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$0.00 GABA Receptors
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THIP
Catalog No. A21738 δ-GABAAR agonistTHIP (Gaboxadol) is a selective δ-aminobutyric acid type A receptor (δ-GABAAR) agonist. Learn More -
CTP354
Catalog No. A15939 GABA(A) modulatorCTP354 a novel deuterated subtype-selective GABA(A) modulator. Learn More -
Vigabatrin
Catalog No. A15277 GABA-transaminase inhibitorVigabatrin is a structural analog of the inhibitory neurotransmitter ??-aminobutyric acid (GABA) that irreversibly inhibits the catabolism of GABA by GABA transaminase. Learn More -
CP-409092
Catalog No. A20152 GABAA receptor partial agonistCP-409092 is a partial agonist of GABAA receptor, with anti-anxiety activity. Learn More -
TPA 023
Catalog No. A20140 GABAA α2/α3 agonistTPA 023 is a GABAA α2/α3 subtype-selective agonist, with Ki of 0.19-0.41 nM. Learn More -
RWJ-51204
Catalog No. A12875 partial agonist of GABA(A) receptorRWJ-51204 is a partial agonist of GABA(A) receptor, with Ki of 0.2-2 nM to the benzodiazepine site on GABA(A) receptors. Learn More -
MRK-016
Catalog No. A12046 GABAA α5 receptor agonistMRK-016 is a selective, orally bioavailable inverse agonist of GABAA α5 receptor, with an EC50 of 3 nM for GABAA α5, and Kis of 0.83, 0.85, 0.77?and 1.4?nM for human?GABAA?α1β3γ2, GABAA?α2β3γ2, GABAA?α3β3γ2, and GABAA?α5β3γ2, respectively; MRK-016 also readily penetrates the CNS. Learn More -
Gabazine
Catalog No. A12627 GABAA receptor antagonistGabazine is a selective and competitive antagonist of GABAA receptor, with an IC50 of ~0.2 μM for GABA receptor. Learn More -
Acamprosate calcium
Catalog No. A11308 GABA receptor agonistAcamprosate calcium(Campral EC) is a GABA receptor agonist and modulator of glutamatergic systems; reduces alcohol consumption in animal models of alcohol addiction. Learn More -
(R)-Baclofen
Catalog No. A16680 GABAB receptor agonist(R)-Baclofen(STX209) is a selective GABAB receptor agonist. Learn More -
L-655708
Catalog No. A21181 GABAA receptor inverse agonistL-655708 is a potent α5 subunit-selective GABAA receptor inverse agonist (Ki = 0.45 nM). Learn More -
Basmisanil
Catalog No. A21321 GABAAα5 modulatorBasmisanil is a highly selective GABAAα5 negative allosteric modulator. Learn More -
CP-409092 hydrochloride
Catalog No. A21397 GABAA receptor partial agonistCP-409092 hydrochloride is a partial agonist of GABAA receptor, with anti-anxiety activity. Learn More -
NS11394
Catalog No. A21425 GABA(A) receptor modulatorNS11394 is a potent and subtype-selective GABA(A) receptor-positive modulator; possesses a functional efficacy selectivity profile of alpha(5) > alpha(3) > alpha(2) > alpha(1) at GABA(A) alpha subunit-containing receptors. Learn More -
SCH 50911
Catalog No. A21630 γ-Aminobutyric acid B GABA(B) receptor antagonistSCH 50911, (+)-(S)-5,5-dimethylmorpholinyl-2-acetic acid, a selective, orally-active and competitive γ-Aminobutyric acid B GABA(B) receptor antagonist. Learn More -
U-101017
Catalog No. A13357 Benzodiazepine receptor/GABAA receptor agonistU-101017 is a partial agonist of benzodiazepine receptor and GABAA receptor, with anxiolytic effects. Learn More -
Gaboxadol hydrochloride
Catalog No. A21730 GABAA receptors agonistGaboxadol hydrochloride (Lu 02-030 hydrochloride) is a selective agonist at GABAA receptors that contain α4-δ subunits, and has anxiolytic and sedative effects. Learn More -
Lorediplon
Catalog No. A13449 GABAA receptor modulatorLorediplon is a novel non-benzodiazepine, hypnotic drug acting as a GABAA receptor modulator, Learn More -
U-93631
Catalog No. A16336 GABAA receptor ligandU-93631 is a GABAA receptor ligand of novel chemical structure with IC50 of 100 nM,and has been shown to induce a rapid, time-dependent decay of GABA-induced whole-cell Cl-currents in recombinant GABAA receptors. Learn More -
Tiagabine hydrochloride
Catalog No. A16135 GABA reuptake inhibitorTiagabine is an anti-convulsive medication. The medication is also utilized in the treatment of panic disorder, as are a few other anticonvulsants. Learn More -
Bemegride
Catalog No. A12298 Bemegride is a central nervous system stimulant and antidote for barbiturate poisoning. Learn More -
Bamaluzole
Catalog No. A17107 -
(-)-Securinine
Catalog No. A17102 GABA receptor antagonist(-)-Securinine is an alkaloid originally isolated from S. suffructicosa. Securinine, is a specific GABA receptor antagonist and has been found to have significant in vivo CNS activity. Learn More -
Cgp 52432
Catalog No. A17140 -
Afloqualone
Catalog No. A17276 GABA receptor agonistAfloqualone, also known as HQ-495, is a centrally acting muscle relaxant. Afloqualone inhibits vestibular nystagmus probably due to both inhibition of selective polysynaptic transmission and enhancement of the effects of GABA and glycine in the lateral vestibular nucleus (LVN), and its GABA-enhancing effect is thought to be attributable to the increased sensitivity of GABA receptors of the LVN neuron site. Learn More -
Homotaurine
Catalog No. A17944 GABA receptor agonistTramiprosate, also known as homotaurine, is a gamma-Aminobutyric acid (GABA) receptor agonist and a glycosaminoglycan mimetic used in the treatment of Alzheimer's disease. Learn More -
Baclofen
Catalog No. A18248 GABA agonistBaclofen is a GABA agonist specific for GABA-B receptors. Baclofen is a synthetic chlorophenyl-butanoic acid derivative used to treat spasms due to spinal cord damage and multiple sclerosis, muscle-relaxing It acts at spinal and supraspinal sites, reducing excitatory transmission. Learn More -
CGP 36742
Catalog No. A18666 GABAB receptor antagonistCGP 36742 is a selective GABAB receptor antagonist that can penetrate the blood?Cbrain barrier after peripheral administration, with an IC50 of 32?μM. CGP 36742 is useful in treatment of depression. Learn More -
Oxiracetam
Catalog No. A14281 Oxiracetam is a cyclic derivative of gamma-aminobutyric acid (GABA). Learn More -
Baicalin
Catalog No. A10121 HIV-1 production InhibitorBaicalin is a known prolyl endopeptidase inhibitor and affects the GABA receptors. Learn More -
Nefiracetam (Translon)
Catalog No. A10631 Nefiracetam is cognitive enhancer. It activates L/N-type calcium channels, cholinergic, monoaminergic and GABAergic systems. Learn More -
SKF 89976A HCl
Catalog No. A10849 GABA uptake inhibitorSKF 89976A hydrochloride is a potent inhibitor of GABA uptake with IC50 of 0.13, 550, 944 and 7210 μM for hGAT-1, rGAT-2, hGAT-3 and hBGT-1 respectively. Learn More -
Flumazenil
Catalog No. A10397 Benzodiazepine antagonistFlumazenil, an imidazobenzodiazepine derivative, antagonizes the actions of benzodiazepines on the central nervous system. Flumazenil competitively inhibits the activity at the benzodiazepine recognition site on the GABA/benzodiazepine receptor complex. Flumazenil is a weak partial agonist in some animal models of activity, but has little or no agonist activity in humans. Learn More -
Furosemide
Catalog No. A10412 Furosemide is a non-competitive antagonist at GABAA receptors with ~ 100-fold greater selectivity for α6-containing receptors than α1-containing receptors. Learn More -
Gabapentin
Catalog No. A10413 Gabapentin (Neurontin) is a pharmaceutical agent, specifically a GABA analogue. Learn More -
Primidone (Mysoline)
Catalog No. A10754 Primidone is an anticonvulsant. Potentiates GABAA receptor function. Learn More -
(+)-Bicuculline
Catalog No. A12590 GABAA antagonist(+)-Bicuculline is a classical GABAA antagonist. Learn More -
AWD 131-138
Catalog No. A13726 GABAA receptor agonistAWD 131-138 is a new low-affinity partial benzodiazepine receptor agonist with potent anticonvulsant and anxiolytic properties in rodent models. Learn More -
2-Hydroxysaclofen
Catalog No. A13696 GABAB receptors antagonist2-Hydroxysaclofen is a potent and selective antagonist at GABAB receptors. Learn More -
Bretazenil
Catalog No. A13784 GABAA agonistBretazenil, a benzodiazepine receptor partial agonist, as an adjunct in the prophylactic treatment of OP poisoning. Learn More -
Piperazine
Catalog No. A16171 GABA receptor agonistPiperazine is an organic compound that consists of a six-membered ring containing two nitrogen atoms at opposite positions in the ring. Learn More -
Cloflubicyne
Catalog No. A13932 GABA antagonistCloflubicyne is a potent non-competitive GABA antagonist, convulsant, laboratory insecticide. Learn More -
a5IA
Catalog No. A14343 Benzodiazepine agonista5IA is a nootropic drug invented in 2004 by a team working for Merck, Sharp and Dohme, which acts as a subtype-selective inverse agonist at the benzodiazepine binding site on the GABAA receptor. Learn More -
RO 15-3890
Catalog No. A14349 benzodiazepine receptor antagonistRo 15-1788 is a benzodiazepine receptor antagonist. Learn More -
Indiplon
Catalog No. A13769 GABAA receptor modulatorIndiplon is a pyrazolopyrimidine that acts as a high-affinity positive allosteric modulator of the GABAA receptor, potentiating GABA-activated chloride currents in a dose-dependent and reversible manner. Learn More -
Guvacine hydrochloride
Catalog No. A13613 GABA uptake inhibitorGuvacine hydrochloride inhibits GABA uptake (IC50 values are 14, 58, 119 and 1870 uM for hGABA T-1, rGABA T-2, hGABA T-3 and hBGT-1 respectively). Learn More -
Muscimol
Catalog No. A14005 GABAA/GABAC agonistMuscimol is a full GABAA agonist and partial GABAC agonist. It binds GABAA on both high- and low-affinity sites (Kd = 10 and 270 nM, respectively), stimulating chloride efflux with an EC50 value of 200 nM. Learn More -
Muscimol hydrobromide
Catalog No. A13459 GABA(A) receptor agonistMuscimol hydrobromide is a potent but toxic structural analog of g-aminobutyric acid (GABA), with a zwitterionic structure. Learn More -
4-Aminobutyric acid
Catalog No. A14934 4-Aminobutyric acid is the chief inhibitory neurotransmitter in the mammalian central nervous system. Learn More
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