Histamine Receptors



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Catalog No. Product Name Application Product Information
A16393

Alcaftadine

H1 histamine receptor antagonist
Alcaftadine is a high affinity ligand for the H1 receptor, with a pKi (8.5) that is comparable with that of other H1 antihistamines. Alcaftadine is also an antagonist for H2 and H4 receptors with no affinity for the H3 receptor.
A16411

Antazoline HCl

Histamine H1 receptor inhibitor
Antazoline HCl is a first generation antihistamine, binding to the histamine H1 receptor and blocking the action of endogenous histamine.
A10091 SALE

Asenapine maleate

H1 antagonist
Asenapine shows high affinity (pKi) for numerous receptors, including the serotonin 5-HT1A (8.6), 5-HT1B (8.4), 5-HT2A (10.2), 5-HT2B (9.8), 5-HT2C (10.5), 5-HT5A (8.8), 5-HT6 (9.5), and 5-HT7 (9.9) receptors, the adrenergic α1 (8.9), α2A (8.9), α2B (9.5), and α2C (8.9) receptors, the dopamine D1 (8.9), D2 (8.9), D3 (9.4), and D4 (9.0) receptors, and the histamine H1 (9.0) and H2 (8.2) receptors.
A13899

Astemizole

H1-receptor antagonist
Astemizole is a potent antihistamine (H1-receptor antagonist, IC50 = 4 nM) that displays selectivity over dopamine, 5-HT, and muscarinic acetylcholine receptors. This compound has shown potent hERG K+ channel blocking activity (IC50 = 0.9 nM), antimalarial activity in multidrug resistant strains in vitro (IC50 = 227 - 734 nM), and has been used as a chaperone to correct folding defects and restore protein function for some mutated forms of hERG channels.
A16418

Azatadine dimaleate

Histamine/cholinergic inhibitor
Azatadine is an histamine and cholinergic inhibitor with IC50 of 6.5 nM and 10 nM, respectively.
A10117 SALE

Azelastine HCl (Allergodil)

-
Azelastine is a potent, second-generation, selective, histamine antagonist (histamine-H1-receptor antagonist).
A15015

Bavisant dihydrochloride

H3 receptor antagonist
Bavisant dihydrochloride is a highly selective, orally active antagonist of the human H3 receptor with a novel mechanism of action, involving wakefulness and cognition, with potential as a treatment for ADHD.
A15016

Bavisant dihydrochloride hydrate

H3 receptor antagonist
Bavisant dihydrochloride hydrate is a highly selective, orally active antagonist of the human H3 receptor with a novel mechanism of action, involving wakefulness and cognition, with potential as a treatment for ADHD.
A12845

Bepotastine

-
Bepotastine is a non-sedating, selective antagonist of the histamine 1 (H1) receptor.
A11340

Bepotastine Besilate

Histamine Receptor antagonist
Bepotastine Beslilate (Bepreve) is a histamine H1 receptor anatagonist.
A12661

Bilastine

-
Bilastine is a novel, nonsedating H1-antihistamine developed for symptomatic treatment of allergic rhinitis and chronic idiopathic urticaria.
A11699 SALE

Brompheniramine

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Brompheniramine is a first-generation antihistamine. Brompheniramine works by acting as an antagonist of histamine H1 receptors. It also functions as a moderately effective anticholinergic agent, and is likely an antimuscarinic agent similar to other common antihistamines such as diphenhydramine.
A15666

Buclizine HCl

-
Buclizine HCl is an antihistamine and anticholinergic of the piperazine derivative family.
A16129

CarbinoxaMine Maleate

histamine-H1 receptor blocking agent
Carbinoxamine maleate is a histamine-H1 receptor blocking agent with antihistamine and anticholinergic properties.
A15041

Cetirizine

H1-receptor antagonist
Cetirizine, a second-generation antihistamine, is a major metabolite of hydroxyzine, and a racemic selective H1 receptor inverse agonist used in the treatment of allergies, hay fever, angioedema, and urticaria.
A10195 SALE

Cetirizine Dihydrochloride

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Cetirizine is a second-generation antihistamine, a major metabolite of hydroxyzine, and a racemic selective H1 receptor inverse agonist used in the treatment of allergies, hay fever, angioedema, and urticaria.
A10205 SALE

Chlorpheniramine maleate

-
Chlorpheniramine maleate is a first-generation alkylamine antihistamine used in the prevention of the symptoms of allergic conditions such as rhinitis and urticaria.
A10218

Cimetidine

H2-receptor antagonist
Cimetidine is a histamine H2-receptor antagonist that inhibits stomach acid production.
A11360

Ciproxifan

-
Ciproxifan is an extremely potent histamine H3 inverse agonist/antagonist.
A11117

Ciproxifan maleate

H3-receptor antagonist
Ciproxifan maleate is a potent, selective H3 histamine receptor antagonist.
A10226 SALE

Clemastine fumarate

Histamine Receptor antagonis
Clemastine is a selective histamine H1 antagonist. It binds to the histamine H1 receptor, thus blocking the action of endogenous histamine, which leads to temporary relief of the negative symptoms caused by histamine.
A13073

Clemizole

H1 histamine receptor antagonist.
Clemizole is an H1 histamine receptor antagonist.
A15047

Clemizole hydrochloride

H1 histamine receptor antagonist
Clemizole hydrochloride is an antagonist of H1 histamine receptor with an IC50 value of 8 mM for NS4B RNA binding.
A16472

Cyclizine 2HCl

Histamine H1 receptor antagonist
Cyclizine 2HCl is a piperazine derivative with Histamine H1 receptor antagonist activity.
A16169

Cyproheptadine hydrochloride

serotonin/histamine2 antagonist
Cyproheptadine hydrochloride sesquihydrate is an antihistamine and is an antagonist of serotonin and histamine2.

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