Total item
Cart Subtotal
$0.00 Adrenergic Receptors
-
OPC-28326
Catalog No. A12762 α2-adrenergic receptor angatonistOPC-28326 is a selective peripheral vasodilator and an angatonist of α2-adrenergic receptor, with Ki of 2040, 285, and 55?nM for α2A-, α2B- and α2C-adrenoceptors, respectively. Learn More -
Norepinephrine
Catalog No. A11306 β1-selective adrenergic receptor agonistNorepinephrine (Levarterenol; L-Noradrenaline) is a β1-selective adrenergic receptor agonist with EC50 of 5.37 μM. Learn More -
Ancarolol
Catalog No. A12534 beta-adrenergic blocking agentAncarolol is a beta-adrenergic blocking agent. Learn More -
AGN 192836
Catalog No. A13013 α2 adrenergic agonistAGN 192836 is a potent and selective α2 adrenergic agonist with EC50s of 8.7, 41 and 6.6 nM for α2A, α2B and α2C receptor, respectively. Learn More -
β3-AR agonist 1
Catalog No. A12777 β3-adrenergic receptor agonistβ3-AR agonist 1 (compound 15) is a highly potent, selective, and orally available β3-adrenergic receptor (β3-AR) agonist (EC50=18 nM), being inactive to β1-, β2-, and α1A-AR (β1/β3, β2/β3, and α1A/β3>556-fold). Learn More -
Asenapine
Catalog No. A18010 adrenergic receptor inhibitorAsenapine(Org 5222) inhibits adrenergic receptor (α1, α2A, α2B, α2C) with Ki of 0.25-1.2 nM and also inhibits 5-HT receptor (1A, 1B, 2A, 2B, 2C, 5A, 6, 7) with Ki of 0.03-4.0 nM. Learn More -
Norepinephrine hydrochloride
Catalog No. A21605 β1-selective adrenergic receptor agonistNorepinephrine hydrochloride (Levarterenol hydrochloride; L-Noradrenaline hydrochloride) is a β1-selective adrenergic receptor agonist with EC50 of 5.37 μM. Learn More -
Synephrine (Oxedrine)
Catalog No. A10882 Adrenergic Receptor agonistSynephrine (Oxedrine) is an amine compound commonly used for weight loss. Learn More -
Salbutamol sulfate (Albuterol)
Catalog No. A10819 Adrenergic Receptor agonistSalbutamol sulfate (Albuterol) is a short-acting β2-adrenergic receptor agonist used for the relief of bronchospasm in conditions such as asthma and chronic obstructive pulmonary disease. Learn More -
Naftopidil 2HCl
Catalog No. A10619 5-HT1A and α1-adrenergic receptor antagonistNaftopidil 2HCl is a selective 5-HT1A and α1-adrenergic receptor antagonist with IC50 of 0.1 μM and 0.2 μM, respectively. Learn More -
Silodosin (Rapaflo)
Catalog No. A10843 α1-adrenoceptor antagonistSilodosin(Rapaflo) is an α1-adrenoceptor antagonist with high uroselectivity. It causes practically no orthostatic hypotension (in contrast to other α1 blockers). Learn More -
Alfuzosin HCl
Catalog No. A10052 Alfuzosin (provided as the hydrochloride salt) is an α1 receptor antagonist used to treat benign prostatic hyperplasia (BPH). It works by relaxing the muscles in the prostate and bladder neck, making it easier to urinate. Learn More -
Bisoprolol fumarate
Catalog No. A10149 β1 adrenergic receptor blockerBisoprolol is a drug belonging to the group of beta blockers, a class of drugs used primarily in cardiovascular diseases. More specifically, it is a selective type β1 adrenergic receptor blocker. Learn More -
Phenylephrine HCl
Catalog No. A11666 α1-adrenergic receptor agonistPhenylephrine is a selective α1-adrenergic receptor agonist used primarily as a decongestant, as an agent to dilate the pupil, and to increase blood pressure. Learn More -
DL-Adrenaline
Catalog No. A11668 DL-Adrenaline is a hormone and a neurotransmitter secreted by the medulla of the adrenal glands. DL-Adrenaline is found in small amounts in the body and is essential for maintaining cardiovascular homeostasis because of its ability to divert blood to tissues under stress. Learn More -
Isoprenaline HCl
Catalog No. A10484 β adrenoceptor agonistIsoprenaline or isoproterenol is a non-selective beta-adrenergic agonist and structurally similar to adrenaline. Learn More -
Apalutamide (ARN-509)
Catalog No. A11923 Androgen Receptor inhibitorARN-509 is an androgen receptor antagonist with potential antineoplastic activity. ARN-509 binds to AR in target tissues thereby preventing androgen-induced receptor activation and facilitating the formation of inactive complexes that cannot be translocated to the nucleus. This prevents binding to and transcription of AR-responsive genes. Learn More -
Metoprolol tartrate
Catalog No. A11713 Beta1 receptor blockerMetoprolol is a selective β1 receptor blocker used in treatment of several diseases of the cardiovascular system, especially hypertension. Learn More -
Betaxolol
Catalog No. A11721 Betaxolol is a selective beta1 receptor blocker used in the treatment of hypertension and glaucoma. Being selective for beta1 receptors, it typically has fewer systemic side effects than non-selective beta-blockers, for example, not causing bronchospasm (mediated by beta2 receptors) as timolol may. Betaxolol also shows greater affininty for beta1 receptors than metoprolol. Learn More -
Formoterol hemifumarate
Catalog No. A11732 Formoterol is a long-acting β2-agonist used in the management of asthma and/or chronic obstructive pulmonary disease (COPD). Learn More -
Betaxolol hydrochloride
Catalog No. A11733 Betaxolol Hydrochloride is a selective beta1 adrenergic receptor blocker used in the treatment of hypertension and glaucoma. Learn More -
Phentolamine mesilate
Catalog No. A11734 Phentolamine is a reversible nonselective alpha-adrenergic antagonist. Learn More -
Terazosin hydrochloride
Catalog No. A11740 Terazosin is a selective alpha 1 antagonist used for treatment of symptoms of an enlarged prostate (BPH). Learn More -
Detomidine hydrochloride
Catalog No. A10298 Adrenergic Receptor agonistDetomidine is a sedative with analgesic properties. α2-adrenergic agonists produce dose-dependent sedative and analgesic effects, mediatated by activation of α2 catecholamine receptors, thus inducing a negative feedback response, reducing production of excitatory neurotransmitters. Learn More -
Asenapine maleate
Catalog No. A10091 H1 antagonistAsenapine shows high affinity (pKi) for numerous receptors, including the serotonin 5-HT1A (8.6), 5-HT1B (8.4), 5-HT2A (10.2), 5-HT2B (9.8), 5-HT2C (10.5), 5-HT5A (8.8), 5-HT6 (9.5), and 5-HT7 (9.9) receptors, the adrenergic α1 (8.9), α2A (8.9), α2B (9.5), and α2C (8.9) receptors, the dopamine D1 (8.9), D2 (8.9), D3 (9.4), and D4 (9.0) receptors, and the histamine H1 (9.0) and H2 (8.2) receptors. Learn More -
Clonidine hydrochloride
Catalog No. A10232 Alpha adrenergic agonistClonidine is classified as a centrally acting alpha adrenergic agonist.Clonidine acts centrally as an imidazoline receptor agonist. Learn More -
Dehydroepiandrosterone
Catalog No. A10296 Dehydroepiandrosterone is an important endogenous steroid hormone. Learn More -
Dobutamine hydrochloride
Catalog No. A10325 Adrenoceptors agonistDobutamine is a direct-acting agent whose primary activity results from stimulation of the β1-adrenoceptors of the heart, increasing contractility and cardiac output. Learn More -
Doxazosin mesylate
Catalog No. A10334 Doxazosin mesylate, a quinazoline compound, is an α1-selective alpha blocker used to treat high blood pressure and urinary retention associated with benign prostatic hyperplasia (BPH). Learn More -
Metroprolol succinate
Catalog No. A11229 Metoprolol succinate is a cardioselective β-adrenergic receptor blocker with IC50 of 42 ng/mL. Learn More -
Prazosin HCl
Catalog No. A11914 Prazosin HCl is an α1 and α2B-adrenoceptor antagonist. Also a potent antagonist at the melatonin MT3 receptor (Ki = 10.2 nM). Learn More -
Procaterol HCl
Catalog No. A11905 Procaterol is a short-acting β2-adrenergic receptor agonist with Kp of 8 nM, used for the treatment of asthma Learn More -
Rilmenidine
Catalog No. A10794 α2 adrenergic agonistRilmenidine is a second-generation imidazoline-α2 adrenergic agonist. Learn More -
Naftopidil (Flivas)
Catalog No. A10618 Naftopidil (Flivas) is a selective α1-adrenergic receptor antagonist or alpha blocker with a Ki of 58.3 nM. Learn More -
Nebivolol HCl
Catalog No. A10630 Nebivolol hydrochloride is t a highly selective antagonist of the β1-adrenoceptor (Ki = 0.88 nM, β2-adrenoceptor Ki = 48 nM). Learn More -
Phenoxybenzamine hydrochloride
Catalog No. A10719 α-adrenergic (AR) antagonist/CaM inhibitorPhenoxybenzamine is a cell-permeable, non-specific, irreversible α-adrenergic (AR) antagonist that also acts as an CaM inhibitor. Learn More -
Carvedilol
Catalog No. A11843 β2-adrenergic receptorCarvedilol is a β1- and β2-adrenergic receptor (AR) agonist with antioxidant properties. Learn More -
Salmeterol
Catalog No. A11788 beta2-adrenergic receptor agonistSalmeterol is a long-acting beta2-adrenergic receptor agonist Learn More -
Adrenalone HCl
Catalog No. A11807 adrenergic agonistAdrenalone is an adrenergic agonist used as a topical vasoconstrictor and hemostatic, mainly acts on alpha-1 adrenergic receptors. Learn More -
Ivabradine HCl (Procoralan)
Catalog No. A11868 Ivabradine Hydrochloride, also known as S-16257, is the hydrochloride salt preparation of Ivabradine, a bradycardic agent. Learn More -
Tamsulosin
Catalog No. A12657 alpha-1A/alpha-1B-adrenoceptor antagonistTamsulosin is an alpha1a-selective alpha blocker used in the symptomatic treatment of benign prostatic hyperplasia (BPH). Learn More -
Arformoterol tartrate
Catalog No. A12795 beta2-adrenergic agonistArformoterol tartrate is a beta2-adrenergic agonist Learn More -
Mirabegron
Catalog No. A12861 β3 adrenergic receptor activatorMirabegron is a potent bladder relaxant and reagent for diabetes remedy. Learn More -
Oxymetazoline hydrochloride
Catalog No. A10686 alpha-1 adrenergic agonistOxymetazoline is a selective alpha-1 agonist and partial alpha-2 agonist topical decongestant, used in the form of Oxymetazoline hydrochloride. Learn More -
Tetrahydrozoline Hydrochloride
Catalog No. A13080 Adrenergic Receptor agonistTetrahydrozoline Hydrochloride is an alpha agonist which causes constriction of conjunctival blood vessels. Learn More -
ICI 118,551 hydrochloride
Catalog No. A13225 β2 adrenergic antagonistICI 118551 hydrochloride is a selective β2 adrenergic antagonist. Learn More -
Maprotiline hydrochloride
Catalog No. A10555 noradrenalin re-uptake inhibitorMaprotiline hydrochloride is a selective noradrenalin re-uptake inhibitor. Learn More -
Bisoprolol
Catalog No. A13406 Bisoprolol is a cardioselective β1-adrenergic blocking agent used for secondary prevention of myocardial infarction (MI), heart failure, angina pectoris and mild to moderate hypertension. Learn More -
Clenbuterol hydrochloride
Catalog No. A13407 Clenbuterol Hydrochloride is a sympathomimetic β2-adrenoceptor agonist that has been used as a bronchodilator in the treatment of pulmonary diseases such as asthma. At higher doses, clenbuterol acts as an anabolic steroid, favoring skeletal muscle protein synthesis at the expense of fat deposition. Learn More -
Octopamine hydrochloride
Catalog No. A13419 Octopamine hydrochloride is an invertebrate biogenic amine neurotransmitter, related to noradrenalin, that is an adrenoceptor agonist. Learn More
FILTER BY:
Shopping Options
- Actions
-
- Inhibitor (7)
- Agonist (45)
- Antagonist (28)
- Activator (1)
- Blocker (9)
Adooq Quality Guarantee
We promise all products perform as described.