CaMK

Catalog No.Inhibitor Name CaMKIICaMKIIICaMKKαCaMKKβOther
A14307NH125
****
PKC,PKA
A11473KN-62
**
A14288KN-93 Phosphate
***
A16345STO-609 acetate
***
****
A13804CID 755673
*
PKD1, PKD2, PKD3, PKC, CAK, PLK1, Akt
A13447A-484954
***

Notes:
1.Hover mouse over " * " to view the IC50 value.(A few compounds have proven potency but without published IC50 data.)
2.For more details about the compound, click on the product name of your interest.
3.The higher the number of " * " is, the more potent the inhibitor or activator is.
4."" refers to compounds which do inhibitory effects on the related isoform, but without specific value.

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  1. KN-62

    Catalog No. A11473
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    CaM kinase II inhibitor
    KN-62 is a selective, cell-permeable inhibitor of CaM kinase II. Learn More
  2. CRT-0066101

    Catalog No. A16318
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    PKD Inhibitor
    CRT-0066101, potent inhibitor of protein kinase D (PKD); inhibits all PKD isoforms (IC50 values are 1, 2 and 2.5 nM for PKD1, PKD3 and PKD2 respectively). Learn More
  3. CID 797718

    Catalog No. A13809
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    PKD1 inhibitor
    CID797718 is a structural analog of CID755673 (Adooq Catalog No. A13804). It was a 10-time less potent PKD1 inhibitor with an IC50 value of 7.0 +/-0.8 uM. Learn More
  4. KN-92 phosphate

    Catalog No. A15139
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    CaMKII inhibitor
    KN-92 is an inactive derivative of KN-93. KN-93 is a selective inhibitor of Ca2+/calmodulin-dependent kinase II (CaMKII), competitively blocking CaM binding to the kinase (Ki = 370 nM). Learn More
  5. KN-92 hydrochloride

    Catalog No. A15138
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    CaMK-II Inhibitor
    KN-92 hydrochloride is a negative control for KN-93. Learn More
  6. KN-92

    Catalog No. A15137
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    CaMK-II Inhibitor
    KN-92 is an inactive derivative of KN-93. KN-93 is a selective inhibitor of Ca2+/calmodulin-dependent kinase II (CaMKII), competitively blocking CaM binding to the kinase (Ki = 370 nM). Learn More
  7. A-484954

    Catalog No. A13447
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    eEF2K (CAMKIII) inhibitor
    A-484954 is a potent, selective inhibitor of eukaryotic longation factor-2 kinase (eEF2K). Learn More
  8. K252a

    Catalog No. A13897
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    CaMK/Phosphorylase inhibitor
    K252a is a highly potent cell permeable inhibitor of CaM kinase and phosphorylase kinase (IC50 = 1.8 and 1.7 nmol/L, respectively). Learn More
  9. NH125

    Catalog No. A14307
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    eEF-2 inhibitor
    NH125 is a selective eEF-2 kinase inhibitor. Learn More
  10. KN-93 Phosphate

    Catalog No. A14288
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    CaMKII inhibitor
    KN-93 Phosphate is a potent and specific inhibitor of Ca2+/calmodulin-dependent protein kinase II (CaMKII) with Ki of 0.37 μM, no remarkable inhibitory effects on APK, PKC, MLCK or Ca2+-PDE activities. Learn More
  11. CID 755673

    Catalog No. A13804
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  12. KN-93

    Catalog No. A13276
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    CaM kinase II inhibitor
    KN-93 is an inhibitor of multifunctional Ca++/calmodulin-dependent protein kinase. Learn More
  13. Phenoxybenzamine hydrochloride

    Catalog No. A10719
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    α-adrenergic (AR) antagonist/CaM inhibitor
    Phenoxybenzamine is a cell-permeable, non-specific, irreversible α-adrenergic (AR) antagonist that also acts as an CaM inhibitor. Learn More
  14. kb NB 142-70

    Catalog No. A12423
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    PKD inhibitor
    kb NB 142-70 is a selective protein kinase D (PKD) inhibitor (IC50 values are 28.3, 58.7 and 53.2 nM for PKD1, 2 and 3 respectively). Learn More
  15. CID 2011756

    Catalog No. A12416
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    PKD inhibitor
    CID 2011756 is a protein kinase D (PKD) inhibitor (IC50 values are 0.6, 0.7 and 3.2 μM for PKD2, PKD3 and PKD1 respectively). Learn More
  16. STO-609 acetate

    Catalog No. A16345
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    CaMKK inhibitor
    STO-609 is a cell-permeable inhibitor of calcium/calmodulin-dependent kinase kinases (CaMKK) isoforms CaMKKα and CaMKKβ (Ki = 80 and 15 ng/ml, respectively). Learn More

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