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Prostanoid Receptors

Prostanoid Receptors

Catalog No.	Product Name	Application	Product Information
A11483 SALE	Laropiprant (MK0524)	DP1 inhibitor	Laropiprant is used in combination with niacin to reduce blood cholesterol. Laropiprant acts as a DP1 antagonist, reducing the vasodilation.
A15968	TG6-10-1	Prostaglandin E2 receptor antagonist	TG6-10-1 is a potent and selective antagonist for the prostaglandin E2 receptor subtype EP2.
A15853	CP544326 (Taprenepag)	EP2 Agonist‎	C-544326 is a potent and selective prostaglandin E2 receptor agonist with EC50 value of 2.8 nM.
A12894	PF-04418948	EP2 Receptor antagonist	PF-04418948 is a potent and selective prostaglandin EP2 receptor antagonist with IC50 of 16 nM. Phase 1.
A15532	MF498	EP4 receptor antagonist	MF498 is a novel and selective E prostanoid receptor 4 (EP4 receptor) antagonist, displayed strong binding affinity for the EP4 receptor with Ki of 0.7 nM,
A15525	GW627368	EP4 receptor antagonist	GW627368 is a novel, potent and selective competitive antagonist of prostanoid EP4 receptor(Ki= 100 nM) with additional human TP receptor affinity(Ki= 150 nM).
A14600	Saikosaponin B2	Prostanoid activator	Saikosaponin B2 is a saponin activator.
A13880 SALE	NS-304 (Selexipag)	prostacyclin receptor agonist	NS-304 is a selective prostacyclin IP1 receptor agonist (Ki values are 260 and 2100 nM and for human and rat IP receptors, and >10 μM for EP1-4, DP, FP, and TP receptors).
A13751	BAY-u 3405	dual antagonist of TP/DP2	BAY-u 3405 is an approved human medication for the treatment of allergic rhinitis that has documented activity as an antagonist of the thromboxane receptor (TP receptor).
A13498	Cloprostenol (sodium salt)	-	Cloprostenol is a synthetic analog of prostaglandin F2α (PGF2α). It is 200 times and 100 times more potent than PGF2α in terminating pregnancy in hamsters and rats, respectively, without the side effects associated with PGF2α.
A11497	MK-2894	EP4 receptor antagonist	MK-2894 is a highly potent and selective second generation EP4 antagonist.
A11742 SALE	Ozagrel hydrochloride	Thromboxane A2 synthesis inhibitor	Ozagrel is an antiplatelet agent working as a thromboxane A2 synthesis inhibitor.
A15964	Grapiprant (CJ-023423)	prostaglandin EP4 receptor antagonist	Grapiprant is a novel, potent and selective prostaglandin EP4 receptor antagonist with antihyperalgesic properties.