Prostanoid Receptors

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  1. Treprostinil sodium

    Catalog No. A21046
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    DP1/EP2 agonist
    Treprostinil sodium is a potent DP1 and EP2 agonist with EC50 values of 0.6??0.1 and 6.2??1.2 nM, respectively. Learn More
  2. Benorylate

    Catalog No. A17501
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    Prostaglandin Receptor inhibitor
    Benorilate, also known as Win-11450, is an ester of aspirin and paracetamol with analgesic, antipyretic, and anti-inflammatory activity used in the treatment of rheumatoid diseases. Benorilate has less severe side effects than aspirin. Learn More
  3. Dinoprost tromethamine

    Catalog No. A17505
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    Prostaglandin Receptor inhibitor
    Dinoprost Tromethamine, also known as Dinoprost Trometamol, is a naturally occurring prostaglandin used in medicine to induce labor and as an abortifacient. Learn More
  4. GSK726701A

    Catalog No. A20101
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    EP4 partial agonist
    GSK726701A is a novel prostaglandin E2 receptor 4 (EP4) partial agonist with a pEC50 of 7.4. Learn More
  5. Aligeron

    Catalog No. A13241
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    prostaglandin (PG) antagonist
    Aligeron is a non-selective prostaglandin (PG) antagonist, and has vasodilatory properties. Learn More
  6. CAY10471 Racemate

    Catalog No. A11760
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    Prostaglandin D2 receptor CRTH2 antagonist
    CAY10471 Racemate (TM30089 Racemate) is a potent and highly selective prostaglandin D2 receptor CRTH2 antagonist. Learn More
  7. ONO-AE3-208

    Catalog No. A11516
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    EP4 antagonist
    ONO-AE3-208 is an EP4 antagonist, and suppresses cell invasion, migration, and metastasis of prostate cancer. Learn More
  8. (+)-Cloprostenol

    Catalog No. A12979
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    prostaglandin F2α (PGF2α) analogue
    (+)-Cloprostenol is a prostaglandin F2α (PGF2α) analogue, and shows selective agonistic activity at the prostaglandin receptor. Learn More
  9. MK-2894 sodium salt

    Catalog No. A11498
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    EP4 antagonist
    MK-2894 sodium salt is a highly potent and selective second generation EP4 antagonist. Learn More
  10. Terutroban

    Catalog No. A20884
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    thromboxane-prostaglandin receptor antagonist
    Terutroban is a thromboxane-prostaglandin receptor antagonist. Learn More
  11. AGN 210676

    Catalog No. A21281
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    prostaglandin EP2 agonist
    AGN 210676 is a selective prostaglandin EP2 agonist extracted from patent US20070203222A1, Compound example 23, has an EC50 of 5 nM. Learn More
  12. CJ-42794

    Catalog No. A21948
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    EP4 antagonist
    CJ-42794 is a selective prostaglandin E receptor subtype 4 (EP4) antagonist, inhibits [3H]-PGE2 binding to the human EP4 receptor with a mean pKi of 8.5, a binding affinity that was at least 200-fold more selective for the human EP4 receptor than other human EP receptor subtypes (EP1, EP2, and EP3). Learn More
  13. Tafluprost

    Catalog No. A17442
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    prostaglandin analogue
    Tafluprost, also known as MK2452 and AFP-168, is a prostaglandin analogue used topically (as eye drops) to control the progression of glaucoma and in the management of ocular hypertension. Learn More
  14. GSK-269984A

    Catalog No. A17096
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    EP1 receptor antagonist
    GSK-269984A is a novel EP1 receptor antagonist. Learn More
  15. Grapiprant (CJ-023423)

    Catalog No. A15964
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    prostaglandin EP4 receptor antagonist
    Grapiprant is a novel, potent and selective prostaglandin EP4 receptor antagonist with antihyperalgesic properties. Learn More
  16. Ozagrel hydrochloride

    Catalog No. A11742
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    Thromboxane A2 synthesis inhibitor
    Ozagrel is an antiplatelet agent working as a thromboxane A2 synthesis inhibitor. Learn More
  17. MK-2894

    Catalog No. A11497
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    EP4 receptor antagonist
    MK-2894 is a highly potent and selective second generation EP4 antagonist. Learn More
  18. Cloprostenol (sodium salt)

    Catalog No. A13498
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    Cloprostenol is a synthetic analog of prostaglandin F2α (PGF2α). It is 200 times and 100 times more potent than PGF2α in terminating pregnancy in hamsters and rats, respectively, without the side effects associated with PGF2α. Learn More
  19. BAY-u 3405

    Catalog No. A13751
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    dual antagonist of TP/DP2
    BAY-u 3405 is an approved human medication for the treatment of allergic rhinitis that has documented activity as an antagonist of the thromboxane receptor (TP receptor). Learn More
  20. NS-304 (Selexipag)

    Catalog No. A13880
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    prostacyclin receptor agonist
    NS-304 is a selective prostacyclin IP1 receptor agonist (Ki values are 260 and 2100 nM and for human and rat IP receptors, and >10 μM for EP1-4, DP, FP, and TP receptors). Learn More
  21. Saikosaponin B2

    Catalog No. A14600
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    Prostanoid activator
    Saikosaponin B2 is a saponin activator. Learn More
  22. GW627368

    Catalog No. A15525
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    EP4 receptor antagonist
    GW627368 is a novel, potent and selective competitive antagonist of prostanoid EP4 receptor(Ki= 100 nM) with additional human TP receptor affinity(Ki= 150 nM). Learn More
  23. MF498

    Catalog No. A15532
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    EP4 receptor antagonist
    MF498 is a novel and selective E prostanoid receptor 4 (EP4 receptor) antagonist, displayed strong binding affinity for the EP4 receptor with Ki of 0.7 nM, Learn More
  24. PF-04418948

    Catalog No. A12894
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    EP2 Receptor antagonist
    PF-04418948 is a potent and selective prostaglandin EP2 receptor antagonist with IC50 of 16 nM. Phase 1. Learn More
  25. KAG-308

    Catalog No. A18389
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    EP4 agonist
    KAG-308, a newly-identified EP4-selective agonist shows efficacy for treating ulcerative colitis and can bring about lower risk of colorectal carcinogenesis by oral administration. Learn More
  26. CP544326 (Taprenepag)

    Catalog No. A15853
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    EP2 Agonist‎
    C-544326 is a potent and selective prostaglandin E2 receptor agonist with EC50 value of 2.8 nM. Learn More
  27. TG6-10-1

    Catalog No. A15968
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    Prostaglandin E2 receptor antagonist
    TG6-10-1 is a potent and selective antagonist for the prostaglandin E2 receptor subtype EP2. Learn More
  28. Laropiprant (MK0524)

    Catalog No. A11483
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    DP1 inhibitor
    Laropiprant is used in combination with niacin to reduce blood cholesterol. Laropiprant acts as a DP1 antagonist, reducing the vasodilation. Learn More

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