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GPR120 modulator 2
Catalog No. A15095 GPR120 modulator 2 is useful for modulating G protein-coupled receptor 120 (GPR120). Learn More -
TC-G-1008
Catalog No. A16364 GPR39 agonistTC-G-1008 is a GPR39 (zinc receptor) agonist (EC50 values are 0.4 and 0.8 nM for rat and human receptors respectively). Learn More -
NCRW0005-F05
Catalog No. A16184 GPR139 antagonistNCRW0005-F05, first antagonist selective for GPR139 (IC50 value 0.21 uM); a useful tool to study GPR139 pharmacology, especially in combination with the GPR139 agonist JNJ 63533054. Learn More -
TUG-770
Catalog No. A12994 FFA1/GPR40 AgonistTUG-770 is a Highly Potent Free Fatty Acid Receptor 1 (FFA1/GPR40) Agonist for Treatment of Type 2 Diabetes. Learn More -
Versipelostatin
Catalog No. A16069 Versipelostatin is a novel GRP78/Bip molecular chaperone down-regulator of microbial origin that was isolated from the metabolite of Streptomyces versipellis strain 4083-SVS6. Learn More -
GSK137647A
Catalog No. A14542 FFA4/GPR120 agonistGSK137647A is a selective FFA4 agonist, with pEC50 of 6.3, 6.2, and 6.1 for human, Mouse and Rat FFA4, respectively. Learn More -
APD597 (JNJ-38431055)
Catalog No. A15452 GPR119 agonistAPD597 is a GPR119 agonist intended for the treatment of type 2 diabetes, with EC50 of 46 nM for hGPR119. Learn More -
NIBR189
Catalog No. A15775 EBI2 (GPR183) receptor antagonistNIBR189 is a small molecule antagonist of the Epstein-Barr virus-induced gene 2 (EBI2; GPR183) receptor with IC50 of 16 nM(Binding) and 11 nM (Functional). Learn More -
6-OAU
Catalog No. A15507 GPR84 agonist6-OAU is a surrogate agonist of GPR84; activates human GPR84 in the presence of Gqi5 chimera in HEK293 cells with an EC50 of 105 nM in the PI assay. Learn More -
OC 000459
Catalog No. A11946 CRTH2 antagonistOC 000459 is a potent, oral and selective CRTH2 (also known as DP2) antagonist. Learn More -
GPR120 modulator 1
Catalog No. A15094 GPR120 modulator 1 is useful for modulating G protein-coupled receptor 120 (GPR120). Learn More -
Deoxycholic acid
Catalog No. A14952 Deoxycholic acid, extracted from Pig bile, Suitability:Ethanol,ether,three oxygen methane,acetone,acetic acid,alkali hydroxide and alkali carbonate solution. Learn More -
AMG 837 calcium hydrate
Catalog No. A13468 GPR40/FFA1 agonistAMG-837 calcium hydrate is a potent, orally bioavailable GPR40 agonist. Learn More -
APD668
Catalog No. A14342 GPR119 agonistAPD668 is a potent GPR119 agonist with EC50 of 2.7 nM and 33 nM for hGPR119 and ratGPR119 respectively. Learn More -
AZD1981
Catalog No. A13186 CRTH2 receptor antagonistAZD1981, as a potent antagonist in a disease relevant cell system, inhibits DK-PGD2-induced CD11b expression in human eosinophils with IC50 of 10 nM. Learn More -
AR-231453
Catalog No. A13716 GPR119 agonistAR-231453 is a potent and selective small molecule agonis of GPR119 that enhances glucose dependent insulin secretion and glucagon like peptide-1 (GLP-1) release. Learn More -
MBX-2982
Catalog No. A12634 GPR119 agonistMBX-2982 is a potential first-in-class treatment for type 2 diabetes that targets G protein-coupled receptor 119 (GPR119), a receptor that interacts with bioactive lipids known to stimulate glucose-dependent insulin secretion. Learn More -
Diphenyleneiodonium chloride
Catalog No. A13359 GPR3 agonist/NOS/ NADPH oxidases inhibitorDiphenyleneiodonium chloride has been shown to be a potent irreversible inhibitor of NOS2 (iNOS) from macrophages and NOS3 (eNOS) from endothelial cells. Learn More
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