LPA Receptor

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  1. BMS-986020 sodium

    Catalog No. A21842
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    LPA1 antagonist
    BMS-986020 sodium is a high-affinity lysophosphatidic acid receptor 1 (LPA1) antagonist. Learn More
  2. LPA2 antagonist 1

    Catalog No. A21308
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    LPA2 antagonist
    LPA2 antagonist 1 is a LPA2 antagonist with an IC50 of 17 nM. Learn More
  3. LPA1 antagonist 1

    Catalog No. A21301
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    LPA1 antagonist
    LPA1 antagonist 1 is a highly selective Lysophosphatidic Acid receptor-1 (LPA1) antagonist with an IC50 of 25 nM. Learn More
  4. SAR-100842

    Catalog No. A12156
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    lysophaphatidic acid 1 (LPA1/Edg-2) receptor inhibitor
    SAR-100842 is a lysophaphatidic acid 1 (LPA1/Edg-2) receptor inhibitor. Learn More
  5. ONO-7300243

    Catalog No. A16644
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    LPA1 antagonist
    ONO-7300243 is a novel, potent lysophosphatidic acid receptor 1 (LPA1) antagonist with IC50 of 0.16 μM. Learn More
  6. Radioprotectin-1

    Catalog No. A18628
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    LPA2 agonist
    Radioprotectin-1 is a potent and specific nonlipid agonist of lysophosphatidic acid receptor 2 (LPA2), with an EC50 value of 25 nM for murine LPA2 subtype. Learn More
  7. AS2717638

    Catalog No. A18630
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    LPA5 antagonist
    AS2717638 is an oral active and selective lysophosphatidic acid receptor 5 (LPA5) antagonist, with an IC50 of 38 nM for hLPA5. AS2717638 also significantly improves PGE2-, PGF2α-, and AMPA-induced allodynia. Learn More
  8. ASP6432

    Catalog No. A18759
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    LPA1 receptor antagonist
    ASP6432 is a potent and selective Type 1 Lysophosphatidic Acid (LPA1) receptor antagonist. Learn More
  9. GRI 977143

    Catalog No. A15343
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    LPA2 agonist
    GRI 977143, selective lysophosphatidic acid 2 (LPA2) receptor non-lipid agonist (EC50 = 3.3 uM). Learn More
  10. AM966

    Catalog No. A13982
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    LPA1 receptor antagonist
    AM966 is a high affinity, selective, oral antagonist of LPA1 receptor (lysophosphatidic acid receptor) with an IC50 value of 17 nM. Learn More
  11. AM095

    Catalog No. A13981
    LPA1 receptor antagonist
    AM095 is a potent LPA1 receptor antagonist because it inhibited GTP??S binding to Chinese hamster ovary (CHO) cell membranes overexpressing recombinant human or mouse LPA1 with IC50 values of 0.98 and 0.73 μM, respectively, and exhibited no LPA1 agonism. Learn More
  12. AM095 free base

    Catalog No. A14180
    LPA1 Receptor antagonist
    AM095 is a novel, potent and orally bioavailable antagonist of lysophosphatidic acid type 1 receptor (LPA1) with IC50 values of 0.73 and 0.98 μM for mouse or recombinant human LPA1, respectively Learn More
  13. Ki16198

    Catalog No. A11966
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    LPA Receptor antagonist
    Ki16198 is a potent LPA receptor antagonist and inhibits LPA1- and LPA3-induced inositol phosphate production with Ki of 0.34 μM and 0.93 μM, respectively. Learn More
  14. Ki16425

    Catalog No. A10501
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    LPA Receptor Antagonist
    Ki16425 is a LPA receptor antagonist with selectivity for LPA1 and LPA3 and exhibits Ki values of 0.34, 6.5, and 0.93 μM for the human LPA1, LPA2, and LPA3 receptors, respectively. Learn More

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