Shop By
Catalog No.
Product Name
Application
Product Information
Product Citation
-
AMPA and Kainate antagonist
GYKI-52466 dihydrochloride is selective non-competitive AMPA receptor antagonist (IC50 values are 10-20, ~ 450 and >> 50 μM for AMPA- , kainate- and NMDA-induced responses respectively). - Ampalex is an ampakine and nootropic that acts as an AMPA receptor positive allosteric modulator
- Mariusz Papp, .et al. , J Psychopharmacol, 2020, Dec;34(12):1418-1430 PMID: 33200659
- Abigail Benn, .et al. , J Neurosci, 2016, May 4; 36(18):4930-4939 PMID: 27147648
-
AMPA desensitization inhibitor
Cyclothiazide is a benzothiadiazide that acts as a potentiator of AMPA receptors, positively modulating its response to glutamic acid (EC50 = 3.8 M). -
AMPA Receptor Blocker
IEM 1754 Dihydrobromide is a voltage-dependent open-channel blocker of AMPA receptors.
