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$0.00 Kinesin
| Catalog No. | Inhibitor Name | Kinesin |
|---|---|---|
| A10486 | Ispinesib | *** |
| A10828 | SB743921 | **** |
| A11170 | AZ 3146 | * |
| A11435 | GSK923295 | ** |
| A14290 | MPI-0479605 | *** |
| A14234 | ARQ 621 |
Notes:
1.Hover mouse over "" to view the IC50 value.(A few compounds have proven potency but without published IC50 data.)
2.For more details about the compound, click on the product name of your interest.
3.The higher the number of "" is, the more potent the inhibitor or activator is.
4."" refers to compounds which do inhibitory effects on the related isoform, but without specific value.
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Litronesib Racemate
Catalog No. A21498 kinesin Eg5 inhibitorLitronesib (Racemate) is the racemate of litronesib. Litronesib is a selective, allosteric inhibitor of kinesin Eg5. Learn More -
Arry-520 (Filanesib)
Catalog No. A11050 KSP inhibitorKSP inhibitor ARRY-520 specifically inhibits KSP (kinesin-5 or Eg5) with potential antineoplastic activity. Learn More -
Ispinesib (SB-715992)
Catalog No. A10486 KSP InhibitorIspinesib (SB-715992) is a potent inhibitor of kinesin spindle protein, a kinesin motor protein essential for the formation of a bipolar mitotic spindle and cell cycle progression through mitosis. Learn More -
AZ 3146
Catalog No. A11170 Mps1 inhibitorAZ 3146 is a potent and selective monopolar spindle 1 (Mps1) kinase inhibitor (IC50 = 35 nM). It interferes with chromosome alignment and overrides spindle assembly checkpoint and also Inhibits the recruitment of Mad1, Mad2 and centromere protein E (CENP-E) to kinetochores.
Learn More -
SB 743921
Catalog No. A10828 KSP InhibitorSB 743921, a second generation KSP inhibitor, is a highly potent and active therapeutic in preclinical models of cancer. Learn More -
Monastrol
Catalog No. A11976 Kinesin-5(KIF11) inhibitorMonastrol is a potent, cell permeable non-tubulin-interacting mitosis inhibitor. Monastrol blocks mitosis (IC5N/A = 14 μM) by binding to the mitotic kinesin Eg5, a motor protein required for spindle bipolarity. Learn More -
GSK-923295
Catalog No. A11435 CENP-E inhibitorGSK-923295, is a small-molecule inhibitor of the mitotic kinesin centromere-associated protein E, (CENP-E). Learn More -
CW069
Catalog No. A13735 Microtubule Associated inhibitorCW069 is an allosteric, and selective inhibitor of microtubule motor protein HSET with IC50 of 75 uM, significant selectivity over KSP. Learn More -
ARQ 621
Catalog No. A14234 Eg5 mitotic motor protein inhibitorARQ 621 is an allosteric, and selective Eg5 mitotic motor protein inhibitor. Learn More -
MPI-0479605
Catalog No. A14290 Mps1 inhibitorMPI-0479605 is an ATP competitive and selective inhibitor of mitotic kinase Mps1 Learn More -
ARRY-520 R enantiomer
Catalog No. A15001 KSP inhibitorARRY-520 R enantiomer is the R form of ARRY-520, which is a synthetic, small molecule kinesin spindle protein (KSP) inhibitor with IC50 of 6 nM. Learn More -
Dimethylenastron
Catalog No. A15841 Kinesin Eg5 inhibitorDimethylenastron is an inhibitor of mitotic motor kinesin Eg5 with IC50 value of 200 nM. Learn More -
K 858
Catalog No. A15844 Kinesin Eg5 inhibitorK 858 is a selective ATP-uncompetitive mitotic kinesin Eg5 inhibitor with IC50 value of 1.3 uM. Learn More -
EMD534085
Catalog No. A15956 Kinesin inhibitorEMD534085 is a kinesin inhibitor currently in clinical development. Learn More
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