Opioid Receptors

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Catalog No. Product Name Application Product Information
A11072 SALE

ADL5859 HCl

Opioid Receptor agonist
ADL5859 HCl is a highly potent and selective δ opioid receptor agonist with Ki value to be 0.84 nM and ED50 value to be 20 nM.


NOP antagonist
BAN ORL 24 is a potent and selective NOP receptor antagonist.

BRL 52537 HCl

Opioid Receptors agonist
BRL 52537 hydrochloride is a highly selective and potent κ-opioid agonist (Ki = 0.24 nM). 25 times more potent than morphine.


opioid receptor agonist
Eluxadoline is a novel, orally-active drug approved for the treatment of diarrhea and abdominal pain in individuals with diarrhea-predominant irritable bowel syndrome (IBS-D).
A10350 SALE

Enalapril maleate

ACE inhibitor
Enalapril is an angiotensin converting enzyme (ACE) inhibitor used in the treatment of hypertension and some types of chronic heart failure.
A11076 SALE


Opioid Receptor antagonist
JTC-801 is a selective antagonist for the nociceptin receptor, also known as the ORL-1 receptor.


k-opioid receptor antagonist
LY2795050 is a novel selective ??-opioid Receptor (KOR) antagonist (IC50=0.72 nM) and has the potential as a PET tracer to image KOR in vivo.
A10561 SALE


NOP receptor agonist
MCOPPB is a compound which acts as a potent and selective agonist for the nociceptin receptor, with a pKi of 10.07.

Methylnaltrexone Bromide

μ-opioid antagonist
Methylnaltrexone Bromide is a pheriphally-acting ??-opioid antagonist that acts on the gastrointestinal tract to decrease opioid-induced constipation.
A13843 SALE

Nalmefene hydrochloride

dopamine receptor agonist
Nalmefene hydrochloride is an opioid receptor antagonist.
A11718 SALE


Trimebutine is a drug with antimuscarinic and weak mu opioid agonist effects.
A15444 SALE

TRV130 HCl (Oliceridine)

µ- opioid receptor agonist
TRV 130 HCl is a novel μ-opioid receptor (MOR) G protein-biased ligand; elicits robust G protein signaling(pEC50=8.1), with potency and efficacy similar to morphine, but with far less beta-arrestin recruitment and receptor internalization.

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