Progesterone Receptors
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Asoprisnil
Catalog No. A19030 Progesterone receptor modulatorAsoprisnil (J867), a selective progesterone receptor modulator, exhibits mixed progesterone agonist and antagonist effects on various progesterone targeted tissues in animal and human. Learn More -
Nomegestrol acetate
Catalog No. A21829 progesterone receptor agonistNomegestrol acetate is a potent, highly selective progestogen, which is characterized as a full agonist at the progesterone receptor, with no or minimal binding to other steroid receptors, including the androgen and glucocorticoid receptors. Learn More -
Ulipristal acetate
Catalog No. A21041 progesterone receptor modulatorUlipristal (acetate) is a novel selective progesterone receptor modulator (SPRM) for the treatment of benign gynecological conditions such as uterine myoma. Learn More -
Tamoxifen Citrate
Catalog No. A10885 Estrogen receptor antagonistTamoxifen Citrateis a selective and potent inhibitor of mammalian sterol isomerase. Learn More -
Drospirenone
Catalog No. A10336 Drospirenone is a synthetic hormone used in birth control pills. Learn More -
Levonorgestrel
Catalog No. A10529 Levonorgestrelis a synthetic progesterone analog; binds to the progesterone receptor (relative binding affinities are < 0.02, 7.5, 17, 58 and 323 % for estrogen receptors, glucocorticoid receptors, mineralocorticoid receptors, androgen receptors and progesterone receptors respectively). Learn More -
Megestrol Acetate
Catalog No. A10563 Megestrol Acetate is a progesterone derivative with antineoplastic properties Learn More -
Lonaprisan
Catalog No. A14130 progesterone receptor antagonistLonaprisan is an orally bioavailable pentafluoroethyl derivative of a mifepristone-related steroid with antiprogestagenic activity. Learn More -
Nestoron
Catalog No. A15184 progesterone receptor agonistNestoron is a 19-norprogesterone derivative and steroidal progestin which is used as a hormonal contraceptive; a high-affinity agonist of the progesterone receptor. Learn More -
Tanaproget
Catalog No. A15256 Progesterone receptor agonistTanaproget is a novel nonsteroidal progesterone receptor agonist which can bind to the PR from various species with a higher relative affinity than reference steroidal progestins. Learn More -
ACT-129968 (Setipiprant)
Catalog No. A15780 -
17-Hydroxyprogesterone
Catalog No. A15860 17-Hydroxyprogesterone is an endogenous progestogen as well as chemical intermediate in the biosynthesis of other steroid hormones, including the corticosteroids and the androgens and the estrogens. Learn More -
Medroxyprogesterone Acetate
Catalog No. A11625 progesterone receptor agonistMedroxyprogesterone acetate is a progestin, a synthetic variant of the human hormone progesterone and a potent progesterone receptor agonist. Learn More -
Etonogestrel
Catalog No. A16117 Etonogestrel is a steroidal progestin used in hormonal contraceptives, most notably the subdermal implant Nexplanon and the vaginal ring NuvaRing. Learn More -
Hydroxyprogesterone caproate
Catalog No. A16143 Hydroxyprogesterone caproate is a synthetic, steroidal progestin; an ester derivative of 17?α-hydroxyprogesterone formed from caproic acid. Learn More -
Desogestrel
Catalog No. A16173 Desogestrel is a synthetic progestational hormone used often as the progestogenic component of combined oral contraceptive agents. Learn More