LPA Receptor

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  1. Ki16425

    Catalog No. A10501
    LPA Receptor Antagonist
    Ki16425 is a LPA receptor antagonist with selectivity for LPA1 and LPA3 and exhibits Ki values of 0.34, 6.5, and 0.93 μM for the human LPA1, LPA2, and LPA3 receptors, respectively. Learn More
  2. Ki16198

    Catalog No. A11966
    LPA Receptor antagonist
    Ki16198 is a potent LPA receptor antagonist and inhibits LPA1- and LPA3-induced inositol phosphate production with Ki of 0.34 μM and 0.93 μM, respectively. Learn More
  3. AM095 free base

    Catalog No. A14180
    LPA1 Receptor antagonist
    AM095 is a novel, potent and orally bioavailable antagonist of lysophosphatidic acid type 1 receptor (LPA1) with IC50 values of 0.73 and 0.98 μM for mouse or recombinant human LPA1, respectively Learn More
  4. AM095

    Catalog No. A13981
    LPA1 receptor antagonist
    AM095 is a potent LPA1 receptor antagonist because it inhibited GTP??S binding to Chinese hamster ovary (CHO) cell membranes overexpressing recombinant human or mouse LPA1 with IC50 values of 0.98 and 0.73 μM, respectively, and exhibited no LPA1 agonism. Learn More
  5. AM966

    Catalog No. A13982
    LPA1 receptor antagonist
    AM966 is a high affinity, selective, oral antagonist of LPA1 receptor (lysophosphatidic acid receptor) with an IC50 value of 17 nM. Learn More
  6. GRI 977143

    Catalog No. A15343
    LPA2 agonist
    GRI 977143, selective lysophosphatidic acid 2 (LPA2) receptor non-lipid agonist (EC50 = 3.3 uM). Learn More

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