LPA Receptor
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ASP6432
Catalog No. A18759 LPA1 receptor antagonistASP6432 is a potent and selective Type 1 Lysophosphatidic Acid (LPA1) receptor antagonist. Learn More -
AS2717638
Catalog No. A18630 LPA5 antagonistAS2717638 is an oral active and selective lysophosphatidic acid receptor 5 (LPA5) antagonist, with an IC50 of 38 nM for hLPA5. AS2717638 also significantly improves PGE2-, PGF2α-, and AMPA-induced allodynia. Learn More -
Radioprotectin-1
Catalog No. A18628 LPA2 agonistRadioprotectin-1 is a potent and specific nonlipid agonist of lysophosphatidic acid receptor 2 (LPA2), with an EC50 value of 25 nM for murine LPA2 subtype. Learn More -
ONO-7300243
Catalog No. A16644 LPA1 antagonistONO-7300243 is a novel, potent lysophosphatidic acid receptor 1 (LPA1) antagonist with IC50 of 0.16 μM. Learn More -
LPA1 antagonist 1
Catalog No. A21301 LPA1 antagonistLPA1 antagonist 1 is a highly selective Lysophosphatidic Acid receptor-1 (LPA1) antagonist with an IC50 of 25 nM. Learn More -
LPA2 antagonist 1
Catalog No. A21308 LPA2 antagonistLPA2 antagonist 1 is a LPA2 antagonist with an IC50 of 17 nM. Learn More -
BMS-986020 sodium
Catalog No. A21842 LPA1 antagonistBMS-986020 sodium is a high-affinity lysophosphatidic acid receptor 1 (LPA1) antagonist. Learn More -
Ki16425
Catalog No. A10501 LPA Receptor AntagonistKi16425 is a LPA receptor antagonist with selectivity for LPA1 and LPA3 and exhibits Ki values of 0.34, 6.5, and 0.93 μM for the human LPA1, LPA2, and LPA3 receptors, respectively. Learn More -
Ki16198
Catalog No. A11966 LPA Receptor antagonistKi16198 is a potent LPA receptor antagonist and inhibits LPA1- and LPA3-induced inositol phosphate production with Ki of 0.34 μM and 0.93 μM, respectively. Learn More -
AM095 free base
Catalog No. A14180 LPA1 Receptor antagonistAM095 is a novel, potent and orally bioavailable antagonist of lysophosphatidic acid type 1 receptor (LPA1) with IC50 values of 0.73 and 0.98 μM for mouse or recombinant human LPA1, respectively Learn More -
AM095
Catalog No. A13981 LPA1 receptor antagonistAM095 is a potent LPA1 receptor antagonist because it inhibited GTP??S binding to Chinese hamster ovary (CHO) cell membranes overexpressing recombinant human or mouse LPA1 with IC50 values of 0.98 and 0.73 μM, respectively, and exhibited no LPA1 agonism. Learn More -
AM966
Catalog No. A13982 LPA1 receptor antagonistAM966 is a high affinity, selective, oral antagonist of LPA1 receptor (lysophosphatidic acid receptor) with an IC50 value of 17 nM. Learn More -
GRI 977143
Catalog No. A15343 LPA2 agonistGRI 977143, selective lysophosphatidic acid 2 (LPA2) receptor non-lipid agonist (EC50 = 3.3 uM). Learn More