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$0.00 Opioid Receptors
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AR-M 1000390 hydrochloride
Catalog No. A21911 δ opioid receptor agonistAR-M 1000390 hydrochloride is an exceptionally selective, potent δ opioid receptor agonist with an EC50 of 7.2??0.9 nM for δ agonist potency. Learn More -
GSK1521498 free base (hydrochloride)
Catalog No. A21792 μ-opioid receptor (MOR) antagonistGSK1521498 free base (hydrochloride) is a potent and selective μ-opioid receptor (MOR) antagonist. Learn More -
CYT-1010 hydrochloride
Catalog No. A21348 mu-opioid receptor agonistCYT-1010 hydrochloride is a mu-opioid receptor agonist extracted from patent WO2013173730A2, with EC50s of 13.1 nM and 0.0053 nM on beta-arrestin recruitment and inhibition of cAMP production, respectively. Learn More -
JDTic
Catalog No. A11468 κ-opioid receptor antagonistJDTic is a highly selective antagonist for the κ-opioid receptor; without affecting the μ- or δ-opioid receptors. Learn More -
DPI-3290
Catalog No. A13699 opioid receptors agonistDPI-3290 (Org 41793) is a potent and specific opioid receptors agonist with Ki values of 0.18 nM, 0.46 nM, and 0.62 nM for δ-, μ-, and κ-opioid receptors, respectively. Learn More -
GSK1521498 free base
Catalog No. A18994 μ-opioid receptor antagonistGSK1521498 free base is a potent and selective μ-opioid receptor (MOR) antagonist. GSK1521498 free base is being used for the treatment of disorders of compulsive consumption of food, alcohol, and drugs. Learn More -
LY2795050
Catalog No. A15149 k-opioid receptor antagonistLY2795050 is a novel selective κ-opioid Receptor (KOR) antagonist (IC50=0.72 nM) and has the potential as a PET tracer to image KOR in vivo. Learn More -
Methylnaltrexone Bromide
Catalog No. A15159 μ-opioid antagonistMethylnaltrexone Bromide is a pheriphally-acting µ-opioid antagonist that acts on the gastrointestinal tract to decrease opioid-induced constipation. Learn More -
Alvimopan dihydrate
Catalog No. A14991 µ-opioid receptor agonistAlvimopan dihydrate(LY 246736, ADL 8-2698) is a peripherally acting mu-opioid receptor (PAM-OR, IC50= 1.7 nM) antagonist for accelerating gastrointestinal recovery after surgery. Learn More -
BTRX-335140
Catalog No. A18583 κ opioid receptor antagonistBTRX-335140 (CYM-53093) is a potent and selective, orally active κ opioid receptor (KOR) antagonist, has antagonist activity for κOR, μOR and δOR with IC50 values of 0.8 nM, 110 nM, and 6500 nM, respectively. Learn More -
Trimebutine maleate
Catalog No. A18115 µ- opioid receptor agonistTrimebutine Maleate is a drug with antimuscarinic and weak mu opioid agonist effects. Trimebutine Maleate modulates the calcium and potassium channels, relieves abdominal pain in patients with irritable bowel syndrome. Learn More -
Bevenopran
Catalog No. A17110 opioid receptor antagonisBevenopran, also known as CB-5945, ADL-5945, MK-2402, OpRA III, is a peripherally selective μ- and δ-opioid receptor antagonist. Learn More -
Cebranopadol (GRT-6005)
Catalog No. A12670 Opioid Receptor AgonistCebranopadol is a potent nociceptin/orphanin FQ peptide (NOP) and opioid receptor agonist Learn More -
Docusate Sodium
Catalog No. A16155 Docusate Sodium is a laxative used to treat constipation, for constipation due to the use of opiates it maybe used with a stimulant laxative, can be taken by mouth or rectally. Learn More -
Naloxegol Oxalate
Catalog No. A15972 Opioid antagonistNaloxegol is a peripherally-selective opioid antagonist for the treatment of opioid-induced constipation. Learn More -
Alvimopan monohydrate
Catalog No. A14992 µ-opioid receptor agonistAlvimopan monohydrate is a peripherally acting mu-opioid receptor (PAM-OR, IC50= 1.7 nM) antagonist for accelerating gastrointestinal recovery after surgery. Learn More -
ADL5859 HCl
Catalog No. A11072 Opioid Receptor agonistADL5859 HCl is a highly potent and selective δ opioid receptor agonist with Ki value to be 0.84 nM and ED50 value to be 20 nM. Learn More -
ADL5747
Catalog No. A13479 δ opioid receptor agonistADL5747 is a selective, nonpeptidic δ opioid receptor agonist. Learn More -
U-69593
Catalog No. A14187 κ1-opioid receptor agonistU-69593 is a potent, selective κ1-opioid receptor agonist (EC50 = 80-109 nM). Active in vivo. Antinociceptive. Learn More -
Nalmefene hydrochloride
Catalog No. A13843 dopamine receptor agonistNalmefene hydrochloride is an opioid receptor antagonist. Learn More -
Nalfurafine hydrochloride
Catalog No. A12579 opioid κ-selective agonistNalfurafine hydrochloride is a kappa-opioid receptor agonist Learn More -
Trimebutine
Catalog No. A11718 Trimebutine is a drug with antimuscarinic and weak mu opioid agonist effects. Learn More -
BAN ORL 24
Catalog No. A11322 NOP antagonistBAN ORL 24 is a potent and selective NOP receptor antagonist. Learn More -
Alvimopan (ADL 8-2698)
Catalog No. A11292 Opioid antagonistAlvimopan behaves as a peripherally acting μ-opioid antagonist. Alvimopan competitively binds to mu-opioid receptor in the gastrointestinal tract. Learn More -
BRL 52537 HCl
Catalog No. A11210 Opioid Receptors agonistBRL 52537 hydrochloride is a highly selective and potent κ-opioid agonist (Ki = 0.24 nM). Learn More -
MCOPPB 3HCl
Catalog No. A10561 NOP receptor agonistMCOPPB is a compound which acts as a potent and selective agonist for the nociceptin receptor, with a pKi of 10.07. Learn More -
JTC-801
Catalog No. A11076 Opioid Receptor antagonistJTC-801 is a selective antagonist for the nociceptin receptor, also known as the ORL-1 receptor. Learn More
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