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Catalog No.
Product Name
Application
Product Information
Product Citation
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AhR antagonist
StemRegenin 1 (SR1) is a cell-permeable purine derivative that acts as an antagonist of aryl hydrocarbon receptor and promotes the self-renewal of hematopoietic stem cells (HSCs). -
AhR antagonist
CH-223191 is a ligand-selective antagonist of the Ah (Dioxin) receptor.- Yukiko Sakakibara, .et al. , Biopharm Drug Dispos, 2022, Oct;43(5):175-182 PMID: 36000181
- Jie Tang, .et al. , Ecotoxicol Environ Saf, 2021, Sep 15;221:112423 PMID: 34146985
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aryl hydrocarbon receptor agonist
L-Kynurenine is a metabolite of the amino acid L-tryptophan. L-Kynurenine is an aryl hydrocarbon receptor agonist. -
AHR antagonist
AHR antagonist 1 is an aryl hydrocarbon receptor (AHR) antagonist extracted from patent WO2017202816A1, example 23, has an IC50 of 39.9 nM in human cell line. -
aryl hydrocarbon receptor activator
1,4-Chrysenequinone, a polycyclic aromatic quinone, acts as an activator of aryl hydrocarbon receptor (AhR). - NSC-703786 (5F-203) is a cytotoxic molecule that forms DNA adducts leading to cell death. NSC-703786 induces aryl hydrocarbon receptor signaling, and elevates expression of CYP1A1. Treatment of cells with NSC-703786 also leads to elevation of reactive oxygen species and activation of p38, JNK and ERK.