Sodium Channels

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Catalog No. Product Name Application Product Information
A11234 SALE

A 803467

Sodium channel Blocker
A 803467 is a selective blocker of NaV1.8 channels (IC50 values are 8, 2450, 6740, 7340 and 7380 nM for hNaV1.8, hNaV1.3, hNaV1.7, hNaV1.5 and hNaV1.2 channels respectively).

Ambroxol HCl

Sodium Channel inhibitor
AmbroxolHCl is a potent inhibitor of the neuronal Na+ channels, inhibits TTX-resistant Na+ currents with IC50 of 35.2 uM and 22.5 uM for tonic and phasic block, inhibits TTX-sensitive Na+ currents with IC50 of 100 uM. Phase 3.
A10064 SALE

Amiloride HCl

Na+ channel blocker
Amiloride hydrochloride is a Na+ channel blocker, also inhibits TRPP3 channels and Na+/H+ exchanger (NHE).
A11728 SALE

Amiloride hydrochloride dihydrate

Amiloride hydrochloride dihydrate is a potent epithelial sodium channel blocker and selective low threshold (T-type) calcium channel protein inhibitor (KD=30μM).


Benzocaine is the ethyl ester of p-aminobenzoic acid (PABA), it is a local anesthetic commonly used as a topical pain reliever or in cough drops.

Benzocaine hydrochloride

Benzocaine hydrochloride is a surface anesthetic that acts by preventing transmission of impulses along nerve fibers and at nerve endings.


Slows neuronal Na+ channel inactivation
beta-Pompilidotoxin is a peptide with the sequence H2N-Arg.
A10168 SALE

Bupivacaine HCl

Bupivacaine is a more potent inhibitor of cAMP production than are chemically related local anesthetics that are less prone to produce cardiovascular toxicity.


late INa Inhibitor
GS967 is a novel, potent, and selective inhibitor of cardiac late sodium current(late INa); inhibits ATX-II-induced late I(Na) in ventricular myocytes and isolated hearts with IC(50) values of 0.13 and 0.21 uM, respectively.
A11750 SALE

Ibutilide fumarate

Ibutilide is a Class III antiarrhythmic agent that is indicated for acute cardioconversion of atrial fibrillation and atrial flutter of a recent onset to sinus rhythm. It exerts its antiarrhythmic effect by induction of slow inward sodium current, which prolongs action potential and refractory period (physiology) of myocardial cells.
A10510 SALE


Lacosamide is a medication developed for the adjunctive treatment of partial-onset seizures and diabetic neuropathic pain.
A11873 SALE


Lamotrigine is a phenyltriazine sodium channel protein inhibitor of presynaptic neurons.


sodium channel inhibitor
Levobupivacaine is a local anaesthetic drug belonging to the amino amide group.
A10530 SALE

Lidocaine (Alphacaine)

Lidocaine (Alphacaine) is an anasthetic and class Ib antiarrhythmic agent. Blocks voltage-gated sodium channels in the inactivated state.
A11712 SALE

Orphenadrine citrate

Orphenadrine is known to have the following pharmacology: mACh receptor antagonist (anticholinergic); H1 receptor antagonist (antihistamine); NMDA receptor antagonist; NET blocker (norepinephrine reuptake inhibitor); Nav1.7, Nav1.8, and Nav1.9 sodium channel blocker; HERG potassium channel blocker.


sodium channel protein inhibitor
Oxcarbazepine is a sodium channel protein inhibitor.


SGLT2 inhibitor
PF-04971729 is a potent and selective inhibitor of the sodium-dependent glucose cotransporter 2.


Nav1.7 Inhibitor
PF-05089771 is a Selective Nav1.7 Inhibitor (IC50 = 11 nM) that interacts with the voltage-sensor domain (VSD) of domain IV.
A10721 SALE

Phenytoin (Lepitoin)

Phenytoin is a sodium channel protein inhibitor.
A10722 SALE

Phenytoin sodium (Dilantin)

Phenytoin sodium (Dilantin) is a sodium channel protein inhibitor.

Pilsicainide HCl

Sodium Channel Blocker
Pilsicainide is a water soluble selective Na+ channel blocker.

Procainamide HCl

Sodium channel blocker
Procainamide HCl is a sodium channel blocker, and also a DNA methyltransferase inhibitor.


voltage-gated sodium channel inhibitor
Procaine is a benzoic acid derivative with local anesthetic and antiarrhythmic properties.
A11715 SALE

Proparacaine HCl

Voltage-gated sodium channels antagonist
Proparacaine HCl is a voltage-gated sodium channels antagonist with ED50 of 3.4 mM.
A13760 SALE

QX 314 chloride

Sodium channel Blocker
QX 314 chloride is a membrane impermeable quaternary derivative of lidocaine, a voltage-activated Na+ channel blocker

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