Adrenergic Receptors

Actions
  1. Agonist (7)
  2. Antagonist (2)
  3. Blocker (1)
  4. Inhibitor (2)


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Catalog No. Product Name Application Product Information
A11807

Adrenalone HCl

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Adrenalone is an adrenergic agonist used as a topical vasoconstrictor and hemostatic, mainly acts on alpha-1 adrenergic receptors.
A10052

Alfuzosin HCl

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Alfuzosin (provided as the hydrochloride salt) is an α1 receptor antagonist used to treat benign prostatic hyperplasia (BPH). It works by relaxing the muscles in the prostate and bladder neck, making it easier to urinate.
A12795

Arformoterol tartrate

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Arformoterol tartrate is a beta2-adrenergic agonist
A11923

ARN-509

Androgen Receptor inhibitor
ARN-509 is an androgen receptor antagonist with potential antineoplastic activity. ARN-509 binds to AR in target tissues thereby preventing androgen-induced receptor activation and facilitating the formation of inactive complexes that cannot be translocated to the nucleus. This prevents binding to and transcription of AR-responsive genes.
A11721

Betaxolol

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Betaxolol is a selective beta1 receptor blocker used in the treatment of hypertension and glaucoma. Being selective for beta1 receptors, it typically has fewer systemic side effects than non-selective beta-blockers, for example, not causing bronchospasm (mediated by beta2 receptors) as timolol may. Betaxolol also shows greater affininty for beta1 receptors than metoprolol.
A11733

Betaxolol hydrochloride

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A13406

Bisoprolol

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A10149

Bisoprolol fumarate

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Bisoprolol is a drug belonging to the group of beta blockers, a class of drugs used primarily in cardiovascular diseases. More specifically, it is a selective type β1 adrenergic receptor blocker.
A11843

Carvedilol

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Carvedilol is a β1- and β2-adrenergic receptor (AR) agonist with antioxidant properties.
A10232

Clonidine hydrochloride

Alpha adrenergic agonist
Clonidine is classified as a centrally acting alpha adrenergic agonist.Clonidine acts centrally as an imidazoline receptor agonist.
A10296

Dehydroepiandrosterone

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Dehydroepiandrosterone is an important endogenous steroid hormone.
A10298

Detomidine hydrochloride

Adrenergic Receptor agonist
Detomidine is a sedative with analgesic properties. α2-adrenergic agonists produce dose-dependent sedative and analgesic effects, mediatated by activation of α2 catecholamine receptors, thus inducing a negative feedback response, reducing production of excitatory neurotransmitters.
A11668

DL-Adrenaline

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DL-Adrenaline is a hormone and a neurotransmitter secreted by the medulla of the adrenal glands. DL-Adrenaline is found in small amounts in the body and is essential for maintaining cardiovascular homeostasis because of its ability to divert blood to tissues under stress.
A10325

Dobutamine hydrochloride

Adrenoceptors agonist
Dobutamine is a direct-acting agent whose primary activity results from stimulation of the β1-adrenoceptors of the heart, increasing contractility and cardiac output.
A10334

Doxazosin mesylate

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Doxazosin mesylate, a quinazoline compound, is an α1-selective alpha blocker used to treat high blood pressure and urinary retention associated with benign prostatic hyperplasia (BPH).
A12844

Formoterol

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Formoterol is a long-acting ??2-agonist used in the management of asthma and/or chronic obstructive pulmonary disease (COPD).
A11732

Formoterol hemifumarate

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Formoterol is a long-acting β2-agonist used in the management of asthma and/or chronic obstructive pulmonary disease (COPD).
A13225

ICI 118,551 hydrochloride

β2 adrenergic antagonist
ICI 118551 hydrochloride is a selective ??2 adrenergic antagonist.
A10484

Isoprenaline HCl

β adrenoceptor agonist
Isoprenaline or isoproterenol is a non-selective beta-adrenergic agonist and structurally similar to adrenaline.
A11868

Ivabradine HCl (Procoralan)

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Ivabradine Hydrochloride, also known as S-16257, is the hydrochloride salt preparation of Ivabradine, a bradycardic agent.
A10555

Maprotiline hydrochloride

noradrenalin re-uptake inhibitor
Maprotiline hydrochloride is a selective noradrenalin re-uptake inhibitor.
A11713

Metoprolol tartrate

Beta1 receptor blocker
Metoprolol is a selective β1 receptor blocker used in treatment of several diseases of the cardiovascular system, especially hypertension.
A11229

Metroprolol succinate

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Metoprolol succinate is a cardioselective β-adrenergic receptor blocker with IC50 of 42 ng/mL.
A10618

Naftopidil (Flivas)

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Naftopidil (Flivas) is a selective α1-adrenergic receptor antagonist or alpha blocker with a Ki of 58.3 nM.
A10619

Naftopidil 2HCl

5-HT1A and α1-adrenergic receptor antagonist
Naftopidil 2HCl is a selective 5-HT1A and α1-adrenergic receptor antagonist with IC50 of 0.1 μM and 0.2 μM, respectively.

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