Opioid Receptors

Actions
  1. Agonist (6)
  2. Antagonist (4)
  3. Inhibitor (1)


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Catalog No. Product Name Application Product Information
A11072

ADL5859 HCl

Opioid Receptor agonist
ADL5859 HCl is a highly potent and selective δ opioid receptor agonist with Ki value to be 0.84 nM and ED50 value to be 20 nM.
A11322

BAN ORL 24

NOP antagonist
BAN ORL 24 is a potent and selective NOP receptor antagonist.
A11210

BRL 52537 HCl

Opioid Receptors agonist
BRL 52537 hydrochloride is a highly selective and potent κ-opioid agonist (Ki = 0.24 nM). 25 times more potent than morphine.
A14085

Eluxadoline

opioid receptor agonist
Eluxadoline is a novel, orally-active drug approved for the treatment of diarrhea and abdominal pain in individuals with diarrhea-predominant irritable bowel syndrome (IBS-D).
A10350

Enalapril maleate

ACE inhibitor
Enalapril is an angiotensin converting enzyme (ACE) inhibitor used in the treatment of hypertension and some types of chronic heart failure.
A11076

JTC-801

Opioid Receptor antagonist
JTC-801 is a selective antagonist for the nociceptin receptor, also known as the ORL-1 receptor.
A15149

LY2795050

k-opioid receptor antagonist
LY2795050 is a novel selective ??-opioid Receptor (KOR) antagonist (IC50=0.72 nM) and has the potential as a PET tracer to image KOR in vivo.
A10561

MCOPPB 3HCl

NOP receptor agonist
MCOPPB is a compound which acts as a potent and selective agonist for the nociceptin receptor, with a pKi of 10.07.
A15159

Methylnaltrexone Bromide

μ-opioid antagonist
Methylnaltrexone Bromide is a pheriphally-acting ??-opioid antagonist that acts on the gastrointestinal tract to decrease opioid-induced constipation.
A13843

Nalmefene hydrochloride

dopamine receptor agonist
Nalmefene hydrochloride is an opioid receptor antagonist.
A11718

Trimebutine

-
Trimebutine is a drug with antimuscarinic and weak mu opioid agonist effects.
A15444

TRV130 HCl (Oliceridine)

µ- opioid receptor agonist
TRV 130 HCl is a novel μ-opioid receptor (MOR) G protein-biased ligand; elicits robust G protein signaling(pEC50=8.1), with potency and efficacy similar to morphine, but with far less beta-arrestin recruitment and receptor internalization.

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