G Protein

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  1. QS 11

    Catalog No. A11228
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    ATPase and GTPase inhibitor
    QS-11 is a GTPase activating protein of ADP-ribosylation factor 1 (ARFGAP1) inhibitor. Learn More
  2. CCG-63802

    Catalog No. A11373
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    CCG-63802 is a reversible inhibitor of regulator of G-protein signaling (RGS) proteins. Selective amongst RGS proteins, with greatest potency at RGS4. Learn More
  3. CASIN

    Catalog No. A12912
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    Cdc42 GTPase inhibitor
    CASIN is a novel and potent Cdc42 inhibitor. Learn More
  4. CCG 50014

    Catalog No. A16432
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    RGS4 inhibitor
    CCG 50014 is a potent and selective inhibitor of RGS4 with IC50 of 30 nM. Learn More
  5. MK-6892

    Catalog No. A12982
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    GPR109A agonist
    MK-6892 is a potent, selective, and full agonist for the high affinity nicotinic acid (NA) receptor GPR109A.K i and GTPγS EC 50 of MK-6892 on the Human GPR109A is 4 nM and 16 nM, respectively. Learn More
  6. CID16020046

    Catalog No. A16818
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    GPR55 antagonist
    CID16020046 is a selective GPR55 antagonist, inhibiting GPR55 constitutive activity with IC50 of 0.15 μM in yeast. It demonstrates weak activity against a broad spectrum of other GPCRs, ion channels, kinases, and nuclear receptor. Learn More
  7. TM N1324

    Catalog No. A17038
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    GPR39 agonist
    TM N1324 is an agonist of G-Protein-Coupled Receptor 39 (GPR39) with EC50s of 9 nM/5 nM in the presence of Zn2+, and 280 nM/180 nM in the absence of Zn2+ for human/murine GPR39. Learn More

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