Shop By
Catalog No.
Product Name
Application
Product Information
Product Citation
-
AdipoR1 and AdipoR2 agonist
AdipoRon is a novel small-molecule AdipoR agonist; binds to both AdipoR1(Kd= 1.8 uM) and AdipoR2(Kd=3.1 uM). IC50 value: 1.8/3.1 uM(AdipoR1/2, Kd)- Weidong Yan, .et al. , Pharmaceutics, 2022, Nov 15;14(11):2467 PMID: 36432657
- Yunjing Yan, .et al. , J Pathol, 2022, Jun;257(2):146-157 PMID: 35072951
- Uchida T, .et al. , J Ocul Pharmacol Ther, 2019, Aug 28 PMID: 31460821
-
motilin receptor agonist
Camicinal hydrochloride (GSK962040 hydrochloride) is a small molecule, selective motilin receptor agonist with pEC50 of 7.9. -
TAAR1
agonist
RO5203648 hydrochloride is a partial agonist of Trace amine-associated receptor 1 (TAAR1).