Histamine Receptors



23 Item(s)

per page

Set Descending Direction
Catalog No. Product Name Application Product Information
A10117

Azelastine HCl (Allergodil)

-
Azelastine is a potent, second-generation, selective, histamine antagonist (histamine-H1-receptor antagonist).
A15015

Bavisant dihydrochloride

-
Bavisant dihydrochloride is a highly selective, orally active antagonist of the human H3 receptor with a novel mechanism of action, involving wakefulness and cognition, with potential as a treatment for ADHD.
A15016

Bavisant dihydrochloride hydrate

-
Bavisant dihydrochloride hydrate is a highly selective, orally active antagonist of the human H3 receptor with a novel mechanism of action, involving wakefulness and cognition, with potential as a treatment for ADHD.
A12845

Bepotastine

-
Bepotastine is a non-sedating, selective antagonist of the histamine 1 (H1) receptor.
A11340

Bepotastine Besilate

Histamine Receptor antagonist
Bepotastine Beslilate (Bepreve) is a histamine H1 receptor anatagonist.
A12661

Bilastine

-
Bilastine is a novel, nonsedating H1-antihistamine developed for symptomatic treatment of allergic rhinitis and chronic idiopathic urticaria.
A11699

Brompheniramine

-
Brompheniramine is a first-generation antihistamine. Brompheniramine works by acting as an antagonist of histamine H1 receptors. It also functions as a moderately effective anticholinergic agent, and is likely an antimuscarinic agent similar to other common antihistamines such as diphenhydramine.
A10195

Cetirizine Dihydrochloride

-
Cetirizine is a second-generation antihistamine, a major metabolite of hydroxyzine, and a racemic selective H1 receptor inverse agonist used in the treatment of allergies, hay fever, angioedema, and urticaria.
A10205

Chlorpheniramine maleate

-
Chlorpheniramine maleate is a first-generation alkylamine antihistamine used in the prevention of the symptoms of allergic conditions such as rhinitis and urticaria.
A10218

Cimetidine

H2-receptor antagonist
Cimetidine is a histamine H2-receptor antagonist that inhibits stomach acid production.
A11360

Ciproxifan

-
Ciproxifan is an extremely potent histamine H3 inverse agonist/antagonist.
A11117

Ciproxifan maleate

H3-receptor antagonist
Ciproxifan maleate is a potent, selective H3 histamine receptor antagonist.
A10226

Clemastine fumarate

Histamine Receptor antagonis
Clemastine is a selective histamine H1 antagonist. It binds to the histamine H1 receptor, thus blocking the action of endogenous histamine, which leads to temporary relief of the negative symptoms caused by histamine.
A11709

Cyproheptadine hydrochloride

-
A11859

Fexofenadine HCl

COX inhibitor/histamine H1 receptor agonist
Fexofenadine HCl is an antihistamine that inhibits Cox-1, Cox-2, and is a histamine H1 receptor agonist
A12713

JNJ7777120

Histamine Antagonist
JNJ7777120 is a potent, selective non-imidazole H4?histamine receptor antagonist.
A10538

Loratadine

-
Loratadine is a non-sedative antihistamine that inhibits histamine-induced activities of IL-6 and IL-8 secretion in endothelial cells. Loratadine is a selective inverse peripheral histamine H1-receptor agonist with an IC50 of >32 μM.
A13086

Metiamide

Histamine H2-receptor antagonist
Metiamide is a histamine H2-receptor antagonist developed from another H2 antagonist, burimamide. It was an intermediate compound in the development of the successful anti-ulcer drug cimetidine.
A11724

Mizolastine

-
Mizolastine is a second generation antihistamine agent with high affinity and specificity for histamine H1 receptors.
A10671

Olopatadine hydrochloride

-
Olopatadine hydrochloride is a dual acting histamine H1-receptor antagonist and mast cell stabilizer
A11921

Roxatidine acetate hydrochloride

-
Roxatidine Acetate Hydrochloride is a histamine H2-receptor antagonist used in ulcer treatment. This compound has been found to inhibit platelet function in vitro.
A11222

Rupatadine

-
Rupatadine is an inhibitor of PAFR and histamine (H1) receptor with Ki of 550 and 102 nM, respectively.
A12356

Rupatadine Fumarate

-
Rupatadine is an inhibitor of PAFR and histamine (H1) receptor with Ki of 550 and 102 nM, respectively.

23 Item(s)

per page

Set Descending Direction