Adrenergic Receptors



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Catalog No. Product Name Application Product Information
A13738

Nebivolol

Beta-1 adrenergic receptor blocker
Nebivolol is a selective inhibits Beta-1 adrenergic receptor with IC50 of 0.8 nM
A13635

Guanabenz acetate

2A-AR adrenergic agonist
Guanabenz acetate is an a2A-AR adrenergic agonist and IGRS (imidazoline I2 binding site) selective ligand.
A13399

BRL 44408 maleate

Adrenoceptors antagonist
BRL 44408 maleate is a high purity Adrenoceptors antagonist. It increases hippocampal noradrenalin release following systemic administration.
A13401

Cimaterol

β-adrenergic receptors agonist
Cimaterol is a potent agonist of β-adrenergic receptors (pEC50 = 8.13, 8.78, and 6.62 for human β1, β2, and β3, respectively).
A13408

HEAT hydrochloride (BE 2254)

Adrenergic α1 Receptor Antagonist
HEAT hydrochloride is a very selective α1-AR adrenoceptor antagonist, precursor of the 3-[125I]-derivative. Adrenoreceptors (AR) or adrenergic receptors are G-protein coupled receptors involved in a variety of sympathetic nervous system processes.
A13409

Idazoxan Hydrochloride

α2- adrenoceptor antagonist / I2 imidazoline receptor agonist
Idazoxan hydrochloride is an α2-AR adrenoceptor antagonist and potential I2 imidazoline receptor agonist. Also displays I1 imidazoline receptor antagonist activity. (pKi values are 5.90, 7.22, 8.01, 7.43, and 7.7 for I1, I2, α 2A, α2B, and α 2C receptors respectively).
A13412

JP 1302 2HCl

α2C antagonist
JP 1302 2HCl is a potent and selective α2C antagonist.
A13417

NAN-190 hydrobromide

5-HT1A receptor antagonist
NAN-190 is a drug and research chemical widely used in scientific studies. It was previously believed to act as a selective 5-HT1A receptor antagonist, but a subsequent discovery showed that it also potently blocks the α2-adrenergic receptor.
A13421

Phentolamine HCl

α-Adrenergic blocker
Phentolamine Hydrochloride is an AR (α-Adrenergic) blocker.
A13623

Celiprolol HCl

adrenergic receptor antagonist
Celiprolol HCl is a b1 adrenergic receptor antagonist and a b2 adrenergic receptor partial agonist that has been shown to relax human arteries and veins with ED50 values of 40-50 M in vitro.
A13676

BRL 37344 Na Salt

β3-adrenergic receptors agonist
BRL-37344 is a b3-AR (b 3-adrenoceptor) selective agonist with lipolytic activity.
A13657

CL 316243 disodium salt

β3 adrenergic agonist
CL 316243 disodium salt, a beta-3 adrenergic agonist, was developed as an anti-obesity and diabetes drug, and causes rapid decreases in blood glucose levels in mice.
A11971

Diprophylline

AR antagonist
Diprophylline is a xanthine derivative with bronchodilator and vasodilator effects.
A14223 SALE

Salmeterol Xinafoate

β2-adrenoceptor agonist
Salmeterol Xinafoate is a long-acting β2-adrenergic receptor agonist with anti-inflammatory effect.
A14239 SALE

Labetalol HCl

alpha1/beta adrenergic receptors antagonist
Labetalol HCl is a dual antagonist for both selective alpha1-adrenergic and nonselective beta-adrenergic receptors.
A14251

Bambuterol HCl

β-adrenoceptor agonist
Bambuterol HCl is a potent β-adrenoceptor agonist, used in the treatment of asthma.
A14258

Carteolol HCl

β-adrenoceptor antagonist
Carteolol HCl is a β-adrenoceptor antagonist
A13902

Atipamezole HCl

α2 adrenergic receptor antagonist
Atipamezole HCl is a selective α2-adrenergic receptor antagonist (Ki values are 1.1, 1.0, 0.89, 1300 and 6500 nM for α2A, α2B, α2C, α1A and α1B receptors respectively). Has been shown to be a brain penetrant.
A11846 SALE

Dexmedetomidine HCl

alpha2-adrenoceptor agonist
Dexmedetomidine hydrochloride is the active isomer of medetomide which acts a potent, highly selective alpha2-AR (alpha2-adrenoceptor) agonist.
A13775

Medetomidine HCl

adrenergic alpha-2 receptor agonist
Medetomidine Hydrochloride is an adrenergic alpha-2 receptor agonist, which is used in veterinary medicine for its analgesic and sedative properties.
A13426

Rauwolscine

α2-adrenergic receptor antagonist
Rauwolscine is a natural alkaloid that acts as a selective and reversible α2-adrenergic receptor antagonist (Ki = 12 nM).
A13427

S-(-)-Atenolol

Adrenoceptors antagonist
S-(-)-Atenolol is the active enantiomer of atenolol that is a cardioselective β-adrenergic blocker.
A13428

S(-)-Propranolol HCl

β-adrenergic blocker
S(-)-Propranolol Hydrochloride is a small molecule β-adrenergic receptor antagonist and the active isomer of (??)-Propranolol preparations.
A15491

Desvenlafaxine succinate hydrate

serotonin (5-HT)/norepinephrine (NE) reuptake inhibitor
Desvenlafaxine succinate hydrate is an antidepressant of the serotonin-norepinephrine reuptake inhibitor (SNRI).
A11538

Pardoprunox HCl (SLV-308)

-
Pardoprunox is an antiparkinsonian drug currently under development by Solvay for the treatment of Parkinson's disease.
A15878

ICI-118551

β2 adrenergic receptor antagonist
ICI-118551 is a selective beta2 adrenergic receptor (adrenoreceptor) antagonist.
A15998 SALE

Vilanterol trifenatate

β2-adrenergic receptor agonist
Vilanterol is a long-acting beta-2 agonist drug, which in May 2013 was approved in combination with fluticasone furoate for sale as Breo Ellipta by GlaxoSmithKline for the treatment of chronic obstructive pulmonary disease (COPD).
A16170

Modafinil

-
Modafinil is a wakefulness-promoting agent (or eugeroic) used for treatment of disorders such as narcolepsy, shift work sleep disorder, and excessive daytime sleepiness associated with obstructive sleep apnea.
A16186

TAK 259

α1D Adrenoceptor Antagonist
TAK-259 is a Novel, Selective, and Orally Active α1D Adrenoceptor Antagonist (α1D, Ki = 1.1 nM) with Anti-urinary Frequency Effects and Reducing Human Ether-a-go-go-Related Gene (hERG) Liabilities.
A15033

Brimonidine Tartrate

α-adrenergic receptor agonist
Brimonidine Tartrate is a highly selective α-adrenergic receptor agonist with EC50 of 0.45 nM for the α2A adrenoreceptor, and used to treat open-angle glaucoma or ocular hypertension.
A16387

Acebutolol HCl

β-adrenergic receptors antagonist
Acebutolol is a β-adrenergic receptors antagonist used in the treatment of hypertension, angina pectoris and cardiac arrhythmias.
A15002

Asenapine HCl

adrenergic receptor/5-HT receptor inhibitor
Asenapine hydrochloride inhibits adrenergic receptor (α1, α2A, α2B, α2C) with Ki of 0.25-1.2 nM and also inhibits 5-HT receptor (1A, 1B, 2A, 2B, 2C, 5A, 6, 7) with Ki of 0.03-4.0 nM.
A15266

Trenbolone

-
Trenbolone is a steroid used by veterinarians on livestock to increase muscle growth and appetite.
A15117

HOKU-81

Metabolites of tulobuterol
HOKU-81, a new bronchodilator, is one of the metabolites of tulobuterol.
A13429

(S)-Timolol maleate

Adrenoceptors antagonist
(S)-Timolol maleate is a adrenergic receptor antagonist selective for β1-AR.
A13430

SR 59230A HCl

Adrenoceptors antagonist
SR 59230A hydrochloride is a β3-adrenoceptor antagonist.
A13432

Tulobuterol

Adrenergic Receptor agonist
Tulobuterol is a beta-adrenergic receptor agonist that is related structurally to Terbutaline.
A13433

UK 14,304 tartrate

Adrenoceptors agonist
UK 14,304 tartrate is a water-soluble form UK 14,304. It is a full α2 adrenergic agonist.
A13434

Xylazine HCl

Adrenergic Receptor agonist
Xylazine hydrochloride is an activator of α2A-AR, α2B-AR and α2C-AR.
A14936

Tamsulosin hydrochloride

α1 receptor antagonist
Tamsulosin hydrochloride is a selective α1 receptor antagonist and a medicine which is used in benign prostatic hyperplasia.
A14964

(R,R)-Formoterol

β2-adrenoceptor agonist
Formoterol is a long-acting β2 agonist used in the management of asthma and chronic obstructive pulmonary disease (COPD).
A15098 SALE

Guanfacine hydrochloride

α2A-adrenoceptor agonist
Guanfacine hydrochloride, an anti-hypertensive agent, is a selective α2A-adrenoceptor agonist with Kd of 31 nM and displays 60-fold selectivity over ??2B-adrenoceptors.
A16465

Clorprenaline HCl

β2-adrenergic receptor agonist
Clorprenaline HCl is a β2-receptor agonist, it has a significant expansion of the bronchial effect.
A13422

Pindolol

Beta adrenergic receptor blocker
Pindolol is a nonselective beta blocker with partial beta-adrenergic receptor agonist activity.
A10882 SALE

Synephrine (Oxedrine)

Adrenergic Receptor agonist
Synephrine (Oxedrine) is an amine compound commonly used for weight loss.
A11732

Formoterol hemifumarate

-
Formoterol is a long-acting β2-agonist used in the management of asthma and/or chronic obstructive pulmonary disease (COPD).
A11733

Betaxolol hydrochloride

-
A11734 SALE

Phentolamine mesilate

-
Phentolamine is a reversible nonselective alpha-adrenergic antagonist.
A11740 SALE

Terazosin hydrochloride

-
Terazosin is a selective alpha 1 antagonist used for treatment of symptoms of an enlarged prostate (BPH).
A10298

Detomidine hydrochloride

Adrenergic Receptor agonist
Detomidine is a sedative with analgesic properties. α2-adrenergic agonists produce dose-dependent sedative and analgesic effects, mediatated by activation of α2 catecholamine receptors, thus inducing a negative feedback response, reducing production of excitatory neurotransmitters.

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