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Pyr6
Catalog No. A21927 TRPC3 inhibitorPyr6 is a selective inhibitor of TRPC3 with IC50 of 0.49 uM(Ca2+ influx inhibition in thapsigargin depleted native RBL-2H3 cells). Learn More -
D-3263
Catalog No. A20935 TRPM8 agonistD-3263 is an agonist of transient receptor potential melastatin member 8 (TRPM8) with potential antineoplastic activity. Learn More -
SN 2
Catalog No. A20839 TRPML3 ion channel activatorSN 2 is a novel and potent activator of TRPML3 ion channel with EC50 of 1.8??0.13 μM. Learn More -
SAR7334
Catalog No. A20836 TRPC6 inhibitorSAR7334 is a potent and specific TRPC6 inhibitor, inhibiting TRPC6 currents with IC50 of 7.9 nM. Learn More -
AMG2850
Catalog No. A19445 TRPM8 antagonistAMG2850 is a potent, orally bioavailable and selective transient receptor potential melastatin 8 (TRPM8) antagonist. Learn More -
AMG-333
Catalog No. A17182 -
PF-4840154
Catalog No. A13996 TrpA1 channel agonistPF-4840154 is a non-electrophilic reference agonist of the TrpA1 channel. The TRPA1 channel is considered an attractive pain target based on the fact that TRPA1 knockout mice showed near complete attenuation of pain behaviors in some pre-clinical development models. Learn More -
Pico145
Catalog No. A13344 TRPC1/4/5 channels inhibitorPico145 is a remarkable inhibitor of TRPC1/4/5 channels, inhibits (?)-englerin A-activated TRPC4/TRPC5 channels, with IC50s of 0.349 and 1.3 nM in cells, and shows no effect on TRPC3, TRPC6, TRPV1, TRPV4, TRPA1, TRPM2, TRPM8. Learn More -
TRPC6-IN-1
Catalog No. A12309 TRPC6 inhibitorTRPC6-IN-1 is a Transient Receptor Potential Canonical 6 Channel (TRPC6) inhibitor, with an EC50 of 4.66 μM. Learn More -
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SAR-7334 HCl
Catalog No. A17237 TRPC6 inhibitorSAR7334 is a novel, highly potent and bioavailable inhibitor of TRPC6 channels that opens new opportunities for the investigation of TRPC channel function in vivo. SAR7334 inhibited TRPC6, TRPC3 and TRPC7-mediated Ca(2+) influx into cells with IC50 s of 9.5, 282 and 226 nM, whereas TRPC4 and TRPC5-mediated Ca(2+) entry was not affected. Learn More -
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WS 12
Catalog No. A17046 TRPM8 AgonistWS-12 is a potent TRPM8 agonist that acts as a cooling agent (EC50 = 193 nM). Learn More -
WS 3
Catalog No. A17047 TRPM8 agonistWS 3 is TRPM8 receptors agonist (EC50 = 3.7 μM) and cooling agent. Learn More -
Evodiamine (Isoevodiamine)
Catalog No. A10376 TRP agonistEvodiamine is a chemical extracted from the Tetradium family of plants. It acts primarily as a thermogenic and stimulant. Learn More -
GsMTx4
Catalog No. A16103 GsMTX4 is a 34 amino acid peptidyl toxin isolated from the Grammostola rosea (Chilean rose) tarantula venom and belongs to the huwentoxin-1 family. Learn More -
RQ-00203078
Catalog No. A15830 TRPM8 antagonistRQ-00203078 is a highly selective, potent and orally available TRPM8 antagonist (IC50 values are 5.3 and 8.3 nM for rat and human channels respectively), exhibits >350-fold selectivity for TRPM8 over TRPV4, TRPV1 and TRPA1. Learn More -
ML204
Catalog No. A15556 TRPC4/C5 inhibitorML204 is a novel potent antagonist that selectively modulates native TRPC4/C5 ion channels. Learn More -
Cannabichromene
Catalog No. A15497 TRPA1 activatior/TRPM8 blockerCannabichromene is a major non-psychotropic phytocannabinoid that inhibits endocannabinoid inactivation and activates the transient receptor potential ankyrin-1 (TRPA1). Both endocannabinoids and TRPA1 may modulate gastrointestinal motility. Learn More -
ACA
Catalog No. A13585 ACA is a channel blocker that acts on several transient receptor potential (TRP) channels, including TRPM2, TRPM8, and TRPC6 (IC50 = 1.7, 3.8, and 2.3 uM, respectively). Learn More -
TCS 5861528
Catalog No. A14126 TRPA1 channel blockerTCS 5861528 is a TRPA1 channel blocker and an antagonizer of AITC- and 4-HNE-evoked calcium influx. Learn More -
HC-030031
Catalog No. A13278 TRPA1 inhibitorHC-030031 is a selective TRPA1 blocker, antagonizing TRPA1-mediated calcium influx induced by AITC and formalin (IC50 = 6.2 and 5.3 uM, respectively). Learn More -
Icilin
Catalog No. A13560 TRPM8 and TRPA1 activatorIcilin is a cooling agent that activates the novel cold receptors TRPM8 (CMR1) and TRPA1 (ANKTM1/TRPN1), members of the TRP ion channel family. Induces currents in CMR1-expressing HEK 293 cells (EC50 = 0.36 μM) Learn More -
Optovin
Catalog No. A12932 photoactive TRPA1 activatorOptovin is a reversible photoactive TRPA1 activator. Learn More -
A 967079
Catalog No. A12353 TRPA1 channel blockerA 967079 is a selective TRPA1 channel blocker (IC50 values are 67 and 289 nM at human and rat TRPA1 receptors respectively). Learn More
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