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| Catalog No. | Inhibitor Name | CaMKII | CaMKIII | CaMKKα | CaMKKβ | Other |
|---|---|---|---|---|---|---|
| A14307 | NH125 | **** | PKC,PKA | |||
| A11473 | KN-62 | ** | ||||
| A14288 | KN-93 Phosphate | *** | ||||
| A16345 | STO-609 acetate | *** | **** | |||
| A13804 | CID 755673 | * | PKD1, PKD2, PKD3, PKC, CAK, PLK1, Akt | |||
| A13447 | A-484954 | *** |
Notes:
1.Hover mouse over "" to view the IC50 value.(A few compounds have proven potency but without published IC50 data.)
2.For more details about the compound, click on the product name of your interest.
3.The higher the number of "" is, the more potent the inhibitor or activator is.
4."" refers to compounds which do inhibitory effects on the related isoform, but without specific value.
17 Item(s)
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CaMKII-IN-1
Catalog No. A21034 CaMKII inhibitorCaMKII-IN-1 is a potent and highly selective CaMKII inhibitor with IC50 of 63 nM. Learn More -
K252a
Catalog No. A13897 CaMK/Phosphorylase inhibitorK252a is a highly potent cell permeable inhibitor of CaM kinase and phosphorylase kinase (IC50 = 1.8 and 1.7 nmol/L, respectively). Learn More -
STO-609 acetate
Catalog No. A16345 CaMKK inhibitorSTO-609 is a cell-permeable inhibitor of calcium/calmodulin-dependent kinase kinases (CaMKK) isoforms CaMKKα and CaMKKβ (Ki = 80 and 15 ng/ml, respectively). Learn More -
CRT-0066101
Catalog No. A16318 PKD InhibitorCRT-0066101, potent inhibitor of protein kinase D (PKD); inhibits all PKD isoforms (IC50 values are 1, 2 and 2.5 nM for PKD1, PKD3 and PKD2 respectively). Learn More -
CID 797718
Catalog No. A13809 PKD1 inhibitorCID797718 is a structural analog of CID755673 (Adooq Catalog No. A13804). It was a 10-time less potent PKD1 inhibitor with an IC50 value of 7.0 +/-0.8 uM. Learn More -
KN-92 phosphate
Catalog No. A15139 CaMKII inhibitorKN-92 is an inactive derivative of KN-93. KN-93 is a selective inhibitor of Ca2+/calmodulin-dependent kinase II (CaMKII), competitively blocking CaM binding to the kinase (Ki = 370 nM). Learn More -
KN-92 hydrochloride
Catalog No. A15138 -
KN-92
Catalog No. A15137 CaMK-II InhibitorKN-92 is an inactive derivative of KN-93. KN-93 is a selective inhibitor of Ca2+/calmodulin-dependent kinase II (CaMKII), competitively blocking CaM binding to the kinase (Ki = 370 nM). Learn More -
A-484954
Catalog No. A13447 eEF2K (CAMKIII) inhibitorA-484954 is a potent, selective inhibitor of eukaryotic longation factor-2 kinase (eEF2K). Learn More -
KN-62
Catalog No. A11473 CaM kinase II inhibitorKN-62 is a selective, cell-permeable inhibitor of CaM kinase II. Learn More -
NH125
Catalog No. A14307 -
KN-93 Phosphate
Catalog No. A14288 CaMKII inhibitorKN-93 Phosphate is a potent and specific inhibitor of Ca2+/calmodulin-dependent protein kinase II (CaMKII) with Ki of 0.37 μM, no remarkable inhibitory effects on APK, PKC, MLCK or Ca2+-PDE activities. Learn More -
CID 755673
Catalog No. A13804 PKD inhibitorCID755673 is a potent PKD inhibitor with IC50s of 182 nM, 280 nM and 227 nM for PKD1, PKD2 and PKD3, respectively. Learn More -
KN-93
Catalog No. A13276 CaM kinase II inhibitorKN-93 is an inhibitor of multifunctional Ca++/calmodulin-dependent protein kinase. Learn More -
Phenoxybenzamine hydrochloride
Catalog No. A10719 α-adrenergic (AR) antagonist/CaM inhibitorPhenoxybenzamine is a cell-permeable, non-specific, irreversible α-adrenergic (AR) antagonist that also acts as an CaM inhibitor. Learn More -
kb NB 142-70
Catalog No. A12423 PKD inhibitorkb NB 142-70 is a selective protein kinase D (PKD) inhibitor (IC50 values are 28.3, 58.7 and 53.2 nM for PKD1, 2 and 3 respectively). Learn More -
CID 2011756
Catalog No. A12416 PKD inhibitorCID 2011756 is a protein kinase D (PKD) inhibitor (IC50 values are 0.6, 0.7 and 3.2 μM for PKD2, PKD3 and PKD1 respectively). Learn More
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