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| Catalog No. | Inhibitor Name | P-gp | Other |
|---|---|---|---|
| A10549 | Zosuquidar 3HCl | ** | |
| A11584 | Tariquidar | *** | |
| A12324 | Elacridar (GF120918) | BCRP |
Notes:
1.Hover mouse over "" to view the IC50 value.(A few compounds have proven potency but without published IC50 data.)
2.For more details about the compound, click on the product name of your interest.
3.The higher the number of "" is, the more potent the inhibitor or activator is.
4."" refers to compounds which do inhibitory effects on the related isoform, but without specific value.
19 Item(s)
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P-gp inhibitor 1
Catalog No. A13384 P-gp inhibitorP-gp inhibitor 1 is a novel inhibitor reversing P-glycoprotein-mediated multidrug resistance. Learn More -
Norverapamil hydrochloride
Catalog No. A12249 P-gp inhibitorNorverapamil hydrochloride ((±)-Norverapamil hydrochloride), an N-demethylated metabolite of Verapamil, is a L-type calcium channel blocker and a P-glycoprotein (P-gp) function inhibitor. Learn More -
TTT-28
Catalog No. A13033 ABCB1 (P-gp/MDR1) inhibitorTTT-28 is a synthesized thiazole-valine peptidomimetic, a novel selective inhibitor of ABCB1 (P-gp/MDR1) with high efficacy and low toxicity. Learn More -
Zosuquidar
Catalog No. A15289 P-gp inhibitorZosuquidar is a potent modulator of P-glycoprotein-mediated multi-drug resistance with Ki of 60 nM. Learn More -
Elacridar hydrochloride
Catalog No. A15077 P-gp inhibitorElacridar hydrochloride is a P-glycoprotein inhibitor, and has been used both in vitro and in vivo as a tool inhibitor of P-glycoprotein (Pgp) to investigate the role of transporters in the disposition of various test molecules. Learn More -
Biricodar dicitrate (VX-710 dicitrate)
Catalog No. A13533 P-gp modulatorBiricodar dicitrate (VX-710 dicitrate) is a modulator of P-glycoprotein and MRP-1; shows effective chemosensitizing activity in multidrug resistant cells. Learn More -
Biricodar
Catalog No. A21464 P-glycoprotein/MRP-1 modulatorBiricodar (VX-710) is a modulator of P-glycoprotein and MRP-1; shows effective chemosensitizing activity in multidrug resistant cells. Learn More -
FD 12-9
Catalog No. A18393 P-gp/BCRP dual inhibitorFD 12-9 is a flavonoid dimer, acts as a dual inhibitor of P-gp and BCRP, with EC50s of 285 nM and 0.9 nM, respectively. Anti-glioblastoma activity. Learn More -
KS-176
Catalog No. A16195 BCRP inhibitorKS-176 is a potent and selective inhibitor of the breast cancer resistance protein (BCRP) multidrug transporter (IC50 values are 0.59 and 1.39 uM in Pheo A and Hoechst 33342 assays respectively). Learn More -
MC 70 HCl
Catalog No. A16080 -
LY335979 (Zosuquidar 3HCl)
Catalog No. A10549 P-gp modulatorLY335979 (Zosuquidar trihydrochloride) is a potent highly selective P-gp inhibitor. Learn More -
Laniquidar
Catalog No. A13532 P-gp inhibitorLaniquidar is a third-generation P-gp inhibitor, which has been used in clinic trials for modulating multidrug resistance transporters. Learn More -
ONT-093
Catalog No. A13531 P-gp inhibitorONT-093 is an orally bioavailable P-glycoprotein pump inhibitor, for the potential reversal of multidrug resistance in patients undergoing cancer chemotherapy. Learn More -
XR9576
Catalog No. A13961 P-glycoprotein inhibitorXR9576 is a P-glycoprotein inhibitor undergoing research as an adjuvant against multidrug resistance in cancer Learn More -
Cynarin
Catalog No. A12004 Cynarin is a phenolic compound found in artichoke. It has antioxidant and choleretic properties. It is a potential immunosuppressive agent. Learn More -
Selamectin
Catalog No. A12363 Selamectin is a topical parasiticide and antihelminthic used on dogs and cats to treat and prevent infections of heartworms, fleas, ear mites, sarcoptic mange, and certain types of ticks in dogs as well as prevent heartworms, fleas, ear mites, hookworms, and roundworms in cats. Learn More -
Tariquidar (XR9576)
Catalog No. A11584 P-gp inhibitorTariquidar (XR9576) is a P-glycoprotein drug efflux pump inhibitor. Learn More -
Elacridar (GF120918)
Catalog No. A12324 P-gp & BCRP inhibitorElacridaris a prototypical BCRP inhibitor which inhibits the Bcrp1-mediated transport. Learn More -
PSC-833 (Valspodar)
Catalog No. A11080 MDR1/P-gp InhibitorPSC-833 is a kind of P-glycoprotein (P-gp) modulator that inhibits P-gp-mediated multidrug-resistance (MDR). Learn More
19 Item(s)
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