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Cannabinoid Receptors



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Catalog No. Product Name Application Product Information
A11096 SALE

UR-144

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UR-144 is a potent synthetic cannabinoid (CB) which preferentially binds the peripheral CB2 receptor (Ki = 1.8 nM) over the central CB1 receptor (Ki = 150 nM).
A16328

Bay 59-3074

CB1/CB2 receptor agonist
Bay 59-3074 is a novel, selective CB1/CB2 receptor partial agonist with Ki values of 48.3 and 45.5 nM at human CB1 and CB2 receptors respectively .
A14993 SALE

AM630

CB2 antagonist
AM630 is a selectivity CB2 antagonist with Ki of 31.2 nM, > 150 fold selectivity over CB1 receptor.
A15200 SALE

Otenabant

CB1 receptor antagonist
Otenabant is a recently discovered selective, high affinity, competitive CB1 receptor antagonist with Ki of 0.7 nM.
A14110

PB-22

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PB-22 is an analog of JWH 018 which differs by having 8-hydroxyquinoline replacing the naphthalene group of JWH 018.
A14189

Tedalinab

CB2 receptor agonist
Tedalinab (GRC-10693) is a drug developed for the treatment of osteoarthritis and neuropathic pain, which acts as a potent and selective cannabinoid CB2 receptor agonist. It has a very high selectivity of 4700x for CB2 over the related CB1 receptor, has good oral bioavailability and has shown promising safety results and effective analgesic and antiinflammatory actions in early clinical trials.
A14174

AM 2201

Cannabinoid inhibitor
AM2201 is a potent synthetic cannabinoid (CB) with Ki values of 1.0 and 2.6 nM for the CB1 and CB2 receptors, respectively
A12914 SALE

AM251

CB1 receptor antagonist
AM251 is a potent CB1 receptor antagonist (IC50 = 8 nM, Ki = 7.49 nM) that displays 306-fold selectivity over CB2 receptors.
A11513

Org 27569

CB1 modulator‎
Org 27569 is a potent CB1 receptor allosteric modulator (pEC50 = 8.24).
A11547 SALE

Rimonabant (SR141716)

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Rimonabant is a selective antagonist of CB1 with IC50 of 13.6 nM and EC50 of 17.3 nM in hCB1 transfected HEK 293 membrane.
A11253

GW842166X

CB2 receptor agonist
GW842166X is a selective non-cannabinoid CB2 receptor agonist, which is undergoing clinical development as a novel oral treatment for inflammatory pain
A11942

CP 945598 HCl (Otenabant HCl)

CB1 antagonist
CP 945598 is a potent and highly selective CB1 antagonist.
A11939

MDA 19

CB2 agonist
MDA 19 is a potent and selective agonist for the cannabinoid receptor CB2, with reasonable selectivity over the psychoactive CB1 receptor.
A11938

BML-190

CB2 receptor ligand
BML-190 is a selective inverse agonist of the human cannabinoid CB2 receptor.
A11932 SALE

WIN 55,212-2 mesylate

CB receptor agonist
WIN 55,212-2 is a potent cannabinoid receptor agonist that has been found to be a potent analgesic in a rat model of neuropathic pain. It activates p42 and p44 MAP kinase via receptor-mediated signaling.
A16397

AM1241

CB2 receptor agonist
AM1241 is a selective cannabinoid CB2 receptor agonist with Ki of 3.4 nM, exhibits 82-fold selectivity over CB1 receptor.

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