Androgen Receptors

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  1. Agonist (1)
  2. Antagonist (7)
  3. Inhibitor (1)
  4. Modulator (3)


14 Item(s)

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Catalog No. Product Name Application Product Information
A10008

(R)-Bicalutamide

Androgen Receptor antagonist
(R)-Bicalutamide is an active competitive non-steroidal androgen receptor antagonist with an IC50 of 0.17 μM for MDA 453 cells.
A10009

17 alpha-propionate

Androgen antagonist
17 alpha-propionate is a new topical and peripherally selective androgen antagonist.
A10076

Andarine (GTX-007)

Androgen Receptor agonist
Andarine (GTX-007) is an investigational selective androgen receptor modulator (SARM).
A12396

AZD3514

AR inhibitor downregulator
AZD-3514 is a potent androgen receptor downregulator with potential anticancer cancer activity.
A10142

Bicalutamide (Casodex)

Androgen Receptor antagonist
Bicalutamide is an oral non-steroidal anti-androgen used in the treatment of prostate cancer and hirsutism.
A12805

BMS564929

Androgen receptor (AR) modulator
BMS-564929 is a novel, highly potent, orally active, nonsteroidal tissue selective androgen receptor (AR) modulator, and this compound has been advanced to clinical trials for the treatment of age-related functional decline.
A13398

Bopindolol malonate

-
A13407

Clenbuterol hydrochloride

-
A15814

EPI-001

Androgen Receptor antagonist
EPI-001 is an antagonist of the androgen receptor (AR) that acts by binding covalently to the N-terminal domain (NTD) of the AR and blocking protein-protein interactions required for transcriptional activity of the AR and its splice variants (IC50 for inhibition of AR NTD transactivation ?? 6 ?M)
A10402

Flutamide

Androgen receptor antagonist
Flutamide is an antiandrogen drug, with its active metablolite binding at androgen receptor with Ki values of 55 nM, and primarily used to treat prostate cancer.
A10562

MDV3100

Androgen receptor antagonist
MDV3100 is androgen-receptor inhibitor. Highly recommended inhibitor in AR research.
A15164

MK-0773

Androgen receptor modulator
MK-0773, one of selective androgen receptor modulators (SARMs), is a 4-aza-steroid that exhibited tissue selectivity in humans (IC50= 6.6 nM).
A15797

ODM-201

Androgen receptor antagonist
ODM-201 is a potent and full antagonists for human AR (hAR) with IC50 values of 26 nM by transactivation assays in AR-HEK293 cells.
A10253

Ostarine (MK-2866, GTx-024)

Androgen Receptor Modulators
Ostarine is an androgen receptor modulator (SARM)

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