NMDA Receptors

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  1. Flupirtine maleate

    Catalog No. A10251
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    NMDA antagonist
    Non-opioid analgesic with muscle relaxant properties. Learn More
  2. Eliprodil

    Catalog No. A12946
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    NMDA antagonist
    Eliprodil is a non-competitive NR2B-NMDA receptor antagonist(IC50=1 uM), less potent for NR2A- and NR2C-containing receptors(IC50> 100 uM). Learn More
  3. CGS19755

    Catalog No. A15791
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    NMDA antagonist
    CGS 19755 (cis-4-phosphonomethyl-2-piperidine carboxylic acid) was found to be a potent, stereospecific inhibitor of N-methyl-D-aspartate (NMDA)-evoked, but not KCl-evoked, [3H] acetylcholine release from slices of the rat striatum. Learn More
  4. (+)-MK 801 Maleate

    Catalog No. A12761
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    NMDA receptor antagonist
    (+)-MK 801 is a potent antagonist of NMDA with Ki value of 30.5nM. Learn More
  5. L-701324

    Catalog No. A15522
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    NMDA/glycine receptor antagonist
    L-701324 is an orally active and long acting anticonvulsant with high affinity and selectivity for the glycine site on the NMDA receptor, Learn More
  6. SDZ 220-581 Ammonium salt

    Catalog No. A15235
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    NMDA receptor antagonist
    SDZ 220-581 ammonium salt is a potent, competitive antagonist at the NMDA glutamate receptor subtype(pKi= 7.7). Learn More
  7. (-)-MK 801 maleate

    Catalog No. A13435
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    NMDA receptor antagonist.
    (-)-MK 801 maleate acts as a potent, selective, and non-competitive NMDA receptor antagonist. It acts by binding to a site located within the NMDA associated ion channel. Learn More
  8. TCN 201

    Catalog No. A11947
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    NMDA Receptor Antagonist
    TCN 201 is a NMDA receptor antagonist selective for NR1/NR2A over NR1/NR2B-containing receptors Learn More
  9. SDZ 220-581

    Catalog No. A12426
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    NMDA receptor antagonist
    SDZ 220-581 is a competitive NMDA receptor antagonist (pKi = 7.7). Learn More
  10. NMDA

    Catalog No. A12751
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    NMDA receptor agonist
    NMDA is a prototypic NMDA receptor agonist. Learn More
  11. Ro 25-6981 maleate

    Catalog No. A13144
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    NMDA receptors Blocker
    Ro 25-6981 is a high-affinity, potent and selective blocker of N-methyl- D-aspartate (NMDA) receptors. Learn More
  12. CNQX

    Catalog No. A16109
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    AMPA/kainate antagonist
    CNQX is a competitive, non-NMDA glutamate receptor antagonist (IC50s = 0.3 and 1.5 uM for AMPA and kainate receptors, respectively, versus IC50 = 25 uM for NMDA receptors). Learn More
  13. 7CKA

    Catalog No. A17070
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    NMDA receptor antagonist
    7CKA is a NMDA receptor antagonist that acts at the glycine site. Learn More
  14. RO 25-6981 maleate

    Catalog No. A16083
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    NMDA receptors blocker
    Ro 25-6981 Maleate is a potent and selective activity-dependent blocker of NMDA receptors containing the NR2B subunit. IC50 values are 0.009 and 52 uM for cloned receptor subunit combinations NR1C/NR2B and NR1C/NR2A respectively. Learn More
  15. D-AP5

    Catalog No. A17044
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    NMDA antagonist
    D-AP5 is a selective N-methyl-D-aspartate (NMDA) receptor antagonist that competitively inhibits the glutamate binding site of NMDA receptors. Learn More
  16. Memantine hydrochloride

    Catalog No. A11708
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    NMDA receptor antagonist
    Memantine hydrochloride is an antagonist at the NMDA receptor, binding to the ion channel site. it was used in the treatment of Parkinsonism. Learn More
  17. Orphenadrine citrate

    Catalog No. A11712
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    Orphenadrine is known to have the following pharmacology: mACh receptor antagonist (anticholinergic); H1 receptor antagonist (antihistamine); NMDA receptor antagonist; NET blocker (norepinephrine reuptake inhibitor); Nav1.7, Nav1.8, and Nav1.9 sodium channel blocker; HERG potassium channel blocker. Learn More
  18. MDL 29951

    Catalog No. A13729
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    NMDA receptor antagonist
    MDL-29951 is a novel glycine antagonist of NMDA receptor activation (Ki=0.14 mM, [3H]glycine binding) in vitro and in vivo. Learn More
  19. CIQ

    Catalog No. A15523
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    NMDA receptors Potentiator
    CIQ is a subunit-selective potentiator of NMDA receptors containing the NR2C or NR2D subunit. Learn More
  20. Felbamate

    Catalog No. A11862
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    Felbamate is an antagonist at the NMDA-associated glycine binding site. Learn More
  21. Ibotenic Acid

    Catalog No. A14006
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    NMDA& mGlu receptor agonist
    Ibotenic acid is a neuroexcitatory amino acid originally isolated from Amanita species that functions as a NMDA and metabotropic glutamate receptor agonist. Learn More
  22. GLYX-13 (Rapastinel)

    Catalog No. A13576
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    NMDAR modulator
    GLYX-13 is a selective weak partial agonist of the glycine site of the NMDA receptor which is under development by Naurex as adjunctive therapy for treatment-resistant depression. Learn More
  23. ARL-15896

    Catalog No. A13858
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    NMDA receptor ion channel antagonist
    ARL-15896 is a novel N-methyl-D-aspartate receptor ion channel antagonist. Learn More
  24. NVP-AAM077 Tetrasodium Hydrate (PEAQX)

    Catalog No. A14071
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    NMDA receptors antagonist
    NVP-AAM077 inhibited progenitor cells proliferation in the subventricular zone and dentate gyrus and reduced the survival of newborn cells in the dentate gyrus in the adult mice. Learn More
  25. Neu-2000

    Catalog No. A17033
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    NMDA receptor antagonist
    Neu-2000 is a NMDA receptor antagonist potentially for the treatment of stroke. Learn More

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