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$0.00 Estrogen Receptors
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4-Hydroxytamoxifen
Catalog No. A20955 estrogen receptor modulator4-Hydroxytamoxifen is a selective estrogen receptor modulator (SERM). Learn More -
Tamoxifen Citrate
Catalog No. A10885 Estrogen receptor antagonistTamoxifen Citrateis a selective and potent inhibitor of mammalian sterol isomerase. Learn More -
Elacestrant
Catalog No. A12244 Estrogen receptor degraderElacestrant (RAD1901) is an orally available selective estrogen receptor degrader (SERD) with IC50s of 48 and 870 nM for ERα and ERβ, respectively. Learn More -
Tamoxifen
Catalog No. A16738 selective estrogen receptor modulator (SERM)Tamoxifen (ICI 47699) is a selective estrogen receptor modulator (SERM) which blocks estrogen action in breast cells and can activate estrogen activity in other cells, such as bone, liver, and uterine cells. Learn More -
Estetrol
Catalog No. A21291 nuclear estrogen receptor modulatorEstetrol, a natural estrogen synthesized exclusively during pregnancy by the human fetal liver, is a selective nuclear estrogen receptor modulator. Learn More -
GDC-0927 Racemate
Catalog No. A21507 estrogen receptor degraderGDC-0927 Racemate (SRN-927 Racemate) is a degrader of estrogen receptor, potently inhibits ER-α activity, with an IC50 of 0.2 nM, and is used in the research of ER-related diseases. Learn More -
Fulvestrant R enantiomer
Catalog No. A21545 estrogen receptor antagonistFulvestrant R enantiomer (ICI 182780 R enantiomer; ZD 9238 R enantiomer; ZM 182780 R enantiomer) is the less active R enantiomer of Fulvestrant. Fulvestrant is a potent estrogen receptor antagonist with an IC50 of 9.4 nM. Learn More -
Pipendoxifene hydrochloride
Catalog No. A21623 estrogen receptor modulatorsPipendoxifene hydrochloride is a selective estrogen receptor modulators (SERMs). Learn More -
H3B-6545 Hydrochloride
Catalog No. A21629 estrogen receptor covalent antagonistH3B-6545 Hydrochloride is an oral, selective estrogen receptor covalent antagonist (SERCA). Learn More -
AZD9496 maleate
Catalog No. A21726 estrogen receptor (ERα) antagonistAZD9496 maleate is a potent and selective estrogen receptor (ERα) antagonist with IC50 of 0.28 nM. AZD9496 maleate is an orally bioavailable selective oestrogen receptor degrader (SERD). Learn More -
Enclomiphene citrate
Catalog No. A21830 oestrogen receptor antagonistEnclomiphene citrate is a potent and orally active oestrogen receptor antagonist, with antioestrogenic property. Learn More -
AZD9496
Catalog No. A15822 estrogen receptor downregulator and antagonistAZD9496 is a potent and orally bioavailable selective estrogen receptor downregulator and antagonist. Learn More -
Toremifene
Catalog No. A15265 Estrogen receptor modulatorToremifene is a second-generation selective estrogen-receptor modulator (SERM) in development for the prevention of osteoporosis. Learn More -
(E/Z)-4-hydroxy Tamoxifen
Catalog No. A12532 Estrogen receptor antagonist(E/Z)-4-hydroxy Tamoxifen is the active metabolite of tamoxifen and a selective estrogen receptor (ER) modulator that is widely used in the therapeutic and chemopreventive treatment of breast cancer. Learn More -
RAD1901 HCl salt
Catalog No. A15990 SERD/SERMRAD1901 is an orally available, selective estrogen receptor degrader (SERD) and selective estrogen receptor modulator (SERM), with potential antineoplastic and estrogen-like activities. Learn More -
GDC-0810 (Brilanestrant)
Catalog No. A15958 Estrogen receptor degraderBrilanestrant (GDC-0810, ARN-810） is a potent ER-α binder (ER-α, IC50 = 6.1 nM; ER-β, IC50 = 8.8 nM), a full transcriptional antagonist with no agonism and displays good potency and efficacy in ER-α degradation (EC50 = 0.7 nM) and MCF-7 breast cancer cell viability (IC50 = 2.5 nM) assays with good selectivity over other nuclear hormone receptors. Learn More -
Endoxifen E-isomer hydrochloride
Catalog No. A16343 Endoxifen (E-isomer hydrochloride) is a tamoxifen metabolite and potent Selective Estrogen Response Modifier (SERM). Learn More -
GSK4716
Catalog No. A16956 ERRβ & ERRγ AgonistGSK4716 is an Estrogen-related receptors ERRβ and ERRγ agonist with minimal activity for ERRα, ERα and ERβ Learn More -
(R)-Equol
Catalog No. A16986 Estrogen receptor agonist(R)-Equol is an agonist of both ERα and ERβ with Kis of 27.4 and 15.4 nM, respectively. Learn More -
Lasofoxifene Tartrate
Catalog No. A18097 selective Estrogen receptor modulatorLasofoxifene tartrate is a third-generation selective estrogen receptor modulator. Learn More -
H3B-6545
Catalog No. A20100 Estrogen receptor antagonistH3B-6545 is an oral, selective estrogen receptor covalent antagonist (SERCA). Learn More -
PROTAC ERRα ligand 2
Catalog No. A18939 ERRα inverse agonistPROTAC ERRα ligand 2 is an estrogen-related receptor α (ERRα) inverse agonist with an IC50 of 5.67 nM. PROTAC ERRα ligand 2 (IC50=5.67 nM) displays a ~11-fold improved potency than XCT790 (IC50=61.3 nM). Learn More -
PROTAC ERRα Degrader-1
Catalog No. A18910 ERRα DegraderPROTAC ERRα Degrader-1 comprises a MDM2 ligand binding group, a linker and an estrogen-related receptor alpha (ERRa) binding group. PROTAC ERRα Degrader-1 is an estrogen-related receptor alpha (ERRa) degrader. Learn More -
PROTAC ER Degrader-3
Catalog No. A18519 PROTAC ER Degrader-3 is an intermediate for synthesis of PAC. PAC, consists the ADCs linker and PROTACs, conjugated to an antibody. PAC extracts from patent WO2017201449A1, compound LP2. PAC conjugated to an antibody is a more marked estrogen receptor-alpha (ERα) degrader compared to PROTAC (without Ab). Learn More -
MK-6913
Catalog No. A12311 Estrogen receptor β agonistTetrahydrofluoroene 52 is a potent and selective estrogen receptor β agonist. Learn More -
GW9508
Catalog No. A11965 GPR40 InhibitorGW 9508 is a cell-permeable aminophenylpropanoate that acts as a potent and selective agonist for the G-protein coupled receptor (GPCR) GRP40/FFA1 receptor (EC50 ?50 nM) with reduced activity towards family members GRP120 (EC50 ?3.5 μM), GRP41/GRP43 (EC50 >50 μM), as well as a panel of eight other free fatty acid (FFA) and prostaglandin receptors. Learn More -
Fulvestrant (Faslodex)
Catalog No. A10410 Aromatase inhibitorFulvestrant is an estrogen receptor antagonist with no agonist effects, which works both by down-regulating and by degrading the estrogen receptor. Learn More -
Dienogest
Catalog No. A10308 Dienogest is an oral progestin that has antiandrogenic activity and as a result can improve androgenic symptoms. Learn More -
Kaempferol
Catalog No. A10495 ERRα and ERRγ inverse agonistKaempferol is found to inhibit bovine aorta myosin light chain kinase with a Ki of 0.3-0.5 microM and also is found to inhibit VEGF expression and in vitro angiogenesis through a novel ERK-NFκB-cMyc-p21 pathway. Learn More -
Hexestrol
Catalog No. A10451 Estrogen/progestogen Receptor agonistHexestrol is a carcinogenic synthetic estrogen that inhibits microtubule polymerization and the formation of ribbon structures. It is an inhibitor of lipid peroxidation. Learn More -
Evista (Raloxifene HCl)
Catalog No. A10375 Raloxifene is an oral selective estrogen receptor modulator (SERM) that has estrogenic actions on bone and anti-estrogenic actions on the uterus and breast. It is used in the prevention of osteoporosis in postmenopausal women. Learn More -
LY500307
Catalog No. A10550 ERβ agonistLY500307 is a potent, selective estrogen receptor beta agonist with an EC50 of 0.66 nM. Learn More -
Bazedoxifene acetate
Catalog No. A11665 Bazedoxifene is a third generation selective estrogen receptor modulator (SERM). Bazedoxifene acetate significantly prevents bone mass loss at 20 mg/day in healthy postmenopausal women with normal or low bone mineral density. Learn More -
Clomifene citrate
Catalog No. A10230 Clomifene inhibits estrogen receptors in hypothalamus, inhibiting negative feedback of estrogen on gonadotropin release, leading to up-regulation of the hypothalamic-Cpituitary-Cadrenal axis. Learn More -
Drospirenone
Catalog No. A10336 Drospirenone is a synthetic hormone used in birth control pills. Learn More -
Endoxifen
Catalog No. A12639 Estrogen receptor antagonistEndoxifen is a secondary metabolite of tamoxifen. It is a primary metabolite responsible for the effectiveness of tamoxifen in ER-positive breast cancer. Learn More -
Mifepristone (Mifeprex)
Catalog No. A10591 Mifepristone, an antioxidant and glucocorticoid receptor antagonist, demonstrates the ability to suppress activation of NFκB, a nuclear transcription factor that affects the expression of various adhesion molecules and several inflammatory genes. Learn More -
Liquiritigenin
Catalog No. A12083 Liquiritigenin is a plant-derived highly selective estrogen receptor ?? agonist Learn More -
Acolbifene (EM 652, SCH57068)
Catalog No. A12771 estrogen receptor modulatoracolbifene is a substance being studied in the prevention of breast cancer in women at high risk of breast cancer. Acolbifene hydrochloride binds to estrogen receptors in the body and blocks the effects of estrogen in the breast. It is a type of selective estrogen receptor modulator (SERM). Learn More -
Zearalenone
Catalog No. A13740 Zearalenone is a phytoestrogenic mycotoxin usually produced by Fusarium species, is shown to be a cytotoxic compound, but alos binds to the estrogen receptor (ER) (IC50 values are 166 and 240 nM for ERβ and ERα respectively) and was found to stimulate the transcriptional activity of both subtypes at concentrations between 1 - 10 nM. Learn More -
Arzoxifene HCl
Catalog No. A13292 Arzoxifene HCl is the hydrochloride salt of arzoxifene, a synthetic aromatic derivative with anti-estrogenic properties. Arzoxifene binds to estrogen receptors as a mixed estrogen agonist/antagonist. Learn More -
XCT 790
Catalog No. A13299 ERRα antagonist/inverse agonistXCT 790 is a potent and specific inverse agonist of ERRα. Learn More -
Ospemifene
Catalog No. A14261 estrogen receptor modulatorOspemifene is a non-hormonal selective estrogen receptor modulator (SERM). Learn More -
IRL-2500
Catalog No. A13638 ETBR antagonistIRL-2500 is a potent, selective ETBR antagonist. It shows some selectivity for ETB receptors (IC50 values are 1.3 and 94 nM for ETB and ETA receptors respectively). Learn More -
Bazedoxifene
Catalog No. A15019 Estrogen modulatorBazedoxifene is a third generation selective modulator of estrogen receptor. Learn More -
DY131
Catalog No. A15071 ERRβ and ERRγ agonistDY131(GSK 9089) is a novel selective agonist of ERRα and ERRβ. Learn More -
TAK-875 (Fasiglifam)
Catalog No. A11018 GPR agonistTAK-875 is a potent, selective, and orally bioavailable GPR40 agonist. Learn More
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