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Androgen Receptors

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Catalog No. Product Name Application Product Information
A10402 SALE


Androgen receptor antagonist
Flutamide is an antiandrogen drug, with its active metablolite binding at androgen receptor with Ki values of 55 nM, and primarily used to treat prostate cancer.


Androgen Receptor antagonist
EPI-001 is an antagonist of the androgen receptor (AR) that acts by binding covalently to the N-terminal domain (NTD) of the AR and blocking protein-protein interactions required for transcriptional activity of the AR and its splice variants (IC50 for inhibition of AR NTD transactivation ?? 6 ?M)
A15797 SALE


Androgen receptor antagonist
ODM-201 is a potent and full antagonists for human AR (hAR) with IC50 values of 26 nM by transactivation assays in AR-HEK293 cells.


Androgen receptor modulator
MK-0773, one of selective androgen receptor modulators (SARMs), is a 4-aza-steroid that exhibited tissue selectivity in humans (IC50= 6.6 nM).

Clenbuterol hydrochloride

A11541 SALE

RU 58841

AR antagonist

N-desMethyl EnzalutaMide

androgen-receptor (AR) antagonist
N-desMethyl EnzalutaMide is used in the treatment of disorders involving androgen, estrogen and progesterone receptors.
A14346 SALE


androgen receptor modulator
LGD-4033 is an investigational selective androgen receptor modulator for treatment of conditions such as muscle wasting and osteoporosis, currently under development by Ligand Pharmaceuticals.

Boldenone Undecylenate

Boldenone undecylenate is a synthetic steroid which has a similar effect as the natural steroid testosterone, it is frequently used in veterinary medicine, though it is also used in humans.
A12645 SALE


androgen receptor modulator
GSK-2881078 is a selective androgen receptor modulator (SARM) that is being evaluated for effects on muscle growth and strength in subjects with muscle wasting to improve their physical function.

Bopindolol malonate

A10563 SALE

Megestrol Acetate

Megestrol Acetate is a progesterone derivative with antineoplastic properties
A12396 SALE


AR inhibitor downregulator
AZD-3514 is a potent androgen receptor downregulator with potential anticancer cancer activity.
A10562 SALE


Androgen receptor antagonist
MDV3100 is androgen-receptor inhibitor. Highly recommended inhibitor in AR research.


Androgen Receptor antagonist
(R)-Bicalutamide is an active competitive non-steroidal androgen receptor antagonist with an IC50 of 0.17 μM for MDA 453 cells.
A10142 SALE

Bicalutamide (Casodex)

Androgen Receptor antagonist
Bicalutamide is an oral non-steroidal anti-androgen used in the treatment of prostate cancer and hirsutism.
A10076 SALE

Andarine (GTX-007)

Androgen Receptor agonist
Andarine (GTX-007) is an investigational selective androgen receptor modulator (SARM).
A11138 SALE

TOK-001 (Galeterone)

CYP17 inhibitor
TOK-001 (Galeterone) is both an androgen receptor antagonist and CYP17A1 inhibitor.
A11409 SALE

Cyproterone acetate

Androgen Receptor antagonist
Cyproterone acetate is a synthetic derivative of 17-hydroxyprogesterone, and acts as an androgen receptor antagonist as well as a weak progesterone receptor agonist with weak progestational and glucocorticoid activity.
A11300 SALE


ASC-J9 suppresses castration-resistant prostate cancer growth through degradation of full-length and splice variant androgen receptors.
A10009 SALE

17 alpha-propionate

Androgen antagonist
17 alpha-propionate is a new topical and peripherally selective androgen antagonist.


Androgen receptor (AR) modulator
BMS-564929 is a novel, highly potent, orally active, nonsteroidal tissue selective androgen receptor (AR) modulator, and this compound has been advanced to clinical trials for the treatment of age-related functional decline.
A10253 SALE

Ostarine (MK-2866, GTx-024)

Androgen Receptor Modulators
Ostarine is an androgen receptor modulator (SARM)

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