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$0.00 Adenosine Receptors
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Reversine
Catalog No. A13250 human A3 adenosine receptor antagonist /Aurora inhibitorReversine is a potent human A3 adenosine receptor antagonist with Ki of 0.66 μM, and a pan-aurora A/B/C kinase inhibitor with IC50 of 12 nM/13 nM/20 nM, respectively. Also used for stem cell dedifferentiation. Learn More -
Pentostatin
Catalog No. A11534 Adenosine deaminase inhibitorPentostatin is an irreversible inhibitor of adenosine deaminase (Ki = 2.5 pM). Learn More -
MT-DADMe-ImmA
Catalog No. A13651 human 5'-methylthioadenosine phosphorylase inhibitorMT-DADMe-ImmA is an inhibitor of human 5'-methylthioadenosine phosphorylase (MTAP) with a Ki of 90 pM. Learn More -
A2A receptor antagonist 1
Catalog No. A12567 adenosine A2A/A1 receptor antagonistA2A receptor antagonist 1 (CPI-444 analog) is an antagonist of both adenosine A2A receptor and A1 receptor with Kis of 4 and 264 nM, respectively. Learn More -
AB-MECA
Catalog No. A12189 A3 adenosine receptor agonistAB-MECA is a high affinity A3 adenosine receptor agonist, has high affinity for recombinant A1 and A3 receptors. Learn More -
CGS 21680
Catalog No. A11354 adenosine A2A receptor agonistCGS 21680 is a selective adenosine A2A receptor agonist, with a Ki of 27 nM. Learn More -
APNEA
Catalog No. A20845 A3 adenosine receptor agonistAPNEA (N6-[2-(4-Aminophenyl)ethyl]adenosine) is a potent, non-selective A3 adenosine receptor agonist. Learn More -
LAS101057
Catalog No. A21203 A2B receptor antagonistLAS101057 is a potent, selective, and orally efficacious A2B receptor antagonist. Learn More -
Tonapofylline
Catalog No. A21328 adenosine A1 receptor antagonistTonapofylline (BG 9928) is an orally active and selective adenosine A1 receptor antagonist with a Ki of 7.4 nM for human adenosine A1 receptor (hA1), which displays 915-fold selectivity versus human adenosine A2A receptor and 12-fold selectivity versus human adenosine A2B receptor and is used in development for the treatment of heart failure. Learn More -
LUF6000
Catalog No. A21532 A3 adenosine receptor allosteric modulatorLUF6000 is an allosteric modulator of the human A3 adenosine receptor (AR). Learn More -
EHNA hydrochloride
Catalog No. A21585 Adenosine deaminase inhibitorEHNA hydrochloride is a specific inhibitor of adenosine deaminase, prevents dAdo degradation and increases mitochondrial dATP levels in fibroblasts. Learn More -
Rolofylline
Catalog No. A21649 adenosine A1 receptor antagonistRolofylline (KW-3902) is a potent, selective adenosine A1 receptor antagonist that is under development for the treatment of patients with acute congestive heart failure and renal impairment. Learn More -
Derenofylline
Catalog No. A21990 adenosine A1 receptor antagonistDerenofylline (SLV 320) is a potent, selective and orally active adenosine A1 receptor antagonist, with Ki values of 1 nM, 200 nM and 398 nM for human A1, A3 and A2A receptors respectively. Learn More -
MRS 1754
Catalog No. A21998 A2B adenosine receptor antagonistMRS 1754 is a selective antagonist radioligand for A2B adenosine receptor with very low affinity for A1 and A3 receptors of both humans and rats. Learn More -
N6-Cyclohexyladenosine
Catalog No. A21008 A1 receptor agonistN6-Cyclohexyladenosine is a selective A1 receptor agonist (EC50 = 8.2 nM). Learn More -
MRS1177
Catalog No. A16871 Adenosine A3 receptor antagonistMRS1177 is a potent and selective human Adenosine A3 receptor (hA3AR) antagonist, with a Ki of 0.3 nM. Learn More -
MRS1186
Catalog No. A16870 Adenosine A3 receptor antagonistMRS1186 is a potent and selective human Adenosine A3 receptor (hA3AR) antagonist, with a Ki of 7.66 nM. Learn More -
AZD-4635 (HTL1071)
Catalog No. A16820 A2AR antagonistAZD-4635 (HTL1071) is an oral A2AR antagonist that binds to human A2AR with a Ki of 1.7 nM and with > 30-fold selectivity over other adenosine receptors. Learn More -
NECA
Catalog No. A16962 Adenosine receptor agonistNECA is a high-affinity adenosine receptor agonist (Ki values are 6.2, 14, and 20 nM for human A3, A1 and A2A receptors respectively; EC50 = 2.4 μM for human A2B). Learn More -
Theophylline-7-acetic acid
Catalog No. A16822 Adenosine receptor antagonistTheophylline-7-acetic acid (Acefylline), acting as an adenosine receptor antagonist, is a stimulant drug of the xanthine chemical class. Learn More -
MRS1706
Catalog No. A16868 adenosine A2B receptor agonistMRS1706 is a selective adenosine A2B receptor inverse agonist with Ki values of 1.39, 157, 112, and 230 nM for human A2B, A1, A2A, and A3 receptors, respectively. Learn More -
BAY-545
Catalog No. A20116 A2B adenosine receptor antagonistBAY-545 is a potent and selective A2B adenosine receptor antagonist, with an IC50 of 59 nM. Learn More -
ST3932
Catalog No. A12880 Adenosine A2A receptor antagonistST3932 is a metabolite of ST1535, acts as an antagonist of adenosine A2A receptor, with Kis of 8 nM and 33 nM for A2A and A1 receptors, respectively. Learn More -
Tecadenoson
Catalog No. A13302 A1 adenosine receptor agonistTecadenoson (CVT-510) is a selective A1 adenosine receptor agonist. Learn More -
CPI-444
Catalog No. A19242 A2AR antagonistCPI-444 is a potent, oral and selective A2A receptor (A2AR) antagonist, which induces antitumor responses. Learn More -
CGS-15943
Catalog No. A14327 Adenosine A Receptor antagonistCGS 15943 is a potent, non-selective Adenosine A Receptor antagonist. It is orally active in vivo. Learn More -
SYN-115 (Tozadenant)
Catalog No. A11560 A2a receptor antagonistSYN115 is an orally administered, potent and selective inhibitor of the adenosine 2a (A2a) receptor that is being developed initially for the treatment of Parkinson’s disease, but may also have utility in other CNS disorders. Learn More -
CGS 21680 HCl Hydrate
Catalog No. A11619 Adenosine A2A Receptor AgonistCGS 21680 is a specific adenosine A2A subtype receptor agonist. Learn More -
Adenosine
Catalog No. A10040 Adenosine plays an important role in biochemical processes, such as energy transfer-as adenosine triphosphate (ATP) and adenosine diphosphate (ADP)-as well as in signal transduction as cyclic adenosine monophosphate, cAMP. It is also an inhibitory neurotransmitter. Learn More -
Aminophylline
Catalog No. A10066 Adenosine receptor antagonistAminophylline is a nonselective adenosine receptor antagonist and phosphodiesterase inhibitor capable of reversing ischemia-induced bradyasystole. Learn More -
Dyphylline
Catalog No. A10339 Adenosine receptor antagonistDyphylline is a xanthine derivative with bronchodilator and vasodilator effects. It acts as an adenosine receptor antagonist and phosphodiesterase inhibitor. Learn More -
SCH 442416
Catalog No. A12695 A2A Receptor AntagonistSCH 442416 is a selective adenosine A2A receptor antagonist; binds to human and rat A2A receptors with high affinity (Ki values are 0.048 and 0.5 nM respectively). Displays > 23000-fold selectivity for hA2A over hA1 in vitro with minimal affinity for hA2B and hA3 receptors (IC50 > 10 μM). Learn More -
Tamsulosin hydrochloride
Catalog No. A12846 Tamsulosin hydrochloride is an antagonist of alpha1A adrenoceptors in the prostate. Learn More -
CVT 6883
Catalog No. A13745 adenosine A2B receptors antagonistCVT-6883, a selective A2B adenosine antagonist, represents a novel potential approach to treating cardiopulmonary diseases. Learn More -
Capadenoson
Catalog No. A14159 Adenosine Receptor agonistCapadenoson is a selective agonist of adenosine-A1 receptor. Learn More -
5-Iodotubercidin
Catalog No. A13948 Adenosine kinase inhibitor5-Iodotubercidin is a potent adenosine kinase inhibitor with IC50 of 26 nM. Learn More -
CF-102
Catalog No. A14402 Adenosine A3 receptor agonistCF-102 is an orally bioavailable, synthetic, highly selective adenosine A3 receptor (A3AR) agonist with potential antineoplastic activity. Learn More -
Proxyphylline
Catalog No. A16821 A1 adenosine receptors antagonistProxyphylline is a derivative of theophylline which is used as a bronchodilator and for its cardiovascular properties. It selectively antagonizes A1 adenosine receptors (Ki = 82 nM for bovine brain) versus A2 adenosine receptors (Ki = 850 μM for platelets). Learn More -
IB-MECA
Catalog No. A14345 Adenosine A3-R agonistIB-MECA has been shown to act as a potent and selective Adenosine A3-R agonist with Ki values of 1.1, 54 and 56 nM for Adenosine A3-R, Adenosine A1-R and Adenosine A2A-R, respectively. Learn More -
ZM-241385
Catalog No. A13517 Adenosine A2A antagonistZM-241385 is a potent and highly selective Adenosine A2A-R antagonist, with a pA2 of 9.02 for Adenosine A2A-R in cardiac vasculature and selectivities of 1000, 91 and 500,000 over Adenosine A1-R, Adenosine A2B-R and Adenosine A3-R sites, respectively. Learn More -
Preladenant
Catalog No. A13504 Adenosine A2A receptor antagonistPreladenant is a potent and selective antagonist at the adenosine A2A receptor. Learn More -
SCH58261
Catalog No. A15886 A2A adenosine receptor antagonistSCH58261 is a potent and selective A2a adenosine receptor antagonist with Ki of 2.3 nM and 2 nM for rat A2a and bovine A2a, respectively. Learn More -
DPCPX
Catalog No. A16104 Adenosine A1-R antagonistDPCPX, a xanthine derivative, is a very potent and selective Adenosine A1-R antagonist. It displays very modest efficacy against Adenosine A2A-R, Adenosine A2B-R and Adenosine A3-R. Learn More -
2-Chloroadenosine (CADO)
Catalog No. A16105 Adenosine A Receptor agonist2-Chloroadenosine is a metabolically stable analog of adenosine that behaves as an Adenosine A Receptor agonist (Ki values are 300, 80 and 1900 nM for Adenosine A1-R, Adenosine A2A-R and Adenosine A3-R, respectively). Learn More -
CGS 21680 HCl
Catalog No. A16441 Adenosine A2 receptor agonistCGS 21680 HCl is an adenosine A2 receptor agonist with IC50 of 22 nM, exhibits 140-fold over A1 receptor. Learn More -
Regadenoson
Catalog No. A12541 A2A adenosine agonistRegadenoson was selective agonist for the A2A adenosine receptor versus the A1, A2B, and A3 receptors in binding and functional studies. Regadenoson was also found to be a full and potent agonist to cause coronary vasodilation, a response that has a very large A2A receptor reserve? Learn More -
Vipadenant (BIIB-014)
Catalog No. A13963 A2A receptor antagonistVipadenant, also known as BIIB014, CEB-4520, is a potent, selective and orally available adenosine A2A receptor antagonist under development for Parkinson's disease. Vipadenant demonstrates strong oral activity in commonly used models of Parkinson's disease. Learn More -
Istradefylline (KW-6002)
Catalog No. A11451 A2A antagonistIstradefylline (KW-6002) is a selective antagonist at the A2A receptor. It has been found to be useful in the treatment of Parkinson's disease. Learn More
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