Dopamine Receptors



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Catalog No. Product Name Application Product Information
A16074

ACR 16 hydrochloride

dopaminergic stabilizer
ACR 16 hydrochloride is a dopaminergic stabilizer (Ki values 17550 nM and 7521 for D2(low) and D2(high), respectively) that state-dependently stabilizes psychomotor activity by the dual actions of functional dopamine D2 receptor antagonism and strengthening of cortical glutamate functions in various settings of perturbed neurotransmission.
A11297

Adoprazine (SLV313)

D2 receptor antagonist
Adoprazine is part of the Antidepressant Agent group
A16394

Alizapride HCl

Dopamine receptor antagonist
Alizapride HCl is a dopamine receptor antagonist used for the theropy of nausea and vomiting.
A10061

Amfebutamone (Bupropion)

-
Amfebutamone (Bupropion) is an atypical antidepressant and smoking cessation aid.
A14998

Amineptine

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Amineptine is a tricyclic antidepressant drug selectively blocking dopamine uptake, on 3H-imipramine binding, which was investigated in platelets of major depressed patients in conjunction with changes in clinical state.
A10067

Amisulpride

Dopamine Receptor antagonist
Amisulpride is an atypical antipsychotic used to treat psychosis in schizophrenia and episodes of mania in bipolar disorder.
A10091 SALE

Asenapine maleate

H1 antagonist
Asenapine shows high affinity (pKi) for numerous receptors, including the serotonin 5-HT1A (8.6), 5-HT1B (8.4), 5-HT2A (10.2), 5-HT2B (9.8), 5-HT2C (10.5), 5-HT5A (8.8), 5-HT6 (9.5), and 5-HT7 (9.9) receptors, the adrenergic α1 (8.9), α2A (8.9), α2B (9.5), and α2C (8.9) receptors, the dopamine D1 (8.9), D2 (8.9), D3 (9.4), and D4 (9.0) receptors, and the histamine H1 (9.0) and H2 (8.2) receptors.
A16416

Azaperone

Dopamine receptor antagonist
Azaperone is a pyridinylpiperazine and butyrophenone neuroleptic drug with sedative and antiemetic effects, which is used mainly as a tranquilizer in veterinary medicine.
A11341

B-HT 920 2HCl

D2 receptor agonist
B-HT 920 is a dopamine agonist that has been proposed as an antiparkinsonian agent. It also has α1-adrenergic and α2-adrenergic agonist activity.
A10125

Benserazide HCl (Serazide)

-
Benserazid hydrochloride is an inhibitor of L-aromatic amino acid decarboxylase.
A11824

Blonanserin

D2/5-HT2 receptor antagonist
Blonanserin is a D2/5-HT2 receptor antagonist; atypical antipsychotic.
A12415 SALE

BP897

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BP 897, is an antagonist at human dopamine D3 receptors and at rat somatodendritic dopamine D3 receptors
A15850

Bupropion

NDR Inhibitor
Bupropion is a medication primarily used as an antidepressant and smoking cessation aid.
A15936 SALE

C-DIM12

Nurr1 activator
C-DIM12 is a novel synthetic activator of Nurr1. C-DIM12 induces dopaminergic gene expression and protects against 6-hydroxydopamine neurotoxicity in vitro.
A13844

Cabergoline

Dopamine receptor agonist
Cabergoline, a lysergic acid amide derivative, is a potent dopamine D2 receptor agonist.
A15036

Cariprazine hydrochloride

D3/D2 Dopamine Receptor Antagonist
Cariprazine hydrochloride is a novel antipsychotic drug candidate that exhibits high selectivity and affinity to dopamine D3(Ki=0.09 nM) and D2 (Ki=0.5 nM) receptors and moderate affinity to serotonin 5-HT(1A) receptors.
A12347 SALE

cis-(Z)-Flupentixol dihydrochloride

Dopamine receptor antagonist
cis-(Z)-Flupentixol dihydrochloride is a dopamine receptor antagonist, antipsychotic, neuroleptic agent.
A10236 SALE

Clozapine

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Clozapine displays a broad range of pharmacological actions; the antipsychotic effects are thought to be mediated principally by 5-HT2A/2C and dopamine receptor blockade.
A10329 SALE

Domperidone

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Domperidone blocks the action of dopamine. It has strong affinities for the D2 and D3 dopamine receptors, which are found in the chemoreceptor trigger zone, located just outside the blood brain barrier, which, among others, regulates nausea and vomiting (area postrema on the floor of the fourth ventricle and rhomboid fossa).
A10331 SALE

Dopamine hydrochloride

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Dopamine (abbreviated as DA), a simple organic chemical in the catecholamine family, is a monoamine neurotransmitter - a chemical released by nerve cells to send signals to other nerve cells.
A13089

ent Naxagolide Hydrochloride

dopamine D2-receptor agonist
ent Naxagolide Hydrochloride is a dopamine D2-receptor agonist which is used for the treatment of extrapyramidal disorders. This compound is an antiparkinsonian drug.
A11720

Fenoldopam

-
Fenoldopam is used as an antihypertensive agent postoperatively, and also intravenously (IV) to treat a hypertensive crisis.
A13128 SALE

GBR 12783 dihydrochloride

dopamine uptake inhibitor
GBR 12783 dihydrochloride is a very potent and selective inhibitor of dopamine uptake (IC50 for inhibition of [3H]-dopamine uptake in rat striatal synaptosomes is 1.8 nM).
A11937 SALE

GBR-12935 2HCl

DAT and SLC6A2 inhibitor
GBR-12935 is a piperazine derivative which is a potent and selective dopamine reuptake inhibitor.
A12991

GR 103691

-
GR 103691 is an effective and selective receptor antagonist of the dopamine D3 receptor (D3DR).

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