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Rislenemdaz
Catalog No. A21907 NMDA receptor GluN2B antagonistRislenemdaz (CERC-301) is an orally bioavailable and selective N-methyl-D-aspartate (NMDA) receptor subunit 2B (GluN2B) antagonist with Ki and IC50 of 8.1 nM and 3.6 nM, respectively. Learn More -
Sarcosine
Catalog No. A16692 GlyT inhibitor/NMDA receptorSarcosine is a glycine transporter type 1 (GlyT) inhibitor and an N-methyl-D-aspartate (NMDA) receptor co-agonist at the glycine binding site. Learn More -
GV-196771A
Catalog No. A13438 NMDA receptor antagonistGV-196771A is the sodium salt form of GV196771, is an NMDA receptor antagonist. Learn More -
Flupirtine maleate
Catalog No. A10251 NMDA antagonistNon-opioid analgesic with muscle relaxant properties. Learn More -
Eliprodil
Catalog No. A12946 NMDA antagonistEliprodil is a non-competitive NR2B-NMDA receptor antagonist(IC50=1 uM), less potent for NR2A- and NR2C-containing receptors(IC50> 100 uM). Learn More -
CGS19755
Catalog No. A15791 NMDA antagonistCGS 19755 (cis-4-phosphonomethyl-2-piperidine carboxylic acid) was found to be a potent, stereospecific inhibitor of N-methyl-D-aspartate (NMDA)-evoked, but not KCl-evoked, [3H] acetylcholine release from slices of the rat striatum. Learn More -
(+)-MK 801 Maleate
Catalog No. A12761 NMDA receptor antagonist(+)-MK 801 is a potent antagonist of NMDA with Ki value of 30.5nM. Learn More -
RPR104632
Catalog No. A13385 NMDA receptor antagonistRPR104632 is a specific antagonist of NMDA receptor, with potent neuroprotective properties. Learn More -
L-701324
Catalog No. A15522 NMDA/glycine receptor antagonistL-701324 is an orally active and long acting anticonvulsant with high affinity and selectivity for the glycine site on the NMDA receptor, Learn More -
SDZ 220-581 Ammonium salt
Catalog No. A15235 NMDA receptor antagonistSDZ 220-581 ammonium salt is a potent, competitive antagonist at the NMDA glutamate receptor subtype(pKi= 7.7). Learn More -
(-)-MK 801 maleate
Catalog No. A13435 NMDA receptor antagonist.(-)-MK 801 maleate acts as a potent, selective, and non-competitive NMDA receptor antagonist. It acts by binding to a site located within the NMDA associated ion channel. Learn More -
Ifenprodil tartrate
Catalog No. A16583 NMDA receptor antagonistIfenprodil tartrate is the atypical N-methyl-D-aspartate (NMDA) receptor antagonist, inhibits NMDA-induced currents at NR1A/NR2B receptors with high affinity (IC50 = 0.34 μM). Learn More -
Transcrocetinate disodium
Catalog No. A21051 NMDA receptor antagonistTranscrocetinate disodium, extracted from saffron (Crocus sativus L.), acts as an NMDA receptor antagonist with high affinity. Learn More -
MDL 105519
Catalog No. A21192 NMDA receptor antagonistMDL 105519 is a potent and selective antagonist of glycine binding to the NMDA receptor. Learn More -
Radiprodil
Catalog No. A21193 NMDA NR2B antagonistRadiprodil (RGH-896) is an orally active and selective NMDA NR2B antagonist. A potential therapeutic agent in treatment of neuropathic pain and possibly other chronic pain conditions. Learn More -
DNQX
Catalog No. A13882 NMDA receptor antagonistDNQX is a non-N-methyl-D-aspartate (non-NMDA) receptor complex antagonist. Learn More -
NMDA-IN-1
Catalog No. A21419 NMDA antagonistNMDA-IN-1 is a potent and NR2B-selective NMDA antagonist with Ki of 0.85 nM. Learn More -
NMDA
Catalog No. A12751 NMDA receptor agonistNMDA is a prototypic NMDA receptor agonist. Learn More -
7-Chlorokynurenic acid sodium salt
Catalog No. A21879 NMDA receptor antagonist7-Chlorokynurenic acid sodium salt is a potent and selective antagonist of the glycine B coagonist site of the N-methyl-D-aspartate (NMDA) receptor (IC50=0.56 μM). Learn More -
SDZ 220-581
Catalog No. A12426 NMDA receptor antagonistSDZ 220-581 is a competitive NMDA receptor antagonist (pKi = 7.7). Learn More -
TCN 201
Catalog No. A11947 NMDA Receptor AntagonistTCN 201 is a NMDA receptor antagonist selective for NR1/NR2A over NR1/NR2B-containing receptors Learn More -
SDZ 220-581 hydrochloride, SDZ220-581, SDZ-220-581
Catalog No. A21897 NMDA receptor antagonistSDZ 220-581 hydrochloride is an orally active, potent, competitive NMDA receptor antagonist with pKi value of 7.7. Learn More -
RO 25-6981 maleate
Catalog No. A16083 NMDA receptors blockerRo 25-6981 Maleate is a potent and selective activity-dependent blocker of NMDA receptors containing the NR2B subunit. IC50 values are 0.009 and 52 uM for cloned receptor subunit combinations NR1C/NR2B and NR1C/NR2A respectively. Learn More -
GNE 0723
Catalog No. A12757 NMDAR modulatorGNE 0723 is a brain permeable positive allosteric modulator of NMDAR, with an EC50 of 21 nM for GluN2A, 7.4 and 6.2 μM for GluN2C and GluN2D, respectively. Learn More -
Glycine
Catalog No. A17936 NMDA antagonistAZD-4282, also known as aminoacetic acid and glycine, is a N-methyl-D-aspartate (NMDA) receptor antagonist potentially for the treatment of neuropathic pain. Learn More -
Mephenesin
Catalog No. A17493 NMDA receptor antagonistMephenesin is an NMDA receptor antagonist, is a centrally acting muscle relaxant. Learn More -
Neu-2000
Catalog No. A17033 NMDA receptor antagonistNeu-2000 is a NMDA receptor antagonist potentially for the treatment of stroke. Learn More -
D-AP5
Catalog No. A17044 NMDA antagonistD-AP5 is a selective N-methyl-D-aspartate (NMDA) receptor antagonist that competitively inhibits the glutamate binding site of NMDA receptors. Learn More -
7CKA
Catalog No. A17070 NMDA receptor antagonist7CKA is a NMDA receptor antagonist that acts at the glycine site. Learn More -
Ro 25-6981 maleate
Catalog No. A13144 NMDA receptors BlockerRo 25-6981 is a high-affinity, potent and selective blocker of N-methyl- D-aspartate (NMDA) receptors. Learn More -
CNQX
Catalog No. A16109 AMPA/kainate antagonistCNQX is a competitive, non-NMDA glutamate receptor antagonist (IC50s = 0.3 and 1.5 uM for AMPA and kainate receptors, respectively, versus IC50 = 25 uM for NMDA receptors). Learn More -
CIQ
Catalog No. A15523 NMDA receptors PotentiatorCIQ is a subunit-selective potentiator of NMDA receptors containing the NR2C or NR2D subunit. Learn More -
Ibotenic Acid
Catalog No. A14006 NMDA& mGlu receptor agonistIbotenic acid is a neuroexcitatory amino acid originally isolated from Amanita species that functions as a NMDA and metabotropic glutamate receptor agonist. Learn More -
GLYX-13 (Rapastinel)
Catalog No. A13576 NMDAR modulatorGLYX-13 is a selective weak partial agonist of the glycine site of the NMDA receptor which is under development by Naurex as adjunctive therapy for treatment-resistant depression. Learn More -
ARL-15896
Catalog No. A13858 NMDA receptor ion channel antagonistARL-15896 is a novel N-methyl-D-aspartate receptor ion channel antagonist. Learn More -
NVP-AAM077 Tetrasodium Hydrate (PEAQX)
Catalog No. A14071 NMDA receptors antagonistNVP-AAM077 inhibited progenitor cells proliferation in the subventricular zone and dentate gyrus and reduced the survival of newborn cells in the dentate gyrus in the adult mice. Learn More -
MDL 29951
Catalog No. A13729 NMDA receptor antagonistMDL-29951 is a novel glycine antagonist of NMDA receptor activation (Ki=0.14 mM, [3H]glycine binding) in vitro and in vivo. Learn More -
Felbamate
Catalog No. A11862 Felbamate is an antagonist at the NMDA-associated glycine binding site. Learn More -
Orphenadrine citrate
Catalog No. A11712 NMDA receptor antagonistOrphenadrine citrate is a NMDA receptor antagonist with Ki of 6.0 +/- 0.7 μM, HERG potassium channel blocker. Learn More -
Memantine hydrochloride
Catalog No. A11708 NMDA receptor antagonistMemantine hydrochloride is an antagonist at the NMDA receptor, binding to the ion channel site. it was used in the treatment of Parkinsonism. Learn More
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