GnRH receptor

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  1. Ozarelix

    Catalog No. A12350
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    GnRH antagonist
    Ozarelix is a fourth generation GnRH antagonist, induces apoptosis in hormone refractory androgen receptor negative prostate cancer cells modulating expression and activity of death receptors. Learn More
  2. Nafarelin Acetate

    Catalog No. A17992
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    GnRH agonist
    Nafarelin is a gonadotropin-releasing hormone agonist (GnRH agonist) which acts as an analog of GnRH. Learn More
  3. Leuprorelin Acetate

    Catalog No. A17986
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    GnRH/LHRH receptor agonist
    Leuprorelin is a Gonadotropin-releasing hormone (GnRH, luteinizing hormone-releasing hormone, LHRH) receptor agonist. Suppresses estradiol, LH and FSH serum levels and represses the growth of experimental rat endometriosis. Learn More
  4. Relugolix

    Catalog No. A17783
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    GnRH antagonist
    Relugolix is a novel, non-peptide, orally active gonadotropin-releasing hormone (GnRH) antagonist with IC50 of 0.33 nM in the presence of 40% fetal bovine serum, TAK-385 possesses higher affinity and potent antagonistic activity compared with TAK-013. Learn More
  5. Goserelin Acetate

    Catalog No. A15959
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    GnRH agonist
    Goserelin is a synthetic decapeptide analog of luteinizing hormone-releasing hormone (LHRH) with antineoplastic activity. Learn More
  6. Triptorelin Acetate

    Catalog No. A15997
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    GnRH agonist
    Triptorelin is a gonadotropin-releasing hormone agonist (GnRH agonist) used as the acetate or pamoate salts. Learn More
  7. Leuprolide Acetate

    Catalog No. A15143
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    GnRH agonist
    Leuprolide acetate is a GnRH analog; leuprolide acetate acts as an agonist at pituitary GnRH receptors. Learn More
  8. AEZS-108

    Catalog No. A13536
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    GnRH-1 agonist
    AEZS-108 is a peptide agonist of the gonadotropin releasing hormone-1 receptor (GnRH-1R) that is conjugated to the anthracycline antibiotic doxorubicin with potential antineoplastic activity. Learn More
  9. Elagolix sodium

    Catalog No. A13893
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    GnRH antagonist
    Elagolix is a Gonadotropin-Releasing Hormone (GnRH) Antagonist. Elagolix inhibits gonadatropin releasing hormone (GnRH) receptors in the pituitary gland and ultimately reduces circulating sex hormone levels. Learn More
  10. GHRP-6 Acetate

    Catalog No. A13464
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    GHRP-6 Acetate is a growth hormone releasing peptide. Learn More
  11. Degarelix acetate

    Catalog No. A12840
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    GnRH antagonist
    Degarelix acetate is a gonadotropin releasing hormone (GnRH) receptor antagonist. Learn More
  12. Ganirelix

    Catalog No. A12862
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    Ganirelix is an injectable competitive gonadotropin-releasing hormone antagonist (GnRH antagonist) Learn More
  13. SR 144528

    Catalog No. A12376
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    CB2 inverse agonist
    SR 144528 is a selective peripheral cannabinoid receptor inverse agonist that displays a Ki value of 0.6 nM for rat spleen and human recombinant CB2 receptors and a Ki value of 400 nM for rat brain and human recombinant CB1 receptors. Learn More
  14. NBI-42902

    Catalog No. A12375
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    GnRH receptor Inhibitor
    NBI-42902 is a novel nonpeptide antagonist of the human gonadotropin-releasing hormone receptor Learn More
  15. Abarelix Acetate

    Catalog No. A12613
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    GnRH antagonist
    Abarelix acetate is a synthetic peptide gonadotropin releasing hormone receptor (GnRH) antagonist Learn More
  16. Cetrorelix Acetate

    Catalog No. A18282
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    GnRH antagonist
    Cetrorelix acetate is a synthetic decapeptide with gonadotropin-releasing hormone (GnRH) antagonistic activity used in infertility treatment. The IC50 of 1.21 nM. Learn More

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