LXR
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Rovazolac
Catalog No. A18354 liver x receptor (LXR) modulatorRovazolac is a liver x receptor (LXR) modulator extracted from patent WO2013130892A1. Learn More -
LXR-623
Catalog No. A21366 LXRα and full LXRβ agonistLXR-623 is a brain-penetrant partial LXRα and full LXRβ agonist, with IC50s of 24 nM and 179 nM, respectively. Learn More -
RGX-104 free Acid
Catalog No. A21513 LXR agonistRGX-104 free Acid is an orally bioavailable and potent liver-X nuclear hormone receptor (LXR) agonist that modulates innate immunity via transcriptional activation of the ApoE gene. Learn More -
AZ876
Catalog No. A21026 -
GW3965 HCl
Catalog No. A11204 LXR-like receptors agonistGW3965 HCl is a selective and orally active liver X receptor (LXR) full agonist. Learn More -
T0901317
Catalog No. A12652 LXR/FXR agonistT0901317 is a potent and selective agonist for LXR and FXR, with EC50s of 50 nM and 5 μM, respectively Learn More -
Cerpegin
Catalog No. A12865 Cerpegin is a naturally occurring pyridinone alkaloid isolated from Roxb, a tradional indian medicine used as an anti-inflammatory, analgesic, antiulcer and tranquilizer. Learn More -
Mogroside II A2
Catalog No. A12166 Mogroside II-A2, a triterpenoid glycoside isolated from the extracts of Luo Han Guo, is a nonsugar sweetener. Mogrosides are sweeter than sucrose. Mogrosides exhibit antioxidant, antidiabetic and anticancer activities. Learn More -
GW3965
Catalog No. A15100 Liver X Receptor AgonistGW3965 is a potent, selective LXR agonist for hLXRα and hLXRβ with EC50 of 190 and 30 nM, respectively. Learn More -
Sobetirome
Catalog No. A15241 TRβ agonistSobetirome is a thyroid hormone receptor β (TRβ)-specific agonist, Sobetirome is designed to bind selectively to TRβ-1 with EC50 of 0.16 μM. Learn More -
SR9243
Catalog No. A15535 LXR agonistSR9243 is a potent and selective LXR inverse agonist. SR9243 kills cancer cells by inhibiting lipid production and the Warburg effect. It induces cell death in multiple types of cancer and does not cause the side effects that have derailed previous attempts to target these processes. Learn More -
SR9238
Catalog No. A15763 LXR Inverse AgonistSR9238 is a potent and selective LXR inverse agonist (IC50 values are 43 and 214 nM for LXRβ and LXRα, respectively). Learn More -
GSK-2033
Catalog No. A17017 LXR antagonistGSK-2033 is a potent cell-active LXR antagonist (pIC50 = 7.5). It enhances T-cell proliferation and blocks T 0901317-antiproliferative activity on T-cells and is cell permeable. Learn More