Calcium Channels

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  1. Tetrandrine (Fanchinine)

    Catalog No. A10921
    Calcium Channel inhibitor
    Tetrandrine is a calcium channel blocker. It inhibits the degranulation of mast cells.Tetrandrine has anti-inflammatory and anti-fibrogenic actions, which make tetrandrine and related compounds potentially useful in the treatment of lung silicosis, liver cirrhosis, and rheumatoid arthritis. Learn More
  2. BAPTA tetrapotassium

    Catalog No. A13989
    Selective calcium chelator
    BAPTA tetrapotassium is a selective calcium chelator with greater affinity for Ca2+ than Mg2+. Learn More
  3. BAPTA/AM

    Catalog No. A14023
    Selective calcium chelator
    BAPTA/AM, an intracellular calcium chelator, induces delayed necrosis by lipoxygenase-mediated free radicals in mouse cortical cultures. Learn More
  4. Dantrolene

    Catalog No. A13928
    Ca2+ release inhibitor
    Dantrolene sodium is a muscle relaxant that acts by abolishing excitation-contraction coupling in muscle cells, probably by action on the ryanodine receptor. Learn More
  5. Atagabalin

    Catalog No. A13402
    Atagabalin is related to gabapentin, which similarly binds to the α2δ calcium channels (1 and 2). Learn More
  6. Berbamine

    Catalog No. A14794
    Calcium channel blocker
    Berbamine is a calcium channel blocker. Learn More
  7. (S)-Amlodipine

    Catalog No. A14935
    Calcium channel blocker
    (S)-Amlodipine is a (S)-Enantiomer of Amlodipine and a dihydropyridine calcium channel blocker with activity resides mainly in the (-)-isomer. Learn More
  8. NNC 55-0396

    Catalog No. A15188
    Calcium channel blocker
    NNC 55-0396, Mibefradil derivative, is a highly selective T-type calcium channel blocker; displays IC50 values of 6.8 and > 100 μM for inhibition of Cav3.1 T-type channels and HVA currents respectively in INS-1 cells. Learn More
  9. NP118809

    Catalog No. A15192
    N-type calcium channel blocker
    NP118809 is a potent N-type calcium channel blockers(IC50= 0.11 uM) ; good selectivity over L-type calcium channels. Learn More
  10. NS6180

    Catalog No. A12405
    K(Ca) 3.1 channel blocker
    NS6180 is a novel potent and selective KCa3.1 channel inhibitor(IC50= 9 nM) prevents T-cell activation and inflammation. Learn More
  11. Bay K 8644

    Catalog No. A15875
    Calcium Channel Activator
    Bay K 8644 is a potent, selective activator of L-type Ca2+ channel with IC50 of 17.3 nM. Learn More
  12. Mibefradil dihydrochloride

    Catalog No. A12482
    Calcium channel blocker
    Mibefradil 2Hcl is calcium channel blocker with moderate selectivity for T-type Ca2+ channels displaying IC50 values of 2.7 uM and 18.6 uM for T-type and L-type channels respectively. Learn More
  13. Dantrolene sodium

    Catalog No. A16146
    Dantrolene sodium ia a skeletal muscle relaxant that acts by interfering with excitation-contraction coupling in the muscle fiber. Learn More
  14. YM-58483

    Catalog No. A16346
    CRAC channel inhibitor
    YM-58483 is the first selective and potent inhibitor of CRAC channels and subsequent Ca2+ signals. Learn More
  15. Chlorocresol

    Catalog No. A16444
    Chlorocresol is an activator of ryanodine receptor. Learn More
  16. Cinepazide maleate

    Catalog No. A16454
    Cinepazide maleate is a maleate salt form of cinepazide which is a vasodilator. Learn More
  17. Nimodipine

    Catalog No. A10645
    Calcium Channel inhibitor
    Nimodipine is a L-type Ca2+ channel blocker. Learn More
  18. Nifedipine

    Catalog No. A10643
    L-type calcium channel blocker.
    Nifedipine is a L-type calcium channel blocker. Learn More
  19. Pinaverium Bromide

    Catalog No. A12684
    Pinaverium Bromide is a spasmolytic agent with low incidence of anticholinergic effects. Pinaverium Bromide is also an antispasmodic. Learn More
  20. Astragaloside A

    Catalog No. A11405
    Ca2+ signaling modulator
    Astragaloside A is a novel regulator of HIF-1α and angiogenesis through the PI3K/Akt pathway in HUVECs that are exposed to hypoxia. Learn More
  21. Myosin activator
    CK-1827452 is a selective cardiac specific myosin activator. Learn More
  22. Manidipine 2HCl

    Catalog No. A10554
    Manidipine 2HCl is a HCl salt form of Manidipine which is a calcium channel blocker for Ca2+ current with IC50 of 2.6 nM. Learn More
  23. Amlodipine

    Catalog No. A10068
    L-type calcium channel blocker
    Amlodipin is L-type calcium channel blocker that displays antihypertensive properties. It inhibits Ca2+-induced contractions in depolarized rat aorta (IC50 = 1.9 nM) and displays vasoprotective effects in cardiovascular disease. Learn More
  24. L-type calcium channel blocker
    Amlodipine-besylate is L-type calcium channel blocker that displays antihypertensive properties. It inhibits Ca2+-induced contractions in depolarized rat aorta (IC50 = 1.9 nM) and displays vasoprotective effects in cardiovascular disease. Learn More
  25. Cilnidipine

    Catalog No. A10215
    Calcium channel blocker
    Cilnidipine is a dual blocker of L-type voltage-gated calcium channels in vascular smooth muscle and N-type calcium channels in sympathetic nerve terminals that supply. Learn More
  26. Isradipine

    Catalog No. A10487
    calcium channel blocker
    Isradipine is a calcium channel blocker of the dihydropyridine class. Learn More
  27. Azelnidipine

    Catalog No. A11219
    calcium channel blocker
    Azelnidipine is a calcium blocker that attenuates liver fibrosis and may increase antioxidant defence. that attenuates liver fibrosis and may increase antioxidant defence. Learn More
  28. Lacidipine

    Catalog No. A11729
    Lacidipine is a calcium channel blocker Learn More
  29. Benidipine hydrochloride

    Catalog No. A11730
    Benidipine hydrochloride is a long-acting T-type calcium channel blocker, on blood pressure and renal function in hypertensive patients with diabetes mellitus. Learn More
  30. Nilvadipine (ARC029)

    Catalog No. A11731
    calcium channel blocker
    Nilvadipine is a calcium channel blocker (CCB) used for the treatment of hypertension and chronic major cerebral artery occlusion Learn More
  31. Clevidipine

    Catalog No. A11746
    Calcium channel blocker
    Clevidipine is a dihydropyridine calcium channel blocker indicated for the reduction of blood pressure when oral therapy is not feasible or not desirable. Learn More
  32. Diethylstilbestrol

    Catalog No. A10309
    Diethylstilbestrol is a synthetic nonsteroidal estrogen that was first synthesized in 1938. It is also classified as an endocrine disruptor. Learn More
  33. Diltiazem HCl

    Catalog No. A10311
    Diltiazem is a nondihydropyridine (non-DHP) member of the class of drugs known as calcium channel blockers, used in the treatment of hypertension, angina pectoris, and some types of arrhythmia. Learn More
  34. Manidipine (Manyper)

    Catalog No. A10553
    Manidipine is a dihydropyridine compound and calcium channel protein inhibitor and antagonist. Learn More
  35. Cinnarizine

    Catalog No. A16455
    calcium channel blocker
    Cinnarizine is a medication derivative of piperazine, and characterized as an antihistamine and a calcium channel blocker. Learn More

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