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$0.00 Calcium Channels
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GV-58
Catalog No. A21966 N- and P/Q-type Ca2+ channels agonistGV-58 is a potent, selective N- and P/Q-type Ca2+ channels agonist with EC50 of 7.21/8.81 uM for N-type/P-Q-type Ca2+ channel; 20-fold less potent CDK inhibitor activity. Learn More -
JTV-519 free base
Catalog No. A21846 Ca2+-dependent blockerTV-519 free base (K201 free base) is a Ca2+-dependent blocker of sarcoplasmic reticulum Ca2+-stimulated ATPase (SERCA) and a partial agonist of ryanodine receptors in striated muscle. Antiarrhythmic and cardioprotective properties. Learn More -
TTA-Q6(isomer)
Catalog No. A21724 T-type Ca2+ channel antagonistTTA-Q6(isomer) is an isomer of TTA-Q6. TTA-Q6 is a selective T-type Ca2+ channel antagonist. Learn More -
TTA-Q6
Catalog No. A21360 T-type Ca2+ channel antagonistTTA-Q6 is a selective T-type Ca2+ channel antagonist, used in the neurological disease. Learn More -
(S)-(-)-Bay-K-8644
Catalog No. A21164 L-type Ca2+ channel agonist(S)-(-)-Bay-K-8644 is an agonist of L-type Ca2+ channel. (S)-(-)-Bay-K-8644 activates Ba2+ currents (IBa) (EC50=32 nM). Learn More -
ABT-639 hydrochloride
Catalog No. A12571 T-type Ca2+ channel blockerABT-639 hydrochloride is a novel, peripherally acting, selective T-type Ca2+ channel blocker. Learn More -
Caldaret
Catalog No. A13148 intracellular Ca2+ handling modulatorCaldaret is an intracellular Ca2+ handling modulator that acts through reverse mode Na+/Ca2+ exchanger inhibition. Learn More -
Aranidipine
Catalog No. A18291 Calcium channel antagonistAranidipine (MPC1304) is a Ca2+ channel antagonist with potent and long-lasting antihypertensive effects. Learn More -
(S)-Amlodipine
Catalog No. A14935 Calcium channel blocker(S)-Amlodipine is a (S)-Enantiomer of Amlodipine and a dihydropyridine calcium channel blocker with activity resides mainly in the (-)-isomer. Learn More -
NNC 55-0396
Catalog No. A15188 Calcium channel blockerNNC 55-0396, Mibefradil derivative, is a highly selective T-type calcium channel blocker; displays IC50 values of 6.8 and > 100 μM for inhibition of Cav3.1 T-type channels and HVA currents respectively in INS-1 cells. Learn More -
NP118809
Catalog No. A15192 N-type calcium channel blockerNP118809 is a potent N-type calcium channel blockers(IC50= 0.11 uM) ; good selectivity over L-type calcium channels. Learn More -
NS6180
Catalog No. A12405 K(Ca) 3.1 channel blockerNS6180 is a novel potent and selective KCa3.1 channel inhibitor(IC50= 9 nM) prevents T-cell activation and inflammation. Learn More -
Bay K 8644
Catalog No. A15875 Calcium Channel ActivatorBay K 8644 is a potent, selective activator of L-type Ca2+ channel with IC50 of 17.3 nM. Learn More -
Mibefradil dihydrochloride
Catalog No. A12482 Calcium channel blockerMibefradil 2Hcl is calcium channel blocker with moderate selectivity for T-type Ca2+ channels displaying IC50 values of 2.7 uM and 18.6 uM for T-type and L-type channels respectively. Learn More -
Dantrolene sodium Hemiheptahydrate
Catalog No. A16146 Dantrolene sodium Hemiheptahydrate is a skeletal muscle relaxant that acts by interfering with excitation-contraction coupling in the muscle fiber. Learn More -
YM-58483
Catalog No. A16346 CRAC channel inhibitorYM-58483 is the first selective and potent inhibitor of CRAC channels and subsequent Ca2+ signals. Learn More -
Cinepazide maleate
Catalog No. A16454 Cinepazide maleate is a maleate salt form of cinepazide which is a vasodilator. Learn More -
Cinnarizine
Catalog No. A16455 calcium channel blockerCinnarizine is a medication derivative of piperazine, and characterized as an antihistamine and a calcium channel blocker. Learn More -
Berbamine
Catalog No. A14794 -
ABT-639
Catalog No. A12330 T-type Ca2+ channel blockerABT-639 is a novel, peripherally acting, selective T-type Ca2+ channel blocker. Learn More -
Ca2+ channel agonist 1
Catalog No. A12186 Ca2+ channel agonist/CDK2 inhibitorCa2+ channel agonist 1 is an agonist of N-type Ca2+ channel and an inhibitor of Cdk2, with EC50s of 14.23 μM and 3.34 μM, respectively, and is used as a potential treatment for motor nerve terminal dysfunction. Learn More -
Barnidipine
Catalog No. A21940 L-type calcium antagonistBarnidipine (Mepirodipine) is an L-type calcium antagonist (CaA) with high affinity for [3H] initrendipine binding sites (Ki=0.21 nmol/l), has selective action against CaA receptors. Learn More -
Dantrolene sodium
Catalog No. A17644 Calcium channel proteins inhibitorDantrolene sodium is a inhibitor of calcium channel proteins, inhibiting the release of Ca2+ from the sarcoplasm. Dantrolene sodium is a skeletal muscle relaxant which acts by blocking muscle contraction beyond the neuromuscular junction. Learn More -
Clevidipine
Catalog No. A11746 Calcium channel blockerClevidipine is a dihydropyridine calcium channel blocker indicated for the reduction of blood pressure when oral therapy is not feasible or not desirable. Learn More -
Astragaloside A
Catalog No. A11405 Ca2+ signaling modulatorAstragaloside A is a novel regulator of HIF-1α and angiogenesis through the PI3K/Akt pathway in HUVECs that are exposed to hypoxia. Learn More -
CK-1827452 (Omecamtiv mecarbil)
Catalog No. A11206 Myosin activatorCK-1827452 is a selective cardiac specific myosin activator. Learn More -
Manidipine 2HCl
Catalog No. A10554 Manidipine 2HCl is a HCl salt form of Manidipine which is a calcium channel blocker for Ca2+ current with IC50 of 2.6 nM. Learn More -
Amlodipine
Catalog No. A10068 L-type calcium channel blockerAmlodipin is L-type calcium channel blocker that displays antihypertensive properties. It inhibits Ca2+-induced contractions in depolarized rat aorta (IC50 = 1.9 nM) and displays vasoprotective effects in cardiovascular disease. Learn More -
Amlodipine besylate (Norvasc)
Catalog No. A10069 L-type calcium channel blockerAmlodipine-besylate is L-type calcium channel blocker that displays antihypertensive properties. It inhibits Ca2+-induced contractions in depolarized rat aorta (IC50 = 1.9 nM) and displays vasoprotective effects in cardiovascular disease. Learn More -
Cilnidipine
Catalog No. A10215 Calcium channel blockerCilnidipine is a dual blocker of L-type voltage-gated calcium channels in vascular smooth muscle and N-type calcium channels in sympathetic nerve terminals that supply. Learn More -
Isradipine
Catalog No. A10487 calcium channel blockerIsradipine is a calcium channel blocker of the dihydropyridine class. Learn More -
Azelnidipine
Catalog No. A11219 calcium channel blockerAzelnidipine is a calcium blocker that attenuates liver fibrosis and may increase antioxidant defence. that attenuates liver fibrosis and may increase antioxidant defence. Learn More -
Benidipine hydrochloride
Catalog No. A11730 Benidipine hydrochloride is a long-acting T-type calcium channel blocker, on blood pressure and renal function in hypertensive patients with diabetes mellitus. Learn More -
Nilvadipine (ARC029)
Catalog No. A11731 calcium channel blockerNilvadipine is a calcium channel blocker (CCB) used for the treatment of hypertension and chronic major cerebral artery occlusion Learn More -
Tetrandrine (Fanchinine)
Catalog No. A10921 Calcium Channel inhibitorTetrandrine is a calcium channel blocker. It inhibits the degranulation of mast cells.Tetrandrine has anti-inflammatory and anti-fibrogenic actions, which make tetrandrine and related compounds potentially useful in the treatment of lung silicosis, liver cirrhosis, and rheumatoid arthritis. Learn More -
Diethylstilbestrol
Catalog No. A10309 Diethylstilbestrol is a synthetic nonsteroidal estrogen that was first synthesized in 1938. It is also classified as an endocrine disruptor. Learn More -
Diltiazem HCl
Catalog No. A10311 Diltiazem is a nondihydropyridine (non-DHP) member of the class of drugs known as calcium channel blockers, used in the treatment of hypertension, angina pectoris, and some types of arrhythmia. Learn More -
Manidipine (Manyper)
Catalog No. A10553 Manidipine is a dihydropyridine compound and calcium channel protein inhibitor and antagonist. Learn More -
Pinaverium Bromide
Catalog No. A12684 Pinaverium Bromide is a spasmolytic agent with low incidence of anticholinergic effects. Pinaverium Bromide is also an antispasmodic. Learn More -
Nifedipine
Catalog No. A10643 L-type calcium channel blocker.Nifedipine is a L-type calcium channel blocker. Learn More -
Nimodipine
Catalog No. A10645 Calcium Channel inhibitorNimodipine is a L-type Ca2+ channel blocker. Learn More -
BAPTA tetrapotassium
Catalog No. A13989 Selective calcium chelatorBAPTA tetrapotassium is a selective calcium chelator with greater affinity for Ca2+ than Mg2+. Learn More -
BAPTA/AM
Catalog No. A14023 Selective calcium chelatorBAPTA/AM, an intracellular calcium chelator, induces delayed necrosis by lipoxygenase-mediated free radicals in mouse cortical cultures. Learn More -
Dantrolene
Catalog No. A13928 Ca2+ release inhibitorDantrolene sodium is a muscle relaxant that acts by abolishing excitation-contraction coupling in muscle cells, probably by action on the ryanodine receptor. Learn More -
Atagabalin
Catalog No. A13402 Atagabalin is related to gabapentin, which similarly binds to the α2δ calcium channels (1 and 2). Learn More
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