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$0.00 Cysteine protease
| Catalog No. | Inhibitor Name | Cysteine Protease | Other |
|---|---|---|---|
| A11265 | Odanacatib (MK-0822) | **** | |
| A13257 | E-64 | *** | |
| A14245 | PD 151746 | * | |
| A15295 | Calpeptin | ** | |
| A11466 | Cathepsin Inhibitor 1 | *** | |
| A11901 | PMSF | chymotrypsin | |
| A13259 | Aloxistatin | ||
| A13258 | Loxistatin Acid (E-64C) | ||
| A14145 | Leupeptin Hemisulfate | serine protease | |
| A14284 | Z-FA-FMK | ||
| A14220 | MG-101 (ALLN) |
Notes:
1.Hover mouse over "" to view the IC50 value.(A few compounds have proven potency but without published IC50 data.)
2.For more details about the compound, click on the product name of your interest.
3.The higher the number of "" is, the more potent the inhibitor or activator is.
4."" refers to compounds which do inhibitory effects on the related isoform, but without specific value.
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Cathepsin Inhibitor 1
Catalog No. A11466 Cathepsin InhibitorCathepsin Inhibitor 1 is an inhibitor of Cathepsin (L, L2, S, K, B) with pIC50 of 7.9, 6.7, 6.0, 5.5 and 5.2, respectively. Learn More -
Calpeptin
Catalog No. A15295 Calpain inhibitorCalpeptin is a cell permeable calpain inhibitor. Learn More -
Acetyl-Calpastatin (184-210) (human)
Catalog No. A15290 Selective calpain inhibitorAcetyl-Calpastatin (184-210) (human), selective calpain inhibitor. Strongly inhibits calpain I (Ki = 0.2 nM) and II but does not inhibit papain, trypsin and cathepsin L (Ki = 6 uM). Increases secretion of amyoid β-protein (Aβ) 42, Aβ40 and Aβ42 ratio. Learn More -
Calpain Inhibitor II, ALLM
Catalog No. A14911 Calpain InhibitorCalpain Inhibitor II, ALLM is a cell-permeable inhibitor of calpain I, calpain II, cathepsin L and cathepsin B with Ki values of 120 nM, 230 nM, 0.6 nM and 100 nM, respectively. Learn More -
MDL 28170
Catalog No. A15303 Calpain Inhibitor IIIMDL 28170 is a cell permeable selective inhibitor of Calpain 1, a Ca2+-dependent cysteine protease which has been implicated in apoptosis of immune cells as well as neuronal cells. Learn More -
SJA6017
Catalog No. A13640 reversible Calpain inhibitorSJA6017 is a cell permeable peptide aldehyde which functions as a reversible calpain inhibitor. Learn More -
PD 150606
Catalog No. A15306 Non-peptide calpain inhibitorPD 150606 is a cell-permeable, non-competitive, selective, non-peptide Ca2+ dependent calpain inhibitor for calpain-1 and for calpain-2 directed towards the Ca2+ binding sites of calpain. Learn More -
Z-FA-FMK
Catalog No. A14284 Irreversible Cysteine Protease inhibitorZ-FA-FMK is an irreversible cysteine protease inhibitor. Learn More -
PD 151746
Catalog No. A14245 Calpain inhibitorPD 151746 is a selective, cell-permeable calpain inhibitor with Ki of 0.26 uM for μ-Calpain, about 20-fold selectivity over m-calpain. Learn More -
MG-101
Catalog No. A14220 Cysteine Protease inhibitorMG-101 (ALLN) is a cell-permeable and potent inhibitor of cysteine proteases including calpains and lysosomal cathepsins. Learn More -
Z-FA-FMK
Catalog No. A16381 Cysteine protease inhibitorZ-FA-FMK is an irreversible inhibitor of cysteine protease Learn More -
Balicatib
Catalog No. A12020 Cathepsin K inhibitorBalicatib, a cathepsin K inhibitor, stimulates periosteal bone formation in monkeys. Learn More -
Cysteine Protease inhibitor
Catalog No. A21048 cysteine protease inhibitorCysteine Protease inhibitor is an inhibitor of cysteine protease. Learn More -
CA-074 Methyl Ester
Catalog No. A13593 Cathepsin B inhibitorCA-074 methyl ester is a cell-permeable analog of CA-074 that acts as an irreversible cathepsin B inhibitor. CA-074 methyl ester is reported to inhibit bone resorption in rodent models and shown to inhibit B16 melanoma cell invasion in vitro. Learn More -
SID 26681509
Catalog No. A15313 Human cathepsin L inhibitorSID 26681509 is a reversible and potent human cathepsin L inhibitor. SID 26681509 displays no inhibitory activity of cathepsin G. Learn More -
L 006235
Catalog No. A15302 Cathepsin K InhibitorL006235 is a potent, reversible cathepsin K inhibitor (IC50 = 0.25 nM) that displays > 4000-fold selectivity over cathepsins B, L and S. Learn More -
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New
SNJ-1945
Catalog No. A17243 Calpain inhibitorSNJ-1945 is a calpain inhibitor with more favorable retinal penetration, high oral bioavailability, and long half-life. SNJ1945 rescued defective function in lissencephaly. Learn More -
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Z-FL-COCHO
Catalog No. A13502 Cathepsin S inhibitorZ-FL-COCHO is a novel Cathepsin S inhibitor. Learn More -
Odanacatib (MK-0822)
Catalog No. A11265 Cathepsin K InhibitorOdanacatib is an inhibitor of cathepsin K,an enzyme involved in bone resorption. Learn More -
Gly-Phe-beta-naphthylamide
Catalog No. A13611 cathepsin C substrateGly-Phe-beta-naphthylamide is a cathepsin C substrate. The compound is described to accumulate inside lysosomes leading to their destruction. Learn More -
E-64
Catalog No. A13257 Cysteine Protease inhibitorE-64 is an irreversible and selective cysteine protease inhibitor with IC50 of 9 nM for papain. Learn More -
Loxistatin Acid (E64-C)
Catalog No. A13258 Cysteine Protease inhibitorLoxistatin Acid, a derivative of E-64, is an irreversible and membrane-permeant cysteine protease inhibitor. Learn More -
Leupeptin hemisulfate
Catalog No. A14145 Cysteine Protease inhibitorLeupeptin hemisulfate is a reversible inhibitor of trypsin-like and cysteine proteases such as calpain. Learn More -
E 64d (Aloxistatin)
Catalog No. A13259 Cysteine Protease inhibitorE-64d is an inhibitor of cathepsins B and L and it is lysosome and cell permeable. Learn More -
CA-074
Catalog No. A13256 Cathepsin B inhibitorCA-074 is a potent inhibitor of cathepsin B with a Ki of 2 to 5 nM. Learn More
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