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$0.00 Androgen Receptors
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Flutamide
Catalog No. A10402 Androgen receptor antagonistFlutamide is an antiandrogen drug, with its active metablolite binding at androgen receptor with Ki values of 55 nM, and primarily used to treat prostate cancer. Learn More -
EPI-001
Catalog No. A15814 Androgen Receptor antagonistEPI-001 is an antagonist of the androgen receptor (AR) that acts by binding covalently to the N-terminal domain (NTD) of the AR and blocking protein-protein interactions required for transcriptional activity of the AR and its splice variants (IC50 for inhibition of AR NTD transactivation ?? 6 μM) Learn More -
ODM-201
Catalog No. A15797 Androgen receptor antagonistODM-201 is a potent and full antagonists for human AR (hAR) with IC50 values of 26 nM by transactivation assays in AR-HEK293 cells. Learn More -
MK-0773
Catalog No. A15164 Androgen receptor modulatorMK-0773, one of selective androgen receptor modulators (SARMs), is a 4-aza-steroid that exhibited tissue selectivity in humans (IC50= 6.6 nM). Learn More -
AZD3514
Catalog No. A12396 AR inhibitor downregulatorAZD-3514 is a potent androgen receptor downregulator with potential anticancer cancer activity. Learn More -
GSK-2881078
Catalog No. A12645 androgen receptor modulatorGSK-2881078 is a selective androgen receptor modulator (SARM) that is being evaluated for effects on muscle growth and strength in subjects with muscle wasting to improve their physical function. Learn More -
N-desMethyl EnzalutaMide
Catalog No. A13964 androgen-receptor (AR) antagonistN-desMethyl EnzalutaMide is used in the treatment of disorders involving androgen, estrogen and progesterone receptors. Learn More -
RU 58841
Catalog No. A11541 AR antagonistRU58841, also known as PSK-3841 or HMR-3841, is a non-steroidal anti-androgen. Learn More -
Bopindolol malonate
Catalog No. A13398 Bopindolol malonate is a non-selective, potent, long-acting beta adrenoceptor antagonist. It demonstrates inhibition of H2O2-induced lipid peroxdiation. Learn More -
Megestrol Acetate
Catalog No. A10563 Megestrol Acetate is a progesterone derivative with antineoplastic properties Learn More -
Ostarine (MK-2866, GTx-024)
Catalog No. A10253 Androgen Receptor ModulatorsOstarine is an androgen receptor modulator (SARM) Learn More -
BMS564929
Catalog No. A12805 Androgen receptor (AR) modulatorBMS-564929 is a novel, highly potent, orally active, nonsteroidal tissue selective androgen receptor (AR) modulator, and this compound has been advanced to clinical trials for the treatment of age-related functional decline. Learn More -
17 alpha-propionate
Catalog No. A10009 Androgen antagonist17 alpha-propionate is a new topical and peripherally selective androgen antagonist. Learn More -
ASC-J9
Catalog No. A11300 ASC-J9 suppresses castration-resistant prostate cancer growth through degradation of full-length and splice variant androgen receptors. Learn More -
Cyproterone acetate
Catalog No. A11409 Androgen Receptor antagonistCyproterone acetate is a synthetic derivative of 17-hydroxyprogesterone, and acts as an androgen receptor antagonist as well as a weak progesterone receptor agonist with weak progestational and glucocorticoid activity. Learn More -
TOK-001 (Galeterone)
Catalog No. A11138 CYP17 inhibitorTOK-001 (Galeterone) is both an androgen receptor antagonist and CYP17A1 inhibitor. Learn More -
Andarine (GTX-007)
Catalog No. A10076 Androgen Receptor agonistAndarine (GTX-007) is an investigational selective androgen receptor modulator (SARM). Learn More -
Bicalutamide (Casodex)
Catalog No. A10142 Androgen Receptor antagonistBicalutamide is an oral non-steroidal anti-androgen used in the treatment of prostate cancer and hirsutism. Learn More -
(R)-Bicalutamide
Catalog No. A10008 Androgen Receptor antagonist(R)-Bicalutamide is an active competitive non-steroidal androgen receptor antagonist with an IC50 of 0.17 μM for MDA 453 cells. Learn More -
MDV3100
Catalog No. A10562 Androgen receptor antagonistMDV3100 is androgen-receptor inhibitor. Highly recommended inhibitor in AR research. Learn More
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