GnRH receptor
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Alarelin Acetate
Catalog No. A20968 -
(R)-Elagolix
Catalog No. A21184 GnRHR antagonistElagolix is a highly potent, selective, orally-active, short-duration, non-peptide antagonist of the gonadotropin-releasing hormone receptor (GnRHR) (KD = 54 pM). Learn More -
Leuprolide Acetate
Catalog No. A15143 GnRH agonistLeuprolide acetate is a GnRH analog; leuprolide acetate acts as an agonist at pituitary GnRH receptors. Learn More -
Goserelin
Catalog No. A21197 GnRH agonistGoserelin(ICI 118630) is an injectable gonadotropin releasing hormone superagonist (GnRH agonist). Learn More -
Cetrorelix Acetate
Catalog No. A18282 GnRH antagonistCetrorelix acetate is a synthetic decapeptide with gonadotropin-releasing hormone (GnRH) antagonistic activity used in infertility treatment. The IC50 of 1.21 nM. Learn More -
Nafarelin Acetate
Catalog No. A17992 GnRH agonistNafarelin is a gonadotropin-releasing hormone agonist (GnRH agonist) which acts as an analog of GnRH. Learn More -
Leuprorelin Acetate
Catalog No. A17986 GnRH/LHRH receptor agonistLeuprorelin is a Gonadotropin-releasing hormone (GnRH, luteinizing hormone-releasing hormone, LHRH) receptor agonist. Suppresses estradiol, LH and FSH serum levels and represses the growth of experimental rat endometriosis. Learn More -
Relugolix
Catalog No. A17783 GnRH antagonistRelugolix is a novel, non-peptide, orally active gonadotropin-releasing hormone (GnRH) antagonist with IC50 of 0.33 nM in the presence of 40% fetal bovine serum, TAK-385 possesses higher affinity and potent antagonistic activity compared with TAK-013. Learn More -
Goserelin Acetate
Catalog No. A15959 GnRH agonistGoserelin is a synthetic decapeptide analog of luteinizing hormone-releasing hormone (LHRH) with antineoplastic activity. Learn More -
Triptorelin Acetate
Catalog No. A15997 GnRH agonistTriptorelin is a gonadotropin-releasing hormone agonist (GnRH agonist) used as the acetate or pamoate salts. Learn More -
Ozarelix
Catalog No. A12350 GnRH antagonistOzarelix is a fourth generation GnRH antagonist, induces apoptosis in hormone refractory androgen receptor negative prostate cancer cells modulating expression and activity of death receptors. Learn More -
AEZS-108
Catalog No. A13536 GnRH-1 agonistAEZS-108 is a peptide agonist of the gonadotropin releasing hormone-1 receptor (GnRH-1R) that is conjugated to the anthracycline antibiotic doxorubicin with potential antineoplastic activity. Learn More -
Elagolix sodium
Catalog No. A13893 GnRH antagonistElagolix is a Gonadotropin-Releasing Hormone (GnRH) Antagonist. Elagolix inhibits gonadatropin releasing hormone (GnRH) receptors in the pituitary gland and ultimately reduces circulating sex hormone levels. Learn More -
GHRP-6 Acetate
Catalog No. A13464 GHRP-6 Acetate is a growth hormone releasing peptide. Learn More -
Degarelix acetate
Catalog No. A12840 GnRH antagonistDegarelix acetate is a gonadotropin releasing hormone (GnRH) receptor antagonist. Learn More -
Ganirelix
Catalog No. A12862 Ganirelix is an injectable competitive gonadotropin-releasing hormone antagonist (GnRH antagonist) Learn More -
SR 144528
Catalog No. A12376 CB2 inverse agonistSR 144528 is a selective peripheral cannabinoid receptor inverse agonist that displays a Ki value of 0.6 nM for rat spleen and human recombinant CB2 receptors and a Ki value of 400 nM for rat brain and human recombinant CB1 receptors. Learn More -
NBI-42902
Catalog No. A12375 GnRH receptor InhibitorNBI-42902 is a novel nonpeptide antagonist of the human gonadotropin-releasing hormone receptor Learn More -
Abarelix Acetate
Catalog No. A12613 GnRH antagonistAbarelix acetate is a synthetic peptide gonadotropin releasing hormone receptor (GnRH) antagonist Learn More