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AMPA receptor

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Catalog No. Product Name Application Product Information

CP 465022 hydrochloride

AMPA antagonist
CP 465022 is a selective, non-competitive AMPA antagonist with IC50 of 25 nM in rat cortical neurons that displays potent anticonvulsant activity.


AMPA/kainate receptor antagonist
Talampanel is a non-competitive antagonist of AMPA-receptor.

YM90K hydrochloride

AMPA antagonist
YM90K hydrochloride is a selective AMPA receptor antagonist that delays neuronal death in a global ischemia model and cerebral infarction in a focal ischemia model following postischemic administration.


AMPA antagonist
Tezampanel is an antagonist at the AMPA and kainate families of ionotropic glutamate receptors, with selectivity for the GluR5 subtype of the kainate receptor.
A10078 SALE


AMPA Receptor Inhibitor
Aniracetam is an ampakine and nootropic of the racetam chemical class purported to be considerably more potent than piracetam.


AMPA/kainate antagonist
CNQX is a competitive, non-NMDA glutamate receptor antagonist (IC50s = 0.3 and 1.5 uM for AMPA and kainate receptors, respectively, versus IC50 = 25 uM for NMDA receptors).


AMPA desensitization inhibitor
Cyclothiazide is a benzothiadiazide that acts as a potentiator of AMPA receptors, positively modulating its response to glutamic acid (EC50 = 3.8 M).


AMPA receptor modulator
Farampator has been investigated for its effect on AMPA receptors and researched for potential use in the treatment of schizophrenia and Alzheimer's Disease. It was found to improve short-term memory, but impaired episodic memory.

IEM 1754 Dihydrobromide

AMPA Receptor Blocker
IEM 1754 Dihydrobromide is a voltage-dependent open-channel blocker of AMPA receptors.


NMDA receptor antagonist
DNQX is a non-N-methyl-D-aspartate (non-NMDA) receptor complex antagonist.
A13109 SALE


AMPA Receptor Antagonist
NBQX is a potent, selective and competitive AMPA receptor antagonist.


LY450108 is an alpha-amino-3-hydroxy-5-methyl-4-isoxazole-propionic acid (AMPA) receptor potentiator.


LY404187 is a selective, potent and centrally active positive allosteric modulator of AMPA receptors.

GYKI-52466 dihydrochloride

AMPA and Kainate antagonist
GYKI-52466 dihydrochloride is selective non-competitive AMPA receptor antagonist (IC50 values are 10-20, ~ 450 and >> 50 μM for AMPA- , kainate- and NMDA-induced responses respectively).
A12349 SALE

Ampalex (CX-516)

Ampalex is an ampakine and nootropic that acts as an AMPA receptor positive allosteric modulator

CNQX disodium salt

AMPA/kainate antagonist
CNQX disodium salt, water-soluble form of AMPA/kainate antagonist CNQX (GLXC-11053).

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