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NMDA Receptors

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Catalog No. Product Name Application Product Information
A10251 SALE

Flupirtine maleate

NMDA antagonist
Non-opioid analgesic with muscle relaxant properties.

SDZ 220-581 Ammonium salt

NMDA receptor antagonist
SDZ 220-581 ammonium salt is a potent, competitive antagonist at the NMDA glutamate receptor subtype(pKi= 7.7).


NMDA/glycine receptor antagonist
L-701324 is an orally active and long acting anticonvulsant with high affinity and selectivity for the glycine site on the NMDA receptor,
A12761 SALE

(+)-MK 801 Maleate

NMDA receptor antagonist
(+)-MK 801 is a potent antagonist of NMDA with Ki value of 30.5nM.
A12751 SALE


NMDA receptor agonist
NMDA is a prototypic NMDA receptor agonist.


NMDA antagonist
CGS 19755 (cis-4-phosphonomethyl-2-piperidine carboxylic acid) was found to be a potent, stereospecific inhibitor of N-methyl-D-aspartate (NMDA)-evoked, but not KCl-evoked, [3H] acetylcholine release from slices of the rat striatum.

SDZ 220-581

NMDA receptor antagonist
SDZ 220-581 is a competitive NMDA receptor antagonist (pKi = 7.7).
A11947 SALE

TCN 201

NMDA Receptor Antagonist
TCN 201 is a NMDA receptor antagonist selective for NR1/NR2A over NR1/NR2B-containing receptors


NMDA antagonist
Eliprodil is a non-competitive NR2B-NMDA receptor antagonist(IC50=1 uM), less potent for NR2A- and NR2C-containing receptors(IC50> 100 uM).
A13435 SALE

(-)-MK 801 maleate

NMDA receptor antagonist.
(-)-MK 801 maleate acts as a potent, selective, and non-competitive NMDA receptor antagonist. It acts by binding to a site located within the NMDA associated ion channel.


NMDA receptors Potentiator
CIQ is a subunit-selective potentiator of NMDA receptors containing the NR2C or NR2D subunit.

RO 25-6981 maleate

NMDA receptors blocker
Ro 25-6981 Maleate is a potent and selective activity-dependent blocker of NMDA receptors containing the NR2B subunit. IC50 values are 0.009 and 52 uM for cloned receptor subunit combinations NR1C/NR2B and NR1C/NR2A respectively.

Ibotenic Acid

NMDA& mGlu receptor agonist
Ibotenic acid is a neuroexcitatory amino acid originally isolated from Amanita species that functions as a NMDA and metabotropic glutamate receptor agonist.
A13576 SALE

GLYX-13 (Rapastinel)

NMDAR modulator
GLYX-13 is a selective weak partial agonist of the glycine site of the NMDA receptor (IA approximately 25%) which is under development by Naurex as an adjunctive therapy for treatment-resistant depression.


NMDA receptor ion channel antagonist
ARL-15896 is a novel N-methyl-D-aspartate receptor ion channel antagonist.

NVP-AAM077 Tetrasodium Hydrate (PEAQX)

NMDA receptors antagonist
NVP-AAM077 inhibited progenitor cells proliferation in the subventricular zone and dentate gyrus and reduced the survival of newborn cells in the dentate gyrus in the adult mice.
A13729 SALE

MDL 29951

NMDA receptor antagonist
MDL-29951 is a novel glycine antagonist of NMDA receptor activation (Ki=0.14 mM, [3H]glycine binding) in vitro and in vivo.


Felbamate is an antagonist at the NMDA-associated glycine binding site.
A11712 SALE

Orphenadrine citrate

Orphenadrine is known to have the following pharmacology: mACh receptor antagonist (anticholinergic); H1 receptor antagonist (antihistamine); NMDA receptor antagonist; NET blocker (norepinephrine reuptake inhibitor); Nav1.7, Nav1.8, and Nav1.9 sodium channel blocker; HERG potassium channel blocker.
A11708 SALE

Memantine hydrochloride

NMDA receptor antagonist
Memantine hydrochloride is an antagonist at the NMDA receptor, binding to the ion channel site. it was used in the treatment of Parkinsonism.


AMPA/kainate antagonist
CNQX is a competitive, non-NMDA glutamate receptor antagonist (IC50s = 0.3 and 1.5 uM for AMPA and kainate receptors, respectively, versus IC50 = 25 uM for NMDA receptors).

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