Adrenergic Receptors

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  1. Diprophylline

    Catalog No. A11971
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    AR antagonist
    Diprophylline is a xanthine derivative with bronchodilator and vasodilator effects. Learn More
  2. BRL 44408 maleate

    Catalog No. A13399
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    Adrenoceptors antagonist
    BRL 44408 maleate is a high purity Adrenoceptors antagonist. It increases hippocampal noradrenalin release following systemic administration. Learn More
  3. Cimaterol

    Catalog No. A13401
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    β-adrenergic receptors agonist
    Cimaterol is a potent agonist of β-adrenergic receptors (pEC50 = 8.13, 8.78, and 6.62 for human β1, β2, and β3, respectively). Learn More
  4. HEAT hydrochloride (BE 2254)

    Catalog No. A13408
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    Adrenergic α1 Receptor Antagonist
    HEAT hydrochloride is a very selective α1-AR adrenoceptor antagonist, precursor of the 3-[125I]-derivative. Adrenoreceptors (AR) or adrenergic receptors are G-protein coupled receptors involved in a variety of sympathetic nervous system processes. Learn More
  5. Idazoxan Hydrochloride

    Catalog No. A13409
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    α2- adrenoceptor antagonist / I2 imidazoline receptor agonist
    Idazoxan hydrochloride is an α2-AR adrenoceptor antagonist and potential I2 imidazoline receptor agonist. Also displays I1 imidazoline receptor antagonist activity. (pKi values are 5.90, 7.22, 8.01, 7.43, and 7.7 for I1, I2, α 2A, α2B, and α 2C receptors respectively). Learn More
  6. JP 1302 2HCl

    Catalog No. A13412
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    α2C antagonist
    JP 1302 2HCl is a potent and selective α2C antagonist. Learn More
  7. NAN-190 hydrobromide

    Catalog No. A13417
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    5-HT1A receptor antagonist
    NAN-190 is a drug and research chemical widely used in scientific studies. It was previously believed to act as a selective 5-HT1A receptor antagonist, but a subsequent discovery showed that it also potently blocks the α2-adrenergic receptor. Learn More
  8. Phentolamine HCl

    Catalog No. A13421
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    α-Adrenergic blocker
    Phentolamine Hydrochloride is an AR (α-Adrenergic) blocker. Learn More
  9. Rauwolscine

    Catalog No. A13426
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    α2-adrenergic receptor antagonist
    Rauwolscine is a natural alkaloid that acts as a selective and reversible α2-adrenergic receptor antagonist (Ki = 12 nM). Learn More
  10. S-(-)-Atenolol

    Catalog No. A13427
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    Adrenoceptors antagonist
    S-(-)-Atenolol is the active enantiomer of atenolol that is a cardioselective β-adrenergic blocker. Learn More
  11. Guanabenz acetate

    Catalog No. A13635
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    2A-AR adrenergic agonist
    Guanabenz acetate is an a2A-AR adrenergic agonist and IGRS (imidazoline I2 binding site) selective ligand. Learn More
  12. Celiprolol HCl

    Catalog No. A13623
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    adrenergic receptor antagonist
    Celiprolol HCl is a b1 adrenergic receptor antagonist and a b2 adrenergic receptor partial agonist that has been shown to relax human arteries and veins with ED50 values of 40-50 M in vitro. Learn More
  13. Salmeterol Xinafoate

    Catalog No. A14223
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    β2-adrenoceptor agonist
    Salmeterol Xinafoate is a long-acting β2-adrenergic receptor agonist with anti-inflammatory effect. Learn More
  14. Labetalol HCl

    Catalog No. A14239
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    alpha1/beta adrenergic receptors antagonist
    Labetalol HCl is a dual antagonist for both selective alpha1-adrenergic and nonselective beta-adrenergic receptors. Learn More
  15. Bambuterol HCl

    Catalog No. A14251
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    β-adrenoceptor agonist
    Bambuterol HCl is a potent β-adrenoceptor agonist, used in the treatment of asthma. Learn More
  16. Carteolol HCl

    Catalog No. A14258
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    β-adrenoceptor antagonist
    Carteolol HCl is a β-adrenoceptor antagonist Learn More
  17. Atipamezole HCl

    Catalog No. A13902
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    α2 adrenergic receptor antagonist
    Atipamezole HCl is a selective α2-adrenergic receptor antagonist (Ki values are 1.1, 1.0, 0.89, 1300 and 6500 nM for α2A, α2B, α2C, α1A and α1B receptors respectively). Has been shown to be a brain penetrant. Learn More
  18. Dexmedetomidine HCl

    Catalog No. A11846
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    alpha2-adrenoceptor agonist
    Dexmedetomidine hydrochloride is the active isomer of medetomide which acts a potent, highly selective alpha2-AR (alpha2-adrenoceptor) agonist. Learn More
  19. Medetomidine HCl

    Catalog No. A13775
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    adrenergic alpha-2 receptor agonist
    Medetomidine Hydrochloride is an adrenergic alpha-2 receptor agonist, which is used in veterinary medicine for its analgesic and sedative properties. Learn More
  20. CL 316243 disodium salt

    Catalog No. A13657
    β3 adrenergic agonist
    CL 316243 disodium salt, a beta-3 adrenergic agonist, was developed as an anti-obesity and diabetes drug, and causes rapid decreases in blood glucose levels in mice. Learn More
  21. BRL 37344 Na Salt

    Catalog No. A13676
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    β3-adrenergic receptors agonist
    BRL-37344 is a b3-AR (b 3-adrenoceptor) selective agonist with lipolytic activity. Learn More
  22. S(-)-Propranolol HCl

    Catalog No. A13428
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    β-adrenergic blocker
    S(-)-Propranolol Hydrochloride is a small molecule β-adrenergic receptor antagonist and the active isomer of (??)-Propranolol preparations. Learn More
  23. (S)-Timolol maleate

    Catalog No. A13429
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    Adrenoceptors antagonist
    (S)-Timolol maleate is a adrenergic receptor antagonist selective for β1-AR. Learn More
  24. Pardoprunox HCl (SLV-308)

    Catalog No. A11538
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    Pardoprunox is an antiparkinsonian drug currently under development by Solvay for the treatment of Parkinson's disease. Learn More
  25. ICI-118551

    Catalog No. A15878
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    β2 adrenergic receptor antagonist
    ICI-118551 is a selective beta2 adrenergic receptor (adrenoreceptor) antagonist. Learn More
  26. Vilanterol trifenatate

    Catalog No. A15998
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    β2-adrenergic receptor agonist
    Vilanterol is a long-acting beta-2 agonist drug, which in May 2013 was approved in combination with fluticasone furoate for sale as Breo Ellipta by GlaxoSmithKline for the treatment of chronic obstructive pulmonary disease (COPD). Learn More
  27. Modafinil

    Catalog No. A16170
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    Modafinil is a wakefulness-promoting agent (or eugeroic) used for treatment of disorders such as narcolepsy, shift work sleep disorder, and excessive daytime sleepiness associated with obstructive sleep apnea. Learn More
  28. TAK 259

    Catalog No. A16186
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    α1D Adrenoceptor Antagonist
    TAK-259 is a Novel, Selective, and Orally Active α1D Adrenoceptor Antagonist (α1D, Ki = 1.1 nM) with Anti-urinary Frequency Effects and Reducing Human Ether-a-go-go-Related Gene (hERG) Liabilities. Learn More
  29. Brimonidine Tartrate

    Catalog No. A15033
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    α-adrenergic receptor agonist
    Brimonidine Tartrate is a highly selective α-adrenergic receptor agonist with EC50 of 0.45 nM for the α2A adrenoreceptor, and used to treat open-angle glaucoma or ocular hypertension. Learn More
  30. Acebutolol HCl

    Catalog No. A16387
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    β-adrenergic receptors antagonist
    Acebutolol is a β-adrenergic receptors antagonist used in the treatment of hypertension, angina pectoris and cardiac arrhythmias. Learn More
  31. Clorprenaline HCl

    Catalog No. A16465
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    β2-adrenergic receptor agonist
    Clorprenaline HCl is a β2-receptor agonist, it has a significant expansion of the bronchial effect. Learn More
  32. Vilanterol

    Catalog No. A13125
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    ultra-long-acting β₂ adrenoreceptor agonist
    Vilanterol is a novel and selective agonist of Beta2-AR with a PEC50 value of 10.37±0.05. Learn More
  33. Desvenlafaxine succinate hydrate

    Catalog No. A15491
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    serotonin (5-HT)/norepinephrine (NE) reuptake inhibitor
    Desvenlafaxine succinate hydrate is an antidepressant of the serotonin-norepinephrine reuptake inhibitor (SNRI). Learn More
  34. Asenapine HCl

    Catalog No. A15002
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    adrenergic receptor/5-HT receptor inhibitor
    Asenapine hydrochloride inhibits adrenergic receptor (α1, α2A, α2B, α2C) with Ki of 0.25-1.2 nM and also inhibits 5-HT receptor (1A, 1B, 2A, 2B, 2C, 5A, 6, 7) with Ki of 0.03-4.0 nM. Learn More
  35. SR 59230A HCl

    Catalog No. A13430
    Adrenoceptors antagonist
    SR 59230A hydrochloride is a β3-adrenoceptor antagonist. Learn More
  36. Tulobuterol

    Catalog No. A13432
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    Adrenergic Receptor agonist
    Tulobuterol is a beta-adrenergic receptor agonist that is related structurally to Terbutaline. Learn More
  37. UK 14,304 tartrate

    Catalog No. A13433
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    Adrenoceptors agonist
    UK 14,304 tartrate is a water-soluble form UK 14,304. It is a full α2 adrenergic agonist. Learn More
  38. Xylazine HCl

    Catalog No. A13434
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    Adrenergic Receptor agonist
    Xylazine hydrochloride is an activator of α2A-AR, α2B-AR and α2C-AR. Learn More
  39. Tamsulosin hydrochloride

    Catalog No. A14936
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    α1 receptor antagonist
    Tamsulosin hydrochloride is a selective α1 receptor antagonist and a medicine which is used in benign prostatic hyperplasia. Learn More
  40. (R,R)-Formoterol

    Catalog No. A14964
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    β2-adrenoceptor agonist
    Formoterol is a long-acting β2 agonist used in the management of asthma and chronic obstructive pulmonary disease (COPD). Learn More
  41. Guanfacine hydrochloride

    Catalog No. A15098
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    α2A-adrenoceptor agonist
    Guanfacine hydrochloride, an anti-hypertensive agent, is a selective α2A-adrenoceptor agonist with Kd of 31 nM and displays 60-fold selectivity over α2B-adrenoceptors. Learn More
  42. HOKU-81

    Catalog No. A15117
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    Metabolites of tulobuterol
    HOKU-81, a new bronchodilator, is one of the metabolites of tulobuterol. Learn More
  43. Trenbolone

    Catalog No. A15266
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    Trenbolone is a steroid used by veterinarians on livestock to increase muscle growth and appetite. Learn More
  44. Urapidil

    Catalog No. A17074
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    α1 adrenoreceptor antagonist
    Urapidil is an α1 adrenoreceptor antagonist and a 5-HT1A receptor agonist. Learn More
  45. Synephrine (Oxedrine)

    Catalog No. A10882
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    Adrenergic Receptor agonist
    Synephrine (Oxedrine) is an amine compound commonly used for weight loss. Learn More
  46. Formoterol hemifumarate

    Catalog No. A11732
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    Formoterol is a long-acting β2-agonist used in the management of asthma and/or chronic obstructive pulmonary disease (COPD). Learn More
  47. Betaxolol hydrochloride

    Catalog No. A11733
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  48. Phentolamine mesilate

    Catalog No. A11734
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    Phentolamine is a reversible nonselective alpha-adrenergic antagonist. Learn More
  49. Terazosin hydrochloride

    Catalog No. A11740
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    Terazosin is a selective alpha 1 antagonist used for treatment of symptoms of an enlarged prostate (BPH). Learn More
  50. Detomidine hydrochloride

    Catalog No. A10298
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    Adrenergic Receptor agonist
    Detomidine is a sedative with analgesic properties. α2-adrenergic agonists produce dose-dependent sedative and analgesic effects, mediatated by activation of α2 catecholamine receptors, thus inducing a negative feedback response, reducing production of excitatory neurotransmitters. Learn More

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