid sodium is also an agonist of GPR35/CXCR8. Learn More -
LY2922470
Catalog No. A12181 GPR40 agonistLY2922470 is a potent, selective and orally available agonist of the G protein-coupled receptor 40 (GPR40), with EC50s of 7 nM, 1 nM and 3 nM for human GPR40, mouse GPR40 and rat GPR40, respectively. Learn More -
G15
Catalog No. A13675 GPER/GPR30 antagonistG15 is a high affinity and selective G-protein-coupled estrogen receptor (GPER/GPR30) antagonist with a Ki of 20 nM. Learn More -
GPR4 antagonist 1
Catalog No. A12340 GPR4 antagonistGPR4 antagonist 1 is a GPR4 antagonist, with an IC50 of 189 nM. Learn More -
DJ-V-159
Catalog No. A18853 GPRC6A agonistDJ-V-159 is an agonist for G protein-coupled receptor family C group 6 member A (GPRC6A). Learn More -
GW-1100
Catalog No. A11445 GPR40 antagonistGW-1100 is a selective GPR40 antagonist with a pIC50 of 6.9. Learn More -
Kynurenic acid
Catalog No. A16581 GPR35/CXCR8 agonistKynurenic acid, an endogenous tryptophan metabolite, is a broad-spectrum antagonist targeting NMDA, glutamate, α7 nicotinic acetylcholine receptor. Kynurenic acid is also an agonist of GPR35/CXCR8. Learn More -
QS 11
Catalog No. A11228 ATPase and GTPase inhibitorQS-11 is a GTPase activating protein of ADP-ribosylation factor 1 (ARFGAP1) inhibitor. Learn More -
TM N1324
Catalog No. A17038 GPR39 agonistTM N1324 is an agonist of G-Protein-Coupled Receptor 39 (GPR39) with EC50s of 9 nM/5 nM in the presence of Zn2+, and 280 nM/180 nM in the absence of Zn2+ for human/murine GPR39. Learn More -
CID16020046
Catalog No. A16818 GPR55 antagonistCID16020046 is a selective GPR55 antagonist, inhibiting GPR55 constitutive activity with IC50 of 0.15 μM in yeast. It demonstrates weak activity against a broad spectrum of other GPCRs, ion channels, kinases, and nuclear receptor. Learn More -
MK-6892
Catalog No. A12982 GPR109A agonistMK-6892 is a potent, selective, and full agonist for the high affinity nicotinic acid (NA) receptor GPR109A.K i and GTPγS EC 50 of MK-6892 on the Human GPR109A is 4 nM and 16 nM, respectively. Learn More -
CCG 50014
Catalog No. A16432 RGS4 inhibitorCCG 50014 is a potent and selective inhibitor of RGS4 with IC50 of 30 nM. Learn More -
CASIN
Catalog No. A12912 Cdc42 GTPase inhibitorCASIN is a novel and potent Cdc42 inhibitor. Learn More -
CCG-63802
Catalog No. A11373 CCG-63802 is a reversible inhibitor of regulator of G-protein signaling (RGS) proteins. Selective amongst RGS proteins, with greatest potency at RGS4. Learn More
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