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A 438079 hydrochloride
Catalog No. A14983 P2X7 receptor antagonistA 438079 Hcl is a competitive P2X7 receptor antagonist (pIC50 = 6.9 for the inhibition of Ca2+ influx in the human recombinant P2X7 cell line). Learn More -
AF-353
Catalog No. A13131 P2X3/P2X2/3 receptor antagonistAF-353 is a novel, potent and orally bioavailable P2X3/P2X2/3 receptor antagonist, inhibits human and rat P2X3 (pIC50= 8.0). Learn More -
JNJ-54175446
Catalog No. A18675 P2X7 receptor antagonistJNJ-54175446 is a potent and selective brain penetrant P2X7 receptor antagonist, with pIC50s of 8.46 and 8.81 for hP2X7 receptor and rP2X7 receptor, respectively. Learn More -
A 839977
Catalog No. A21178 -
CE-224535
Catalog No. A21183 -
GW791343 trihydrochloride
Catalog No. A21204 P2X7 allosteric modulatorGW791343 3Hcl is a P2X7 allosteric modulator; exhibits species-specific activity and acts as a negative allosteric modulator of human P2X7 (pIC50 = 6.9 - 7.2). Learn More -
Minodronic acid
Catalog No. A21975 purinergic P2X2/3 receptors antagonistMinodronic acid (YM-529) is an antagonist of purinergic P2X2/3 receptors involved in pain. Learn More -
GW791343 HCl
Catalog No. A11107 P2X7 modulatorGW791343 2HCl acts as a negative allosteric modulator of human P2X7 (pIC50 = 6.9 - 7.2) and a positive allosteric modulator of rat P2X7. Learn More -
Ticlopidine HCl
Catalog No. A11690 Ticlopidine is an adenosine diphosphate (ADP) receptor inhibitor. It inhibits platelet aggregation by altering the function of platelet membranes by blocking ADP receptors. This prevents the conformational change of glycoprotein IIb/IIIa which allows platelet binding to fibrinogen. Learn More -
A 740003
Catalog No. A11316 P2X7 receptor antagonistA 740003 is a novel competitive antagonist of P2X7 receptors (IC50 values = 40 nM for human and 18 nM for rat). Learn More -
NF 279
Catalog No. A11972 P2X1 antagonistNF279 is a suramin analog that acts as a highly selective, competitive, and reversible ATP-antagonist of P2X receptor (IC50/KB ~ 1 μM in smooth muscle). Learn More -
A-317491 sodium salt hydrate
Catalog No. A12412 P2X3 and P2X2/3 receptor antagonistA-317491 sodium salt hydrate is a non-nucleotide P2X3 and P2X2/3 receptor antagonist, which inhibits calcium flux mediated by the receptors. Learn More -
A-804598
Catalog No. A16066 P2X7 receptor antagonistA-804598 is a P2X7 selective, competitive antagonist with the IC50s value for human, rat and mouse channels of 11, 10 and 9 nM, respectively. Learn More -
A-438079 HCl
Catalog No. A12597 P2X7 receptor antagonistA-438079 HCl is a competitive P2X7 receptor antagonist (pIC50 = 6.9 for the inhibition of Ca2+ influx in the human recombinant P2X7 cell line). Devoid of activity at other P2 receptors (IC50 >> 10 uM). Learn More
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