Adrenergic Receptors

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  1. OPC-28326

    Catalog No. A12762
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    α2-adrenergic receptor angatonist
    OPC-28326 is a selective peripheral vasodilator and an angatonist of α2-adrenergic receptor, with Ki of 2040, 285, and 55?nM for α2A-, α2B- and α2C-adrenoceptors, respectively. Learn More
  2. Norepinephrine

    Catalog No. A11306
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    β1-selective adrenergic receptor agonist
    Norepinephrine (Levarterenol; L-Noradrenaline) is a β1-selective adrenergic receptor agonist with EC50 of 5.37 μM. Learn More
  3. Ancarolol

    Catalog No. A12534
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    beta-adrenergic blocking agent
    Ancarolol is a beta-adrenergic blocking agent. Learn More
  4. AGN 192836

    Catalog No. A13013
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    α2 adrenergic agonist
    AGN 192836 is a potent and selective α2 adrenergic agonist with EC50s of 8.7, 41 and 6.6 nM for α2A, α2B and α2C receptor, respectively. Learn More
  5. β3-AR agonist 1

    Catalog No. A12777
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    β3-adrenergic receptor agonist
    β3-AR agonist 1 (compound 15) is a highly potent, selective, and orally available β3-adrenergic receptor (β3-AR) agonist (EC50=18 nM), being inactive to β1-, β2-, and α1A-AR (β1/β3, β2/β3, and α1A/β3>556-fold). Learn More
  6. Asenapine

    Catalog No. A18010
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    adrenergic receptor inhibitor
    Asenapine(Org 5222) inhibits adrenergic receptor (α1, α2A, α2B, α2C) with Ki of 0.25-1.2 nM and also inhibits 5-HT receptor (1A, 1B, 2A, 2B, 2C, 5A, 6, 7) with Ki of 0.03-4.0 nM. Learn More
  7. Norepinephrine hydrochloride

    Catalog No. A21605
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    β1-selective adrenergic receptor agonist
    Norepinephrine hydrochloride (Levarterenol hydrochloride; L-Noradrenaline hydrochloride) is a β1-selective adrenergic receptor agonist with EC50 of 5.37 μM. Learn More
  8. Synephrine (Oxedrine)

    Catalog No. A10882
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    Adrenergic Receptor agonist
    Synephrine (Oxedrine) is an amine compound commonly used for weight loss. Learn More
  9. Salbutamol sulfate (Albuterol)

    Catalog No. A10819
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    Adrenergic Receptor agonist
    Salbutamol sulfate (Albuterol) is a short-acting β2-adrenergic receptor agonist used for the relief of bronchospasm in conditions such as asthma and chronic obstructive pulmonary disease. Learn More
  10. Naftopidil 2HCl

    Catalog No. A10619
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    5-HT1A and α1-adrenergic receptor antagonist
    Naftopidil 2HCl is a selective 5-HT1A and α1-adrenergic receptor antagonist with IC50 of 0.1 μM and 0.2 μM, respectively. Learn More
  11. Silodosin (Rapaflo)

    Catalog No. A10843
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    α1-adrenoceptor antagonist
    Silodosin(Rapaflo) is an α1-adrenoceptor antagonist with high uroselectivity. It causes practically no orthostatic hypotension (in contrast to other α1 blockers). Learn More
  12. Alfuzosin HCl

    Catalog No. A10052
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    Alfuzosin (provided as the hydrochloride salt) is an α1 receptor antagonist used to treat benign prostatic hyperplasia (BPH). It works by relaxing the muscles in the prostate and bladder neck, making it easier to urinate. Learn More
  13. Bisoprolol fumarate

    Catalog No. A10149
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    β1 adrenergic receptor blocker
    Bisoprolol is a drug belonging to the group of beta blockers, a class of drugs used primarily in cardiovascular diseases. More specifically, it is a selective type β1 adrenergic receptor blocker. Learn More
  14. Phenylephrine HCl

    Catalog No. A11666
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    α1-adrenergic receptor agonist
    Phenylephrine is a selective α1-adrenergic receptor agonist used primarily as a decongestant, as an agent to dilate the pupil, and to increase blood pressure. Learn More
  15. DL-Adrenaline

    Catalog No. A11668
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    DL-Adrenaline is a hormone and a neurotransmitter secreted by the medulla of the adrenal glands. DL-Adrenaline is found in small amounts in the body and is essential for maintaining cardiovascular homeostasis because of its ability to divert blood to tissues under stress. Learn More
  16. Isoprenaline HCl

    Catalog No. A10484
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    β adrenoceptor agonist
    Isoprenaline or isoproterenol is a non-selective beta-adrenergic agonist and structurally similar to adrenaline. Learn More
  17. Apalutamide (ARN-509)

    Catalog No. A11923
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    Androgen Receptor inhibitor
    ARN-509 is an androgen receptor antagonist with potential antineoplastic activity. ARN-509 binds to AR in target tissues thereby preventing androgen-induced receptor activation and facilitating the formation of inactive complexes that cannot be translocated to the nucleus. This prevents binding to and transcription of AR-responsive genes. Learn More
  18. Metoprolol tartrate

    Catalog No. A11713
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    Beta1 receptor blocker
    Metoprolol is a selective β1 receptor blocker used in treatment of several diseases of the cardiovascular system, especially hypertension. Learn More
  19. Betaxolol

    Catalog No. A11721
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    Betaxolol is a selective beta1 receptor blocker used in the treatment of hypertension and glaucoma. Being selective for beta1 receptors, it typically has fewer systemic side effects than non-selective beta-blockers, for example, not causing bronchospasm (mediated by beta2 receptors) as timolol may. Betaxolol also shows greater affininty for beta1 receptors than metoprolol. Learn More
  20. Formoterol hemifumarate

    Catalog No. A11732
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    Formoterol is a long-acting β2-agonist used in the management of asthma and/or chronic obstructive pulmonary disease (COPD). Learn More
  21. Betaxolol hydrochloride

    Catalog No. A11733
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    Betaxolol Hydrochloride is a selective beta1 adrenergic receptor blocker used in the treatment of hypertension and glaucoma. Learn More
  22. Phentolamine mesilate

    Catalog No. A11734
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    Phentolamine is a reversible nonselective alpha-adrenergic antagonist. Learn More
  23. Terazosin hydrochloride

    Catalog No. A11740
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    Terazosin is a selective alpha 1 antagonist used for treatment of symptoms of an enlarged prostate (BPH). Learn More
  24. Detomidine hydrochloride

    Catalog No. A10298
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    Adrenergic Receptor agonist
    Detomidine is a sedative with analgesic properties. α2-adrenergic agonists produce dose-dependent sedative and analgesic effects, mediatated by activation of α2 catecholamine receptors, thus inducing a negative feedback response, reducing production of excitatory neurotransmitters. Learn More
  25. Asenapine maleate

    Catalog No. A10091
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    H1 antagonist
    Asenapine shows high affinity (pKi) for numerous receptors, including the serotonin 5-HT1A (8.6), 5-HT1B (8.4), 5-HT2A (10.2), 5-HT2B (9.8), 5-HT2C (10.5), 5-HT5A (8.8), 5-HT6 (9.5), and 5-HT7 (9.9) receptors, the adrenergic α1 (8.9), α2A (8.9), α2B (9.5), and α2C (8.9) receptors, the dopamine D1 (8.9), D2 (8.9), D3 (9.4), and D4 (9.0) receptors, and the histamine H1 (9.0) and H2 (8.2) receptors. Learn More
  26. Clonidine hydrochloride

    Catalog No. A10232
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    Alpha adrenergic agonist
    Clonidine is classified as a centrally acting alpha adrenergic agonist.Clonidine acts centrally as an imidazoline receptor agonist. Learn More
  27. Dehydroepiandrosterone

    Catalog No. A10296
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    Dehydroepiandrosterone is an important endogenous steroid hormone. Learn More
  28. Dobutamine hydrochloride

    Catalog No. A10325
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    Adrenoceptors agonist
    Dobutamine is a direct-acting agent whose primary activity results from stimulation of the β1-adrenoceptors of the heart, increasing contractility and cardiac output. Learn More
  29. Doxazosin mesylate

    Catalog No. A10334
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    Doxazosin mesylate, a quinazoline compound, is an α1-selective alpha blocker used to treat high blood pressure and urinary retention associated with benign prostatic hyperplasia (BPH). Learn More
  30. Metroprolol succinate

    Catalog No. A11229
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    Metoprolol succinate is a cardioselective β-adrenergic receptor blocker with IC50 of 42 ng/mL. Learn More
  31. Prazosin HCl

    Catalog No. A11914
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    Prazosin HCl is an α1 and α2B-adrenoceptor antagonist. Also a potent antagonist at the melatonin MT3 receptor (Ki = 10.2 nM). Learn More
  32. Procaterol HCl

    Catalog No. A11905
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    Procaterol is a short-acting β2-adrenergic receptor agonist with Kp of 8 nM, used for the treatment of asthma Learn More
  33. Rilmenidine

    Catalog No. A10794
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    α2 adrenergic agonist
    Rilmenidine is a second-generation imidazoline-α2 adrenergic agonist. Learn More
  34. Naftopidil (Flivas)

    Catalog No. A10618
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    Naftopidil (Flivas) is a selective α1-adrenergic receptor antagonist or alpha blocker with a Ki of 58.3 nM. Learn More
  35. Nebivolol HCl

    Catalog No. A10630
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    Nebivolol hydrochloride is t a highly selective antagonist of the β1-adrenoceptor (Ki = 0.88 nM, β2-adrenoceptor Ki = 48 nM). Learn More
  36. Phenoxybenzamine hydrochloride

    Catalog No. A10719
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    α-adrenergic (AR) antagonist/CaM inhibitor
    Phenoxybenzamine is a cell-permeable, non-specific, irreversible α-adrenergic (AR) antagonist that also acts as an CaM inhibitor. Learn More
  37. Carvedilol

    Catalog No. A11843
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    β2-adrenergic receptor
    Carvedilol is a β1- and β2-adrenergic receptor (AR) agonist with antioxidant properties. Learn More
  38. Salmeterol

    Catalog No. A11788
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    beta2-adrenergic receptor agonist
    Salmeterol is a long-acting beta2-adrenergic receptor agonist Learn More
  39. Adrenalone HCl

    Catalog No. A11807
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    adrenergic agonist
    Adrenalone is an adrenergic agonist used as a topical vasoconstrictor and hemostatic, mainly acts on alpha-1 adrenergic receptors. Learn More
  40. Ivabradine HCl (Procoralan)

    Catalog No. A11868
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    Ivabradine Hydrochloride, also known as S-16257, is the hydrochloride salt preparation of Ivabradine, a bradycardic agent. Learn More
  41. Tamsulosin

    Catalog No. A12657
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    alpha-1A/alpha-1B-adrenoceptor antagonist
    Tamsulosin is an alpha1a-selective alpha blocker used in the symptomatic treatment of benign prostatic hyperplasia (BPH). Learn More
  42. Arformoterol tartrate

    Catalog No. A12795
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    beta2-adrenergic agonist
    Arformoterol tartrate is a beta2-adrenergic agonist Learn More
  43. Mirabegron

    Catalog No. A12861
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    β3 adrenergic receptor activator
    Mirabegron is a potent bladder relaxant and reagent for diabetes remedy. Learn More
  44. Oxymetazoline hydrochloride

    Catalog No. A10686
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    alpha-1 adrenergic agonist
    Oxymetazoline is a selective alpha-1 agonist and partial alpha-2 agonist topical decongestant, used in the form of Oxymetazoline hydrochloride. Learn More
  45. Tetrahydrozoline Hydrochloride

    Catalog No. A13080
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    Adrenergic Receptor agonist
    Tetrahydrozoline Hydrochloride is an alpha agonist which causes constriction of conjunctival blood vessels. Learn More
  46. ICI 118,551 hydrochloride

    Catalog No. A13225
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    β2 adrenergic antagonist
    ICI 118551 hydrochloride is a selective β2 adrenergic antagonist. Learn More
  47. Maprotiline hydrochloride

    Catalog No. A10555
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    noradrenalin re-uptake inhibitor
    Maprotiline hydrochloride is a selective noradrenalin re-uptake inhibitor. Learn More
  48. Bisoprolol

    Catalog No. A13406
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    Bisoprolol is a cardioselective β1-adrenergic blocking agent used for secondary prevention of myocardial infarction (MI), heart failure, angina pectoris and mild to moderate hypertension. Learn More
  49. Clenbuterol hydrochloride

    Catalog No. A13407
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    Clenbuterol Hydrochloride is a sympathomimetic β2-adrenoceptor agonist that has been used as a bronchodilator in the treatment of pulmonary diseases such as asthma. At higher doses, clenbuterol acts as an anabolic steroid, favoring skeletal muscle protein synthesis at the expense of fat deposition. Learn More
  50. Octopamine hydrochloride

    Catalog No. A13419
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    Octopamine hydrochloride is an invertebrate biogenic amine neurotransmitter, related to noradrenalin, that is an adrenoceptor agonist. Learn More

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