Adrenergic Receptors

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  1. Asenapine maleate

    Catalog No. A10091
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    H1 antagonist
    Asenapine shows high affinity (pKi) for numerous receptors, including the serotonin 5-HT1A (8.6), 5-HT1B (8.4), 5-HT2A (10.2), 5-HT2B (9.8), 5-HT2C (10.5), 5-HT5A (8.8), 5-HT6 (9.5), and 5-HT7 (9.9) receptors, the adrenergic α1 (8.9), α2A (8.9), α2B (9.5), and α2C (8.9) receptors, the dopamine D1 (8.9), D2 (8.9), D3 (9.4), and D4 (9.0) receptors, and the histamine H1 (9.0) and H2 (8.2) receptors. Learn More
  2. Clonidine hydrochloride

    Catalog No. A10232
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    Alpha adrenergic agonist
    Clonidine is classified as a centrally acting alpha adrenergic agonist.Clonidine acts centrally as an imidazoline receptor agonist. Learn More
  3. Dehydroepiandrosterone

    Catalog No. A10296
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    Dehydroepiandrosterone is an important endogenous steroid hormone. Learn More
  4. Dobutamine hydrochloride

    Catalog No. A10325
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    Adrenoceptors agonist
    Dobutamine is a direct-acting agent whose primary activity results from stimulation of the β1-adrenoceptors of the heart, increasing contractility and cardiac output. Learn More
  5. Betaxolol

    Catalog No. A11721
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    Betaxolol is a selective beta1 receptor blocker used in the treatment of hypertension and glaucoma. Being selective for beta1 receptors, it typically has fewer systemic side effects than non-selective beta-blockers, for example, not causing bronchospasm (mediated by beta2 receptors) as timolol may. Betaxolol also shows greater affininty for beta1 receptors than metoprolol. Learn More
  6. Metoprolol tartrate

    Catalog No. A11713
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    Beta1 receptor blocker
    Metoprolol is a selective β1 receptor blocker used in treatment of several diseases of the cardiovascular system, especially hypertension. Learn More
  7. Salbutamol sulfate (Albuterol)

    Catalog No. A10819
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    Adrenergic Receptor agonist
    Salbutamol sulfate (Albuterol) is a short-acting β2-adrenergic receptor agonist used for the relief of bronchospasm in conditions such as asthma and chronic obstructive pulmonary disease. Learn More
  8. Naftopidil 2HCl

    Catalog No. A10619
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    5-HT1A and α1-adrenergic receptor antagonist
    Naftopidil 2HCl is a selective 5-HT1A and α1-adrenergic receptor antagonist with IC50 of 0.1 μM and 0.2 μM, respectively. Learn More
  9. Silodosin (Rapaflo)

    Catalog No. A10843
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    α1-adrenoceptor antagonist
    Silodosin(Rapaflo) is an α1-adrenoceptor antagonist with high uroselectivity. It causes practically no orthostatic hypotension (in contrast to other α1 blockers). Learn More
  10. Alfuzosin HCl

    Catalog No. A10052
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    Alfuzosin (provided as the hydrochloride salt) is an α1 receptor antagonist used to treat benign prostatic hyperplasia (BPH). It works by relaxing the muscles in the prostate and bladder neck, making it easier to urinate. Learn More
  11. Bisoprolol fumarate

    Catalog No. A10149
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    β1 adrenergic receptor blocker
    Bisoprolol is a drug belonging to the group of beta blockers, a class of drugs used primarily in cardiovascular diseases. More specifically, it is a selective type β1 adrenergic receptor blocker. Learn More
  12. Phenylephrine HCl

    Catalog No. A11666
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    α1-adrenergic receptor agonist
    Phenylephrine is a selective α1-adrenergic receptor agonist used primarily as a decongestant, as an agent to dilate the pupil, and to increase blood pressure. Learn More
  13. DL-Adrenaline

    Catalog No. A11668
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    DL-Adrenaline is a hormone and a neurotransmitter secreted by the medulla of the adrenal glands. DL-Adrenaline is found in small amounts in the body and is essential for maintaining cardiovascular homeostasis because of its ability to divert blood to tissues under stress. Learn More
  14. Isoprenaline HCl

    Catalog No. A10484
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    β adrenoceptor agonist
    Isoprenaline or isoproterenol is a non-selective beta-adrenergic agonist and structurally similar to adrenaline. Learn More
  15. Apalutamide (ARN-509)

    Catalog No. A11923
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    Androgen Receptor inhibitor
    ARN-509 is an androgen receptor antagonist with potential antineoplastic activity. ARN-509 binds to AR in target tissues thereby preventing androgen-induced receptor activation and facilitating the formation of inactive complexes that cannot be translocated to the nucleus. This prevents binding to and transcription of AR-responsive genes. Learn More
  16. Doxazosin mesylate

    Catalog No. A10334
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    Doxazosin mesylate, a quinazoline compound, is an α1-selective alpha blocker used to treat high blood pressure and urinary retention associated with benign prostatic hyperplasia (BPH). Learn More
  17. Metroprolol succinate

    Catalog No. A11229
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    Metoprolol succinate is a cardioselective β-adrenergic receptor blocker with IC50 of 42 ng/mL. Learn More
  18. Arformoterol tartrate

    Catalog No. A12795
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    beta2-adrenergic agonist
    Arformoterol tartrate is a beta2-adrenergic agonist Learn More
  19. Mirabegron

    Catalog No. A12861
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    β3 adrenergic receptor activator
    Mirabegron is a potent bladder relaxant and reagent for diabetes remedy. Learn More
  20. Oxymetazoline hydrochloride

    Catalog No. A10686
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    alpha-1 adrenergic agonist
    Oxymetazoline is a selective alpha-1 agonist and partial alpha-2 agonist topical decongestant, used in the form of Oxymetazoline hydrochloride. Learn More
  21. Tetrahydrozoline Hydrochloride

    Catalog No. A13080
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    Adrenergic Receptor agonist
    Tetrahydrozoline Hydrochloride is an alpha agonist which causes constriction of conjunctival blood vessels. Learn More
  22. ICI 118,551 hydrochloride

    Catalog No. A13225
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    β2 adrenergic antagonist
    ICI 118551 hydrochloride is a selective β2 adrenergic antagonist. Learn More
  23. Maprotiline hydrochloride

    Catalog No. A10555
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    noradrenalin re-uptake inhibitor
    Maprotiline hydrochloride is a selective noradrenalin re-uptake inhibitor. Learn More
  24. Bisoprolol

    Catalog No. A13406
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  25. Octopamine hydrochloride

    Catalog No. A13419
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    Octopamine hydrochloride is an invertebrate biogenic amine neurotransmitter, related to noradrenalin, that is an adrenoceptor agonist. Learn More
  26. Pindolol

    Catalog No. A13422
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    Beta adrenergic receptor blocker
    Pindolol is a nonselective beta blocker with partial beta-adrenergic receptor agonist activity. Learn More
  27. Tamsulosin

    Catalog No. A12657
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    alpha-1A/alpha-1B-adrenoceptor antagonist
    Tamsulosin is an alpha1a-selective alpha blocker used in the symptomatic treatment of benign prostatic hyperplasia (BPH). Learn More
  28. Ivabradine HCl (Procoralan)

    Catalog No. A11868
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    Ivabradine Hydrochloride, also known as S-16257, is the hydrochloride salt preparation of Ivabradine, a bradycardic agent. Learn More
  29. Prazosin HCl

    Catalog No. A11914
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    Prazosin HCl is an α1 and α2B-adrenoceptor antagonist. Also a potent antagonist at the melatonin MT3 receptor (Ki = 10.2 nM). Learn More
  30. Procaterol HCl

    Catalog No. A11905
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    Procaterol is a short-acting β2-adrenergic receptor agonist with Kp of 8 nM, used for the treatment of asthma Learn More
  31. Rilmenidine

    Catalog No. A10794
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    α2 adrenergic agonist
    Rilmenidine is a second-generation imidazoline-α2 adrenergic agonist. Learn More
  32. Naftopidil (Flivas)

    Catalog No. A10618
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    Naftopidil (Flivas) is a selective α1-adrenergic receptor antagonist or alpha blocker with a Ki of 58.3 nM. Learn More
  33. Nebivolol HCl

    Catalog No. A10630
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    Nebivolol hydrochloride is t a highly selective antagonist of the β1-adrenoceptor (Ki = 0.88 nM, β2-adrenoceptor Ki = 48 nM). Learn More
  34. Phenoxybenzamine hydrochloride

    Catalog No. A10719
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    α-adrenergic (AR) antagonist/CaM inhibitor
    Phenoxybenzamine is a cell-permeable, non-specific, irreversible α-adrenergic (AR) antagonist that also acts as an CaM inhibitor. Learn More
  35. Carvedilol

    Catalog No. A11843
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    β2-adrenergic receptor
    Carvedilol is a β1- and β2-adrenergic receptor (AR) agonist with antioxidant properties. Learn More
  36. Salmeterol

    Catalog No. A11788
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    beta2-adrenergic receptor agonist
    Salmeterol is a long-acting beta2-adrenergic receptor agonist Learn More
  37. Adrenalone HCl

    Catalog No. A11807
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    adrenergic agonist
    Adrenalone is an adrenergic agonist used as a topical vasoconstrictor and hemostatic, mainly acts on alpha-1 adrenergic receptors. Learn More
  38. Nebivolol

    Catalog No. A13738
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    Beta-1 adrenergic receptor blocker
    Nebivolol is a selective inhibits Beta-1 adrenergic receptor with IC50 of 0.8 nM Learn More

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