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Catalog No.
Product Name
Application
Product Information
Product Citation
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AMPK activator
Acadesine is a selective activator of AMPK in both hepatocytes and adipocytes.
- R. Lim, .et al. , Placenta, 2015, Apr;36(4):454-62 PMID: 25659498
- Stella Liong, .et al. , J Physiol Biochem, 2015, Dec;71(4):703-17 PMID: 26407807
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AMPK activator
A-769662 is a new activator of AMP-activated protein kinase (AMPK).- Daniel Missailidis, .et al. , Int J Mol Sci., 2021, Feb; 22(4): 2046 PMID: 33669532
- Lieberthal W, .et al. , Am J Physiol Renal Physiol, 2019, 2019 PMID: 30995114
- Kikuchi H, .et al. , Kidney Int, 2018, Nov 13. pii: S0085-2538(18)30635-5 PMID: 30455054
- Schneider H, .et al. , Hypertension, 2015, Jul;66(1):108-16 PMID: 26034200
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AMPK activator
EX229 (compound 991) is a potent AMPK activator that is 5-10-fold more potent than A769662 in activating AMPK.- CN Koyani, .et al. , Pharmacol Res, 2020, May 17;158:104870 PMID: 32434052
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AMPK activator
PF-06409577 is orally bioavailable AMPK activator with EC50 of 7 nM for α1β1γ1 in the TR-FRET assay and it shows no detectable inhibition of hERG in a patch-clamp assay (100 μM) and was not an inhibitor (IC50 > 100 μM) of the microsomal activities of major human cytochrome P450 isoforms. -
AMPK activator
7-Methoxyisoflavone is an isoflavone derivative and also an activator of adenosine monophosphate-activated protein kinase (AMPK).
